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TR201905392T4 - Ağrı tedavisi. - Google Patents

Ağrı tedavisi. Download PDF

Info

Publication number
TR201905392T4
TR201905392T4 TR2019/05392T TR201905392T TR201905392T4 TR 201905392 T4 TR201905392 T4 TR 201905392T4 TR 2019/05392 T TR2019/05392 T TR 2019/05392T TR 201905392 T TR201905392 T TR 201905392T TR 201905392 T4 TR201905392 T4 TR 201905392T4
Authority
TR
Turkey
Prior art keywords
pain relief
imidazo
tetrahydro
carboxylate
pyridine
Prior art date
Application number
TR2019/05392T
Other languages
English (en)
Inventor
Gonzalez Isabel
Pritchard Martyn
Richardson Peter
Original Assignee
Benevolentai Cambridge Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Benevolentai Cambridge Ltd filed Critical Benevolentai Cambridge Ltd
Publication of TR201905392T4 publication Critical patent/TR201905392T4/tr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00Anaesthetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Ağrı tedavisinde kullanıma yönelik (3S)-Tetrahidrofuran-3-il(4S)-4-izopropil-1,4,6,7-tetrahidro-5H-imidazo[4,5-c]-piridin-5-karboksilat ve bunların tuzu.
TR2019/05392T 2015-04-24 2016-04-22 Ağrı tedavisi. TR201905392T4 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB1507048.5A GB201507048D0 (en) 2015-04-24 2015-04-24 Treatment of pain

Publications (1)

Publication Number Publication Date
TR201905392T4 true TR201905392T4 (tr) 2019-05-21

Family

ID=53488643

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2019/05392T TR201905392T4 (tr) 2015-04-24 2016-04-22 Ağrı tedavisi.

Country Status (22)

Country Link
US (1) US20180104223A1 (tr)
EP (1) EP3285767B8 (tr)
JP (2) JP2018520984A (tr)
KR (1) KR20170139047A (tr)
CN (1) CN107530330A (tr)
AU (1) AU2016252237B2 (tr)
BR (1) BR112017019337A2 (tr)
CA (1) CA2979160A1 (tr)
DK (1) DK3285767T3 (tr)
EA (1) EA032512B1 (tr)
ES (1) ES2720035T3 (tr)
GB (1) GB201507048D0 (tr)
HK (1) HK1249865B (tr)
HU (1) HUE043871T2 (tr)
IL (1) IL254155B (tr)
MX (1) MX2017013047A (tr)
PL (1) PL3285767T3 (tr)
PT (1) PT3285767T (tr)
SG (1) SG11201707870SA (tr)
TR (1) TR201905392T4 (tr)
WO (1) WO2016170353A1 (tr)
ZA (1) ZA201705847B (tr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB201304526D0 (en) 2013-03-13 2013-04-24 Proximagen Ltd New compounds
GB201507036D0 (en) * 2015-04-24 2015-06-10 Proximagen Ltd Crystalline enzyme inhibitor compound
GB201507031D0 (en) * 2015-04-24 2015-06-10 Proximagen Ltd New pharmaceutical salt forms
HK1256174A1 (zh) * 2015-12-07 2019-09-13 Benevolentai Cambridge Limited 用於治疗疼痛的 vap-1 抑制剂
GB201618029D0 (en) 2016-10-25 2016-12-07 Proximagen Ltd New process
GB201709136D0 (en) * 2017-06-08 2017-07-26 Proximagen Ltd New therapeutic uses of enzyme inhibitors

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0639972A1 (en) * 1992-05-15 1995-03-01 University Of Saskatchewan Method for preventing endothelium damage in mammals and for alleviating pain associated with gout and arthritis
EP1791835A2 (en) * 2004-09-09 2007-06-06 Astellas Pharma Inc. Thiazole derivatives having vap-1 inhibitory activity
US20070066646A1 (en) * 2005-08-02 2007-03-22 Genmedica Therapeutics Sl Compounds for Inhibiting Copper-Containing Amine Oxidases and Uses Thereof
EP2029164B1 (en) 2006-06-07 2015-12-23 The Board of Trustees of the Leland Stanford Junior University Anti-leukocyte recruitment therapy for the treatment of seizures and epilepsy
TWI490214B (zh) * 2008-05-30 2015-07-01 艾德克 上野股份有限公司 苯或噻吩衍生物及該等作為vap-1抑制劑之用途
BRPI0918602B8 (pt) * 2008-09-16 2021-05-25 Benevolentai Cambridge Ltd inibidores da atividade de ssao, seu uso, e formulação farmacêutica
FI20115234A0 (fi) * 2011-03-08 2011-03-08 Biotie Therapies Corp Uusia pyridatsinoni- ja pyridoniyhdisteitä
CA2915163A1 (en) * 2013-06-12 2014-12-18 Proximagen Limited New therapeutic uses of enzyme inhibitors
US9790193B2 (en) * 2014-04-15 2017-10-17 Pécsi Tudományegyetem Semicarbazide-sensitive amine oxidase inhibitors for use as analgesics in traumatic neuropathy and neurogenic inflammation
GB201507036D0 (en) * 2015-04-24 2015-06-10 Proximagen Ltd Crystalline enzyme inhibitor compound
GB201507031D0 (en) * 2015-04-24 2015-06-10 Proximagen Ltd New pharmaceutical salt forms

Also Published As

Publication number Publication date
KR20170139047A (ko) 2017-12-18
EP3285767B1 (en) 2019-03-20
PT3285767T (pt) 2019-05-20
EP3285767B8 (en) 2019-05-22
CA2979160A1 (en) 2016-10-27
ZA201705847B (en) 2020-03-25
MX2017013047A (es) 2017-12-08
AU2016252237B2 (en) 2021-04-08
EA032512B1 (ru) 2019-06-28
DK3285767T3 (en) 2019-04-29
IL254155A0 (en) 2017-10-31
ES2720035T3 (es) 2019-07-17
GB201507048D0 (en) 2015-06-10
EA201792123A1 (ru) 2018-03-30
JP2018520984A (ja) 2018-08-02
JP2021073257A (ja) 2021-05-13
WO2016170353A1 (en) 2016-10-27
EP3285767A1 (en) 2018-02-28
US20180104223A1 (en) 2018-04-19
BR112017019337A2 (pt) 2018-06-05
PL3285767T3 (pl) 2019-09-30
IL254155B (en) 2021-02-28
CN107530330A (zh) 2018-01-02
AU2016252237A1 (en) 2017-10-05
SG11201707870SA (en) 2017-11-29
HK1249865B (en) 2019-12-06
HUE043871T2 (hu) 2019-09-30

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