UA94921C2 - 1-orthofluorophenyl substituted 1, 2, 5-thiazolidinedione derivatives as ptp-as inhibitors - Google Patents

1-orthofluorophenyl substituted 1, 2, 5-thiazolidinedione derivatives as ptp-as inhibitors

Info

Publication number: UA94921C2
Authority: UA; Ukraine
Prior art keywords: employed; compounds; inhibitors; formula; treatment
Prior art date: 2005-12-08

Application number

UAA200807752A

Other languages

English (en)

Inventor

Девид Барнес

Гари Марк Коппола

Тревис Стемс

Сидни Вулф Топиол

Original Assignee

Новартис Аг

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2005-12-08

Filing date

2006-06-12

Publication date

2011-06-25

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37903424&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UA94921(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2006-06-12 Application filed by Новартис Аг filed Critical Новартис Аг

2011-06-25 Publication of UA94921C2 publication Critical patent/UA94921C2/ru

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/433—Thidiazoles
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- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/10—1,2,5-Thiadiazoles; Hydrogenated 1,2,5-thiadiazoles

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Cardiology (AREA)
Biomedical Technology (AREA)
Heart & Thoracic Surgery (AREA)
Diabetes (AREA)
Obesity (AREA)
Physical Education & Sports Medicine (AREA)
Hematology (AREA)
Rheumatology (AREA)
Immunology (AREA)
Orthopedic Medicine & Surgery (AREA)
Urology & Nephrology (AREA)
Psychology (AREA)
Hospice & Palliative Care (AREA)
Vascular Medicine (AREA)
Pain & Pain Management (AREA)
Oncology (AREA)
Emergency Medicine (AREA)
Endocrinology (AREA)
Psychiatry (AREA)
Communicable Diseases (AREA)
Ophthalmology & Optometry (AREA)
Child & Adolescent Psychology (AREA)
Pulmonology (AREA)

UAA200807752A 2005-12-08 2006-06-12 1-orthofluorophenyl substituted 1, 2, 5-thiazolidinedione derivatives as ptp-as inhibitors UA94921C2 (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US74849205P	2005-12-08	2005-12-08

Publications (1)

Publication Number	Publication Date
UA94921C2 true UA94921C2 (en)	2011-06-25

Family

ID=37903424

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
UAA200807752A UA94921C2 (en)	2005-12-08	2006-06-12	1-orthofluorophenyl substituted 1, 2, 5-thiazolidinedione derivatives as ptp-as inhibitors

Country Status (23)

Country	Link
US (1)	US8252820B2 (ru)
EP (1)	EP1963293A1 (ru)
JP (1)	JP2009518419A (ru)
KR (1)	KR20080075218A (ru)
CN (1)	CN101336235A (ru)
AR (1)	AR058285A1 (ru)
AU (1)	AU2006321902B2 (ru)
BR (1)	BRPI0619567A2 (ru)
CA (1)	CA2631007A1 (ru)
CR (1)	CR10047A (ru)
EC (1)	ECSP088509A (ru)
GT (1)	GT200800093A (ru)
IL (1)	IL191711A0 (ru)
MA (1)	MA30018B1 (ru)
NO (1)	NO20083030L (ru)
NZ (1)	NZ568663A (ru)
PE (2)	PE20100470A1 (ru)
RU (1)	RU2008127262A (ru)
TN (1)	TNSN08248A1 (ru)
TW (1)	TW200800928A (ru)
UA (1)	UA94921C2 (ru)
WO (1)	WO2007067612A1 (ru)
ZA (1)	ZA200804489B (ru)

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CN112739687B (zh)	2018-09-18	2025-07-04	巴斯夫欧洲公司	二氨基三嗪化合物
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AR128379A1 (es)	2022-01-31	2024-04-24	Bristol Myers Squibb Co	Inhibidores de la proteína tirosina fosfatasa, composiciones y métodos de uso
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- 2006-12-06 JP JP2008544464A patent/JP2009518419A/ja active Pending
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- 2006-12-06 AU AU2006321902A patent/AU2006321902B2/en not_active Ceased
- 2006-12-06 CN CNA2006800524439A patent/CN101336235A/zh active Pending
- 2006-12-07 TW TW095145872A patent/TW200800928A/zh unknown
2008
- 2008-05-26 IL IL191711A patent/IL191711A0/en unknown
- 2008-05-27 ZA ZA200804489A patent/ZA200804489B/xx unknown
- 2008-06-02 MA MA30986A patent/MA30018B1/fr unknown
- 2008-06-05 CR CR10047A patent/CR10047A/es not_active Application Discontinuation
- 2008-06-06 GT GT200800093A patent/GT200800093A/es unknown
- 2008-06-06 TN TNP2008000248A patent/TNSN08248A1/en unknown
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Also Published As

Publication number	Publication date
ECSP088509A (es)	2008-07-30
PE20100470A1 (es)	2010-07-13
ZA200804489B (en)	2009-08-26
JP2009518419A (ja)	2009-05-07
BRPI0619567A2 (pt)	2011-10-04
CR10047A (es)	2008-10-16
TNSN08248A1 (en)	2009-10-30
AU2006321902B2 (en)	2011-11-10
AU2006321902A1 (en)	2007-06-14
PE20071094A1 (es)	2008-01-07
GT200800093A (es)	2010-07-09
AR058285A1 (es)	2008-01-30
CA2631007A1 (en)	2007-06-14
US20100035942A1 (en)	2010-02-11
US8252820B2 (en)	2012-08-28
RU2008127262A (ru)	2010-01-20
WO2007067612A1 (en)	2007-06-14
CN101336235A (zh)	2008-12-31
IL191711A0 (en)	2008-12-29
TW200800928A (en)	2008-01-01
KR20080075218A (ko)	2008-08-14
MA30018B1 (fr)	2008-12-01
EP1963293A1 (en)	2008-09-03
NZ568663A (en)	2011-07-29
NO20083030L (no)	2008-08-28

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