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UY30052A1 - 3-aminociclopentanocarboxamidas como moduladores de receptores de quimioquinas - Google Patents

3-aminociclopentanocarboxamidas como moduladores de receptores de quimioquinas

Info

Publication number
UY30052A1
UY30052A1 UY30052A UY30052A UY30052A1 UY 30052 A1 UY30052 A1 UY 30052A1 UY 30052 A UY30052 A UY 30052A UY 30052 A UY30052 A UY 30052A UY 30052 A1 UY30052 A1 UY 30052A1
Authority
UY
Uruguay
Prior art keywords
chemiokin
aminociclopentanocarboxamids
receptors modulators
receptors
compounds
Prior art date
Application number
UY30052A
Other languages
English (en)
Inventor
Chu-Biao Xue
Original Assignee
Incyte Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38126410&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY30052(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Incyte Corp filed Critical Incyte Corp
Publication of UY30052A1 publication Critical patent/UY30052A1/es

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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  • Life Sciences & Earth Sciences (AREA)
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  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
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Abstract

La presente invención se refiere a compuestos de Fórmula I: que son moduladores de receptores de quimioquinas. Los compuestos de la invención, y las composiciones de los mismos, son útiles en el tratamiento de enfermedades relacionadas con la expresión y/o actividad de receptores de quimioquinas,
UY30052A 2005-12-21 2006-12-21 3-aminociclopentanocarboxamidas como moduladores de receptores de quimioquinas UY30052A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US75232005P 2005-12-21 2005-12-21
US75247705P 2005-12-21 2005-12-21

Publications (1)

Publication Number Publication Date
UY30052A1 true UY30052A1 (es) 2007-07-31

Family

ID=38126410

Family Applications (1)

Application Number Title Priority Date Filing Date
UY30052A UY30052A1 (es) 2005-12-21 2006-12-21 3-aminociclopentanocarboxamidas como moduladores de receptores de quimioquinas

Country Status (21)

Country Link
US (2) US7700624B2 (es)
EP (1) EP1971576A2 (es)
JP (1) JP2009520809A (es)
KR (1) KR20080070868A (es)
AP (1) AP2008004487A0 (es)
AR (1) AR058402A1 (es)
AU (1) AU2006327823A1 (es)
BR (1) BRPI0620073A2 (es)
CA (1) CA2634636A1 (es)
CR (1) CR10060A (es)
EA (1) EA200801220A1 (es)
EC (1) ECSP088527A (es)
IL (1) IL191602A0 (es)
MA (1) MA30077B1 (es)
ME (1) MEP1008A (es)
NL (1) NL2000380C2 (es)
NO (1) NO20082285L (es)
RS (1) RS20080246A (es)
TW (1) TW200734323A (es)
UY (1) UY30052A1 (es)
WO (1) WO2007072201A2 (es)

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MEP1008A (xx) * 2005-12-21 2010-02-10 Incyte Corp 3-aminociklopentankarboksamidi kao modulatori receptora hemokina
US7910108B2 (en) 2006-06-05 2011-03-22 Incyte Corporation Sheddase inhibitors combined with CD30-binding immunotherapeutics for the treatment of CD30 positive diseases
HRP20130409T2 (hr) 2008-11-26 2013-11-22 Pfizer Inc. 3-aminociklopentankarboksamidi kao modulatori kemokinskih receptora
JP5786257B2 (ja) * 2011-06-16 2015-09-30 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 新規の選択的ｃｃｒ２拮抗薬
TW201613864A (en) 2014-02-20 2016-04-16 Takeda Pharmaceutical Novel compounds
MX381819B (es) 2014-08-04 2025-03-13 Nuevolution As Derivados de heterociclico opcionalmente condensados de pirimidina útiles para el tratamiento de enfermedades inflamatorias, metabólicas oncológicas y autoinmunitarias.
MX2022007265A (es) 2019-12-20 2022-09-09 Nuevolution As Compuestos activos frente a receptores nucleares.
JP7746259B2 (ja) 2019-12-20 2025-09-30 ヌエヴォリューション・アクティーゼルスカブ 核内受容体に対して活性の化合物
WO2021198955A1 (en) 2020-03-31 2021-10-07 Nuevolution A/S Compounds active towards nuclear receptors
EP4126875A1 (en) 2020-03-31 2023-02-08 Nuevolution A/S Compounds active towards nuclear receptors
CN119968355A (zh) 2022-10-07 2025-05-09 橘生药品工业株式会社 环戊烷化合物

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NL2000380A1 (nl) 2007-06-25
JP2009520809A (ja) 2009-05-28
EA200801220A1 (ru) 2008-12-30
RS20080246A (sr) 2009-07-15
WO2007072201A3 (en) 2007-10-04
EP1971576A2 (en) 2008-09-24
US20100203039A1 (en) 2010-08-12
IL191602A0 (en) 2009-02-11
NL2000380C2 (nl) 2007-11-28
AU2006327823A1 (en) 2007-06-28
BRPI0620073A2 (pt) 2011-11-01
TW200734323A (en) 2007-09-16
AP2008004487A0 (en) 2008-06-30
MEP1008A (xx) 2010-02-10
CR10060A (es) 2008-07-17
ECSP088527A (es) 2008-07-30
US20070149532A1 (en) 2007-06-28
AR058402A1 (es) 2008-01-30
CA2634636A1 (en) 2007-06-28
KR20080070868A (ko) 2008-07-31
WO2007072201A2 (en) 2007-06-28
US7700624B2 (en) 2010-04-20
NO20082285L (no) 2008-06-18
MA30077B1 (fr) 2008-12-01

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