UY31704A - Compuesto heterociclico fusionado - Google Patents
Compuesto heterociclico fusionadoInfo
- Publication number
- UY31704A UY31704A UY0001031704A UY31704A UY31704A UY 31704 A UY31704 A UY 31704A UY 0001031704 A UY0001031704 A UY 0001031704A UY 31704 A UY31704 A UY 31704A UY 31704 A UY31704 A UY 31704A
- Authority
- UY
- Uruguay
- Prior art keywords
- fused
- compound
- heterociclic
- represented
- formula
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title 1
- 102000004022 Protein-Tyrosine Kinases Human genes 0.000 abstract 1
- 108090000412 Protein-Tyrosine Kinases Proteins 0.000 abstract 1
- 150000002391 heterocyclic compounds Chemical class 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Oncology (AREA)
- Virology (AREA)
- Communicable Diseases (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hematology (AREA)
- Vascular Medicine (AREA)
- AIDS & HIV (AREA)
- Tropical Medicine & Parasitology (AREA)
- Molecular Biology (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
La presente invención provee un compuesto heterocíclico fusionado que tiene una acción inhibidora de tirosina quinasa que está representada por la fórmula
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2008063363 | 2008-03-12 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UY31704A true UY31704A (es) | 2009-11-10 |
Family
ID=41063727
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UY0001031704A UY31704A (es) | 2008-03-12 | 2009-03-11 | Compuesto heterociclico fusionado |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20090233937A1 (es) |
| EP (1) | EP2253633A4 (es) |
| JP (1) | JPWO2009113560A1 (es) |
| AR (1) | AR070874A1 (es) |
| PE (1) | PE20091580A1 (es) |
| TW (1) | TW200944528A (es) |
| UY (1) | UY31704A (es) |
| WO (1) | WO2009113560A1 (es) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2389731C2 (ru) * | 2004-06-02 | 2010-05-20 | Такеда Фармасьютикал Компани Лимитед | Конденсированное гетероциклическое соединение |
| WO2011040212A1 (en) | 2009-10-01 | 2011-04-07 | Takeda Pharmaceutical Company Limited | Therapeutic agent for brain tumor |
| HUE024504T2 (en) | 2010-12-23 | 2016-01-28 | Sanofi Sa | Pyrimidine derivatives, a process for their preparation and their use in medicine |
| KR20130015400A (ko) | 2011-08-03 | 2013-02-14 | 삼성디스플레이 주식회사 | 헤테로고리 화합물 및 이를 포함하는 유기 전계 발광 소자 |
| KR101930848B1 (ko) | 2011-08-11 | 2018-12-20 | 삼성디스플레이 주식회사 | 헤테로고리 화합물 및 이를 포함하는 유기 전계 발광 소자 |
| KR101971198B1 (ko) | 2011-10-19 | 2019-04-23 | 삼성디스플레이 주식회사 | 헤테로시클릭 화합물, 이를 포함하는 유기 발광 소자 및 평판 표시 장치 |
| RU2712220C2 (ru) * | 2013-07-31 | 2020-01-27 | Мерк Патент Гмбх | Пиридины, пиримидины и пиразины в качестве ингибиторов тирозинкиназы брутона и их применение |
Family Cites Families (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL112249A (en) * | 1994-01-25 | 2001-11-25 | Warner Lambert Co | Pharmaceutical compositions containing di and tricyclic pyrimidine derivatives for inhibiting tyrosine kinases of the epidermal growth factor receptor family and some new such compounds |
| JP3290666B2 (ja) | 1995-06-07 | 2002-06-10 | ファイザー・インコーポレーテッド | 複素環式の縮合環ピリミジン誘導体 |
| US6395733B1 (en) * | 1995-06-07 | 2002-05-28 | Pfizer Inc | Heterocyclic ring-fused pyrimidine derivatives |
