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UY30546A1 - Derivados de avermectina - Google Patents

Derivados de avermectina

Info

Publication number
UY30546A1
UY30546A1 UY30546A UY30546A UY30546A1 UY 30546 A1 UY30546 A1 UY 30546A1 UY 30546 A UY30546 A UY 30546A UY 30546 A UY30546 A UY 30546A UY 30546 A1 UY30546 A1 UY 30546A1
Authority
UY
Uruguay
Prior art keywords
avermectin derivatives
preparation
new
derivatives
avermectin
Prior art date
Application number
UY30546A
Other languages
English (en)
Inventor
Dr Andreas Turberg
Dr Achim Harder
Dr Erich Sanwald
Dr Christian Arnold
Ulrich Gorgens
Dr Olga Malsam
Dr Reiner Fischer
Dr Robert Velten
Dr Gunter Karig
Dr Peter Jeschke
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of UY30546A1 publication Critical patent/UY30546A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A61P33/12—Schistosomicides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H13/00—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids
    • C07H13/02—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by carboxylic acids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Veterinary Medicine (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pest Control & Pesticides (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Agronomy & Crop Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Saccharide Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

Nuevos derivados de avermectina de formula (I) en la que -C22R1-A-C23R2, R3, R4 y R5 tienen los significados dados en la descripcion, procedimiento para la preparacion de estas sustancias y su uso para combatir parásitos animales así como nuevos productos intermedios y su preparacion.
UY30546A 2006-08-17 2007-08-16 Derivados de avermectina UY30546A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102006038632 2006-08-17
DE102007007750A DE102007007750A1 (de) 2006-08-17 2007-02-16 Avermectinderivate

Publications (1)

Publication Number Publication Date
UY30546A1 true UY30546A1 (es) 2008-03-31

Family

ID=38920558

Family Applications (1)

Application Number Title Priority Date Filing Date
UY30546A UY30546A1 (es) 2006-08-17 2007-08-16 Derivados de avermectina

Country Status (19)

Country Link
US (1) US8183351B2 (es)
EP (1) EP2054427B1 (es)
JP (1) JP2010500982A (es)
KR (1) KR20090040384A (es)
AR (1) AR063689A1 (es)
AT (1) ATE473994T1 (es)
AU (1) AU2007286506B2 (es)
BR (1) BRPI0715789A2 (es)
CA (1) CA2660751A1 (es)
CL (1) CL2007002393A1 (es)
DE (2) DE102007007750A1 (es)
ES (1) ES2347292T3 (es)
MX (1) MX2009001766A (es)
NZ (1) NZ574886A (es)
PE (1) PE20080910A1 (es)
RU (1) RU2009109347A (es)
TW (1) TW200823221A (es)
UY (1) UY30546A1 (es)
WO (1) WO2008019784A2 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2723648A1 (en) 2008-04-10 2009-10-15 Piyush Gupta Methods for identification and use of agents targeting cancer stem cells

