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AR102810A1 - Derivado de macrólido sustituido en la posición c-4 - Google Patents

Derivado de macrólido sustituido en la posición c-4

Info

Publication number
AR102810A1
AR102810A1 ARP150102636A ARP150102636A AR102810A1 AR 102810 A1 AR102810 A1 AR 102810A1 AR P150102636 A ARP150102636 A AR P150102636A AR P150102636 A ARP150102636 A AR P150102636A AR 102810 A1 AR102810 A1 AR 102810A1
Authority
AR
Argentina
Prior art keywords
macrolid
derivative replaced
derivative
replaced
solvate
Prior art date
Application number
ARP150102636A
Other languages
English (en)
Inventor
Kawaguchi Takanori
Hayashi Masato
Sugimoto Tomohiro
Original Assignee
Taisho Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Taisho Pharmaceutical Co Ltd filed Critical Taisho Pharmaceutical Co Ltd
Publication of AR102810A1 publication Critical patent/AR102810A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

La presente provee un compuesto representado por la fórmula (1), o una sal farmacéuticamente aceptable del mismo, o un hidrato o un solvato del mismo.
ARP150102636A 2014-08-18 2015-08-14 Derivado de macrólido sustituido en la posición c-4 AR102810A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2014165848 2014-08-18

Publications (1)

Publication Number Publication Date
AR102810A1 true AR102810A1 (es) 2017-03-29

Family

ID=55350700

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP150102636A AR102810A1 (es) 2014-08-18 2015-08-14 Derivado de macrólido sustituido en la posición c-4

Country Status (19)

Country Link
US (1) US20170267708A1 (es)
EP (1) EP3192798A4 (es)
JP (1) JP5874871B1 (es)
KR (1) KR20170036106A (es)
CN (1) CN106573953A (es)
AR (1) AR102810A1 (es)
AU (1) AU2015304439A1 (es)
BR (1) BR112017000606A2 (es)
CA (1) CA2957628A1 (es)
CL (1) CL2017000395A1 (es)
CO (1) CO2017002440A2 (es)
IL (1) IL250559A0 (es)
MX (1) MX2017002223A (es)
PE (1) PE20170467A1 (es)
PH (1) PH12017500223A1 (es)
RU (1) RU2017108908A (es)
SG (1) SG11201701146TA (es)
TW (1) TW201625656A (es)
WO (1) WO2016027755A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2017142002A1 (ja) * 2016-02-17 2017-08-24 大正製薬株式会社 C-4"位置換マクロライド化合物フリー体及び塩の結晶形並びにそれらの製造方法
CN114231430B (zh) * 2021-06-11 2024-02-09 常州大学 一种红霉素降解菌iurm f57及其应用

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS54967A (en) 1977-06-06 1979-01-06 Mitsubishi Electric Corp Output circuit
YU43006B (en) 1981-03-06 1989-02-28 Pliva Pharm & Chem Works Process for preparing n-methyl-11-aza-10-deoxo-10-dihydro erythromycin and derivatives thereof
US4474768A (en) 1982-07-19 1984-10-02 Pfizer Inc. N-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates therefor
DE69733723T2 (de) 1996-09-04 2006-04-20 Abbott Laboratories, Abbott Park 6-o-Substituierte Ketoliden mit antibakteriellen Wirkung
HN1998000074A (es) 1997-06-11 1999-01-08 Pfizer Prod Inc Derivados de macrolidos c-4 sustituidos
UY26964A1 (es) 2000-10-16 2002-06-20 Abbott Lab Derivados de eritromicina 6-0-sustituidos con mayor tolerancia gastrointestinal
AR085286A1 (es) * 2011-02-21 2013-09-18 Taisho Pharmaceutical Co Ltd Derivado de macrolido sustituido en la posicion c-4
JP2014058508A (ja) * 2012-08-20 2014-04-03 Taisho Pharmaceutical Co Ltd 9位オキシム置換マクロライド誘導体
JP5857008B2 (ja) * 2012-08-20 2016-02-10 大正製薬株式会社 C−4”位置換マクロライド誘導体を含有する医薬
JP2014058507A (ja) * 2012-08-20 2014-04-03 Taisho Pharmaceutical Co Ltd 11位アミノ置換マクロライド誘導体

Also Published As

Publication number Publication date
CA2957628A1 (en) 2016-02-25
CN106573953A (zh) 2017-04-19
PE20170467A1 (es) 2017-04-26
US20170267708A1 (en) 2017-09-21
CL2017000395A1 (es) 2018-01-05
MX2017002223A (es) 2017-05-09
SG11201701146TA (en) 2017-03-30
IL250559A0 (en) 2017-03-30
BR112017000606A2 (pt) 2017-11-07
RU2017108908A (ru) 2018-09-21
PH12017500223A1 (en) 2017-07-10
EP3192798A4 (en) 2018-01-03
WO2016027755A1 (ja) 2016-02-25
EP3192798A1 (en) 2017-07-19
JP5874871B1 (ja) 2016-03-02
AU2015304439A1 (en) 2017-03-16
KR20170036106A (ko) 2017-03-31
TW201625656A (zh) 2016-07-16
JPWO2016027755A1 (ja) 2017-04-27
CO2017002440A2 (es) 2017-04-28

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