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PE20080910A1 - Derivados de avermectina - Google Patents

Derivados de avermectina

Info

Publication number
PE20080910A1
PE20080910A1 PE2007001104A PE2007001104A PE20080910A1 PE 20080910 A1 PE20080910 A1 PE 20080910A1 PE 2007001104 A PE2007001104 A PE 2007001104A PE 2007001104 A PE2007001104 A PE 2007001104A PE 20080910 A1 PE20080910 A1 PE 20080910A1
Authority
PE
Peru
Prior art keywords
avermectin
derivatives
parasiticides
alkinyl
cyclohexyl
Prior art date
Application number
PE2007001104A
Other languages
English (en)
Inventor
Peter Jeschke
Gunter Karig
Robert Velten
Reiner Fischer
Olga Malsam
Ulrich Gorgens
Christian Arnold
Erich Sanwald
Achim Harder
Andreas Turberg
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of PE20080910A1 publication Critical patent/PE20080910A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A61P33/12—Schistosomicides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H13/00—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids
    • C07H13/02—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by carboxylic acids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Veterinary Medicine (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pest Control & Pesticides (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Agronomy & Crop Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Saccharide Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

REFERIDA A DERIVADOS DE AVERMECTINA DE FORMULA (I), DONDE -C22R1-A-C23R2- ES -HC=CH-, -H2C-CH(OH)- O -H2C-CH2-; R3 ES SEC-BUTILO, ISO-PROPILO O CICLOHEXILO; R5 ES H, METILO O ALQUIL C1-C4-CARBONILO; R4 ES ALQUENILO C2-C6, ALQUINILO C2-C6, ARILO, ENTRE OTROS. TAMBIEN ESTA REFERIDA A UN PROCEDIMIENTO DE PREPARACION Y A UNA COMPOSICION QUIMICA. DICHOS COMPUESTOS SON UTILES COMO PARASITICIDAS
PE2007001104A 2006-08-17 2007-08-16 Derivados de avermectina PE20080910A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102006038632 2006-08-17
DE102007007750A DE102007007750A1 (de) 2006-08-17 2007-02-16 Avermectinderivate

Publications (1)

Publication Number Publication Date
PE20080910A1 true PE20080910A1 (es) 2008-09-05

Family

ID=38920558

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2007001104A PE20080910A1 (es) 2006-08-17 2007-08-16 Derivados de avermectina

Country Status (19)

Country Link
US (1) US8183351B2 (es)
EP (1) EP2054427B1 (es)
JP (1) JP2010500982A (es)
KR (1) KR20090040384A (es)
AR (1) AR063689A1 (es)
AT (1) ATE473994T1 (es)
AU (1) AU2007286506B2 (es)
BR (1) BRPI0715789A2 (es)
CA (1) CA2660751A1 (es)
CL (1) CL2007002393A1 (es)
DE (2) DE102007007750A1 (es)
ES (1) ES2347292T3 (es)
MX (1) MX2009001766A (es)
NZ (1) NZ574886A (es)
PE (1) PE20080910A1 (es)
RU (1) RU2009109347A (es)
TW (1) TW200823221A (es)
UY (1) UY30546A1 (es)
WO (1) WO2008019784A2 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009126310A2 (en) 2008-04-10 2009-10-15 Massachusetts Institute Of Technology Methods for identification and use of agents targeting cancer stem cells