Family Cites Families (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4024163A (en) * 1972-05-25 1977-05-17 National Research Development Corporation Insecticides
SE434277B (sv) * 1976-04-19 1984-07-16 Merck & Co Inc Sett att framstella nya antihelmintiskt verkande foreningar genom odling av streptomyces avermitilis
US4183948A (en) * 1977-01-24 1980-01-15 Imperial Chemical Industries Limited Halogenated esters
US4206205A (en) * 1977-10-03 1980-06-03 Merck & Co., Inc. Monosaccharide and aglycone derivatives of C-076
US4201861A (en) * 1977-10-03 1980-05-06 Merck & Co., Inc. Acyl derivatives of C-076 compounds
US4199569A (en) * 1977-10-03 1980-04-22 Merck & Co., Inc. Selective hydrogenation products of C-076 compounds and derivatives thereof
NZ188459A (en) 1977-10-03 1982-09-07 Merck & Co Inc Derivatives of c-076 compounds and pesticidal compositions
FR2421867A1 (fr) * 1978-04-04 1979-11-02 Azote & Prod Chim Procede de fabrication de nitroparaffines par nitration en phase gazeuse
EP0235085A1 (de) 1986-02-20 1987-09-02 Ciba-Geigy Ag 13-Beta-Zuckerderivate von Milbemycinen, deren Herstellung und Verwendung gegen Ekto-und Endoparasiten am Nutztier oder an der Nutzpflanze
US5023241A (en) * 1989-07-31 1991-06-11 Merck & Co., Inc. Avermectin derivatives
ATE198493T1 (de) 1992-03-23 2001-01-15 Merck & Co Inc Ein streptomyces avermitilis-stamm glykosyliert avermectin-verbindungen
US5229415A (en) * 1992-03-24 1993-07-20 Merck & Co., Inc. Alkylthio alkyl avermectins are active antiparasitic agents
US5229416A (en) * 1992-04-29 1993-07-20 Merck & Co., Inc. Avermectin difluoro derivatives
GB9300883D0 (en) 1993-01-18 1993-03-10 Pfizer Ltd Antiparasitic agents
GB9312154D0 (en) 1993-06-12 1993-07-28 Pfizer Ltd Antiparasitic agents
GB9315108D0 (en) 1993-07-21 1993-09-01 Pfizer Ltd Antiparasitic agents
US5981500A (en) * 1994-01-12 1999-11-09 Pfizer Inc. Antiparasitic agents related to the milbemycins and avermectins
DE19503827A1 (de) 1995-02-06 1996-08-08 Basf Ag Verwendung von schwerflüchtigen Pyrazolderivaten mit hydrophilen Gruppen als Nitrifikationsinhibitoren
EP0929524A1 (de) 1996-09-18 1999-07-21 Basf Aktiengesellschaft Pyridinderivate, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von tierischen schädlingen und schadpilzen
WO1999067209A1 (en) 1998-06-20 1999-12-29 Hoechst Schering Agrevo Gmbh Hydroximic acid derivatives, process for their preparation and intermediates therefor
US20040087519A1 (en) 2000-08-09 2004-05-06 Satoshi Omura Avermectin derivatives
WO2002059078A1 (en) 2001-01-23 2002-08-01 Sankyo Agro Company, Limited PROCESS FOR PRODUCING Z-α-ALKOXYIMINOPHENYLACETIC ACID DERIVATIVE
GB0320176D0 (en) 2003-08-28 2003-10-01 Syngenta Participations Ag Avermectins and avermectin monosaccharides substitued in the 4'-and 4"-positionhaving pesticidal properties
WO2005102335A2 (en) * 2004-04-23 2005-11-03 Hypnion, Inc. Methods of treating sleep disorders

Also Published As

Publication number Publication date
TW200823221A (en) 2008-06-01
AU2007286506B2 (en) 2011-11-03
CL2007002393A1 (es) 2008-04-04
DE102007007750A1 (de) 2008-02-21
PE20080910A1 (es) 2008-09-05
BRPI0715789A2 (pt) 2014-08-19
US20100234312A1 (en) 2010-09-16
AR063689A1 (es) 2009-02-11
WO2008019784A2 (de) 2008-02-21
WO2008019784A8 (de) 2009-07-23
WO2008019784A3 (de) 2008-09-25
ES2347292T3 (es) 2010-10-27
US8183351B2 (en) 2012-05-22
JP2010500982A (ja) 2010-01-14
RU2009109347A (ru) 2010-09-27
NZ574886A (en) 2010-10-29
AU2007286506A1 (en) 2008-02-21
MX2009001766A (es) 2009-04-17
KR20090040384A (ko) 2009-04-23
EP2054427B1 (de) 2010-07-14
DE502007004416D1 (de) 2010-08-26
CA2660751A1 (en) 2008-02-21
EP2054427A2 (de) 2009-05-06
ATE473994T1 (de) 2010-07-15

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Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20170725