UY26964A1 - Derivados de eritromicina 6-0-sustituidos con mayor tolerancia gastrointestinal - Google Patents
Derivados de eritromicina 6-0-sustituidos con mayor tolerancia gastrointestinalInfo
- Publication number
- UY26964A1 UY26964A1 UY26964A UY26964A UY26964A1 UY 26964 A1 UY26964 A1 UY 26964A1 UY 26964 A UY26964 A UY 26964A UY 26964 A UY26964 A UY 26964A UY 26964 A1 UY26964 A1 UY 26964A1
- Authority
- UY
- Uruguay
- Prior art keywords
- erythromycin
- derivatives
- replaced
- gastrointestinal tolerance
- greater gastrointestinal
- Prior art date
Links
- 230000002496 gastric effect Effects 0.000 title abstract 2
- ULGZDMOVFRHVEP-RWJQBGPGSA-N Erythromycin Chemical class O([C@@H]1[C@@H](C)C(=O)O[C@@H]([C@@]([C@H](O)[C@@H](C)C(=O)[C@H](C)C[C@@](C)(O)[C@H](O[C@H]2[C@@H]([C@H](C[C@@H](C)O2)N(C)C)O)[C@H]1C)(C)O)CC)[C@H]1C[C@@](C)(OC)[C@@H](O)[C@H](C)O1 ULGZDMOVFRHVEP-RWJQBGPGSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 208000035143 Bacterial infection Diseases 0.000 abstract 1
- 208000022362 bacterial infectious disease Diseases 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- Communicable Diseases (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Abstract
Compuestos de fórmula I son útiles para el tratamiento de infeciones bacterianas pero sin producir el efecto colateral de intolerancia gastrointestinal. También se revelan composiciones que contienen los compuestos y métodos de tratamiento que los utilizan.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US24077700P | 2000-10-16 | 2000-10-16 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UY26964A1 true UY26964A1 (es) | 2002-06-20 |
Family
ID=22907903
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UY26964A UY26964A1 (es) | 2000-10-16 | 2001-10-12 | Derivados de eritromicina 6-0-sustituidos con mayor tolerancia gastrointestinal |
Country Status (9)
| Country | Link |
|---|---|
| EP (1) | EP1328534A2 (es) |
| JP (1) | JP2004529857A (es) |
| AU (1) | AU2002213267A1 (es) |
| BR (1) | BR0109946A (es) |
| CA (1) | CA2420012A1 (es) |
| MX (1) | MXPA03003311A (es) |
| PE (1) | PE20020522A1 (es) |
| UY (1) | UY26964A1 (es) |
| WO (1) | WO2002032919A2 (es) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2004117082A (ru) | 2001-12-05 | 2005-04-10 | Орто-Макнейл Фармасьютикал, Инк. (Us) | Кетолидные 6-0-ацил-производные эритромицина в качестве антибактериальных средств |
| EP1501845A1 (en) * | 2002-04-30 | 2005-02-02 | Abbott Laboratories | Antibacterial compounds with improved pharmacokinetic profiles |
| US6727229B2 (en) * | 2002-08-19 | 2004-04-27 | Enanta Pharmaceuticals, Inc. | 11,12-substituted lactone ketolide derivatives having antibacterial activity |
| WO2004078771A1 (ja) * | 2003-03-07 | 2004-09-16 | Taisho Pharmaceutical Co., Ltd. | ２－フルオロ－６－ｏ－置換ケトライド誘導体 |
| JP2007223900A (ja) * | 2004-02-03 | 2007-09-06 | Taisho Pharmaceut Co Ltd | ６−ｏ−置換ケトライド誘導体 |
| JP2007254285A (ja) * | 2004-03-16 | 2007-10-04 | Taisho Pharmaceut Co Ltd | ２−フルオロ−６−ｏ−置換ケトライド誘導体 |
| EP1985620A4 (en) | 2006-02-07 | 2012-08-15 | Taisho Pharmaceutical Co Ltd | COMPOUND 10a-AZALIDE |
| US8293715B2 (en) | 2007-08-06 | 2012-10-23 | Taisho Pharmaceutical Co., Ltd. | 10a-Azalide compound crosslinked at 10a- and 12-positions |
| US8299035B2 (en) | 2008-05-15 | 2012-10-30 | Taisho Pharmaceutucal Co., Ltd. | 10a-azalide compound having 4-membered ring structure |
| CN102234302B (zh) * | 2010-05-07 | 2014-05-07 | 北京理工大学 | 一种酮内酯衍生物、制备方法及其药物组合物 |
| AR085286A1 (es) | 2011-02-21 | 2013-09-18 | Taisho Pharmaceutical Co Ltd | Derivado de macrolido sustituido en la posicion c-4 |
| AR102810A1 (es) | 2014-08-18 | 2017-03-29 | Taisho Pharmaceutical Co Ltd | Derivado de macrólido sustituido en la posición c-4 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6054435A (en) * | 1999-03-19 | 2000-04-25 | Abbott Laboratories | 6-O-substituted macrolides having antibacterial activity |
-
2001
- 2001-10-12 UY UY26964A patent/UY26964A1/es not_active Application Discontinuation
- 2001-10-15 PE PE2001001021A patent/PE20020522A1/es not_active Application Discontinuation
- 2001-10-16 AU AU2002213267A patent/AU2002213267A1/en not_active Abandoned
- 2001-10-16 JP JP2002536300A patent/JP2004529857A/ja not_active Withdrawn
- 2001-10-16 MX MXPA03003311A patent/MXPA03003311A/es unknown
- 2001-10-16 BR BR0109946-9A patent/BR0109946A/pt not_active Application Discontinuation
- 2001-10-16 WO PCT/US2001/032278 patent/WO2002032919A2/en not_active Ceased
- 2001-10-16 CA CA002420012A patent/CA2420012A1/en not_active Abandoned
- 2001-10-16 EP EP01981637A patent/EP1328534A2/en not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| BR0109946A (pt) | 2005-08-02 |
| EP1328534A2 (en) | 2003-07-23 |
| CA2420012A1 (en) | 2002-04-25 |
| JP2004529857A (ja) | 2004-09-30 |
| PE20020522A1 (es) | 2002-06-25 |
| MXPA03003311A (es) | 2003-09-10 |
| WO2002032919A3 (en) | 2002-09-19 |
| WO2002032919A2 (en) | 2002-04-25 |
| AU2002213267A1 (en) | 2002-04-29 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 109 | Application deemed to be withdrawn |
Effective date: 20150126 |