Family Cites Families (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4024163A (en) * 1972-05-25 1977-05-17 National Research Development Corporation Insecticides
SE434277B (sv) * 1976-04-19 1984-07-16 Merck & Co Inc Sett att framstella nya antihelmintiskt verkande foreningar genom odling av streptomyces avermitilis
US4183948A (en) * 1977-01-24 1980-01-15 Imperial Chemical Industries Limited Halogenated esters
US4206205A (en) * 1977-10-03 1980-06-03 Merck & Co., Inc. Monosaccharide and aglycone derivatives of C-076
NZ188459A (en) 1977-10-03 1982-09-07 Merck & Co Inc Derivatives of c-076 compounds and pesticidal compositions
US4199569A (en) * 1977-10-03 1980-04-22 Merck & Co., Inc. Selective hydrogenation products of C-076 compounds and derivatives thereof
US4201861A (en) * 1977-10-03 1980-05-06 Merck & Co., Inc. Acyl derivatives of C-076 compounds
FR2421867A1 (fr) * 1978-04-04 1979-11-02 Azote & Prod Chim Procede de fabrication de nitroparaffines par nitration en phase gazeuse
EP0235085A1 (de) * 1986-02-20 1987-09-02 Ciba-Geigy Ag 13-Beta-Zuckerderivate von Milbemycinen, deren Herstellung und Verwendung gegen Ekto-und Endoparasiten am Nutztier oder an der Nutzpflanze
US5023241A (en) * 1989-07-31 1991-06-11 Merck & Co., Inc. Avermectin derivatives
DE69329821T2 (de) 1992-03-23 2001-07-19 Merck & Co., Inc. Ein streptomyces avermitilis-stamm glykosyliert avermectin-verbindungen
US5229415A (en) * 1992-03-24 1993-07-20 Merck & Co., Inc. Alkylthio alkyl avermectins are active antiparasitic agents
US5229416A (en) * 1992-04-29 1993-07-20 Merck & Co., Inc. Avermectin difluoro derivatives
GB9300883D0 (en) 1993-01-18 1993-03-10 Pfizer Ltd Antiparasitic agents
GB9312154D0 (en) 1993-06-12 1993-07-28 Pfizer Ltd Antiparasitic agents
GB9315108D0 (en) 1993-07-21 1993-09-01 Pfizer Ltd Antiparasitic agents
US5981500A (en) * 1994-01-12 1999-11-09 Pfizer Inc. Antiparasitic agents related to the milbemycins and avermectins
DE19503827A1 (de) 1995-02-06 1996-08-08 Basf Ag Verwendung von schwerflüchtigen Pyrazolderivaten mit hydrophilen Gruppen als Nitrifikationsinhibitoren
US6228810B1 (en) 1996-09-18 2001-05-08 Basf Ag Pyridine derivatives, process for preparing the same and their use for controlling animal pests and harmful fungi
AU4377799A (en) 1998-06-20 2000-01-10 Hoechst Schering Agrevo Gmbh Hydroximic acid derivatives, process for their preparation and intermediates therefor
WO2002012248A1 (en) 2000-08-09 2002-02-14 The Kitasato Institute Avermectin derivatives
WO2002059078A1 (en) 2001-01-23 2002-08-01 Sankyo Agro Company, Limited PROCESS FOR PRODUCING Z-α-ALKOXYIMINOPHENYLACETIC ACID DERIVATIVE
GB0320176D0 (en) 2003-08-28 2003-10-01 Syngenta Participations Ag Avermectins and avermectin monosaccharides substitued in the 4'-and 4"-positionhaving pesticidal properties
WO2005102335A2 (en) * 2004-04-23 2005-11-03 Hypnion, Inc. Methods of treating sleep disorders

Also Published As

Publication number Publication date
BRPI0715789A2 (pt) 2014-08-19
US20100234312A1 (en) 2010-09-16
WO2008019784A8 (de) 2009-07-23
AR063689A1 (es) 2009-02-11
US8183351B2 (en) 2012-05-22
WO2008019784A3 (de) 2008-09-25
AU2007286506A1 (en) 2008-02-21
EP2054427A2 (de) 2009-05-06
WO2008019784A2 (de) 2008-02-21
JP2010500982A (ja) 2010-01-14
UY30546A1 (es) 2008-03-31
DE102007007750A1 (de) 2008-02-21
RU2009109347A (ru) 2010-09-27
MX2009001766A (es) 2009-04-17
ES2347292T3 (es) 2010-10-27
DE502007004416D1 (de) 2010-08-26
CL2007002393A1 (es) 2008-04-04
KR20090040384A (ko) 2009-04-23
NZ574886A (en) 2010-10-29
AU2007286506B2 (en) 2011-11-03
EP2054427B1 (de) 2010-07-14
ATE473994T1 (de) 2010-07-15
CA2660751A1 (en) 2008-02-21
TW200823221A (en) 2008-06-01

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