| AR004010A1 (es) | 1995-10-11 | 1998-09-30 | Glaxo Group Ltd | Compuestos heterociclicos |
| DE69718472T2 (de) | 1996-07-13 | 2003-11-06 | Glaxo Group Ltd., Greenford | Bicyclische heteroaromatische verbindungen als protein tyrosine kinase inhibitoren |
| AU3461797A (en) | 1996-07-19 | 1998-02-10 | Takeda Chemical Industries Ltd. | Fas ligand-like protein, its production and use |
| BR9713552A (pt) | 1996-11-27 | 2000-01-25 | Pfizer | Derivados de pirimidina bicìclicos condensados |
| UA71945C2 (en) * | 1999-01-27 | 2005-01-17 | Pfizer Prod Inc | Substituted bicyclic derivatives being used as anticancer agents |
| PE20011178A1 (es) | 2000-04-07 | 2001-11-19 | Takeda Chemical Industries Ltd | Compuestos heterociclicos y su produccion |
| WO2001098277A2 (en) | 2000-06-22 | 2001-12-27 | Pfizer Products Inc. | Substituted bicyclic derivatives for the treatment of abnormal cell growth |
| AU7307101A (en) | 2000-06-30 | 2002-01-14 | Glaxo Group Ltd | Quinazoline ditosylate salt compounds |
| WO2003031442A1 (en) | 2001-10-05 | 2003-04-17 | Takeda Chemical Industries, Ltd. | Heterocyclic compounds, oxazole derivatives, process for preparation of the same and use thereof |
| HRP20040530A2 (en) | 2001-12-12 | 2004-10-31 | Pfizer Prod Inc | Salt forms of e-2-methoxy-n-(3-(4-(3-methyl-pyridin-3-yloxy)-phenylamino)-quinazolin-6-yl)-allyl)-acetamide, its preparation and its use against cancer |
| BR0214499A (pt) | 2001-12-12 | 2005-05-10 | Pfizer Prod Inc | Derivados de quinazolina para o tratamento do crescimento anormal das células |
| US20050009845A1 (en) | 2001-12-19 | 2005-01-13 | Caferro Thomas R. | Thienopyrimidine compounds as protein tyrosine kinase inhibitors |
| RU2389731C2 (ru) * | 2004-06-02 | 2010-05-20 | Такеда Фармасьютикал Компани Лимитед | Конденсированное гетероциклическое соединение |
| TW200730527A (en) * | 2005-12-02 | 2007-08-16 | Takeda Pharmaceuticals Co | Fused heterocyclic compound |
| JP4504337B2 (ja) | 2006-09-04 | 2010-07-14 | 株式会社御池鐵工所 | ガス化炉及びガス化炉システム |
| RU2009126576A (ru) * | 2006-12-12 | 2011-01-20 | Такеда Фармасьютикал Компани Лимитед (Jp) | Конденсированное гетероциклическое соединение |
-
2009
- 2009-03-11 WO PCT/JP2009/054603 patent/WO2009113560A1/ja not_active Ceased
- 2009-03-11 UY UY0001031704A patent/UY31704A/es not_active Application Discontinuation
- 2009-03-11 EP EP09719847A patent/EP2253633A4/en not_active Withdrawn
- 2009-03-11 PE PE2009000360A patent/PE20091580A1/es not_active Application Discontinuation
- 2009-03-11 JP JP2010502844A patent/JPWO2009113560A1/ja not_active Withdrawn
- 2009-03-11 US US12/402,259 patent/US20090233937A1/en not_active Abandoned
- 2009-03-11 AR ARP090100856A patent/AR070874A1/es unknown
- 2009-03-11 TW TW098107816A patent/TW200944528A/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2009113560A1 (ja) | 2009-09-17 |
| EP2253633A4 (en) | 2012-02-29 |
| JPWO2009113560A1 (ja) | 2011-07-21 |
| EP2253633A1 (en) | 2010-11-24 |
| TW200944528A (en) | 2009-11-01 |
| PE20091580A1 (es) | 2009-11-05 |
| US20090233937A1 (en) | 2009-09-17 |
| AR070874A1 (es) | 2010-05-12 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 104 | Application deemed to be withdrawn (no substantive examination fee paid) |
Effective date: 20100604 |