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TR200102817T2 - Antiinflamatuar ajanlar olarak faydalı bileşikler - Google Patents

Antiinflamatuar ajanlar olarak faydalı bileşikler

Info

Publication number
TR200102817T2
TR200102817T2 TR2001/02817T TR200102817T TR200102817T2 TR 200102817 T2 TR200102817 T2 TR 200102817T2 TR 2001/02817 T TR2001/02817 T TR 2001/02817T TR 200102817 T TR200102817 T TR 200102817T TR 200102817 T2 TR200102817 T2 TR 200102817T2
Authority
TR
Turkey
Prior art keywords
compounds useful
inflammatory agents
inflammatory diseases
compounds
processes
Prior art date
Application number
TR2001/02817T
Other languages
English (en)
Inventor
Betageri Rajashehar
Breitfelder Steffen
Francesco Cirillo Pier
A. Gilmore Thomas
Richard Hickey Eugene
M. Kirrane Thomas
Helen Moriak Monica
Moss Neil
R. Patel Usha
Robert Proudfoot John
Robinson Regan John
Sharma Rajiv
Sun Sanxing
David Swinamer Alan
Takahoshi Hidenori
Original Assignee
Boehringer Ingelheim Pharmaceuticals, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharmaceuticals, Inc. filed Critical Boehringer Ingelheim Pharmaceuticals, Inc.
Publication of TR200102817T2 publication Critical patent/TR200102817T2/tr

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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
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    • A—HUMAN NECESSITIES
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    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/36—Radicals substituted by singly-bound nitrogen atoms
    • C07D213/38—Radicals substituted by singly-bound nitrogen atoms having only hydrogen or hydrocarbon radicals attached to the substituent nitrogen atom
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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
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  • Urology & Nephrology (AREA)
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Abstract

Bu patent içinde kronik inflamatuar hastaliklar gibi inflamasyon yapan hastaliklarin veya patolojik durumlarin tedavisinde yararli yeni aromatik bilesikler yer almaktadir. Ayrica bu bilesikleri içeren farmasötik bilesimler ve bu bilesiklerin hazirlanmasi islemleri de yer almaktadir.
TR2001/02817T 1999-03-12 2000-02-16 Antiinflamatuar ajanlar olarak faydalı bileşikler TR200102817T2 (tr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US12414899P 1999-03-12 1999-03-12
US16586799P 1999-11-16 1999-11-16

Publications (1)

Publication Number Publication Date
TR200102817T2 true TR200102817T2 (tr) 2002-05-21

Family

ID=26822256

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2001/02817T TR200102817T2 (tr) 1999-03-12 2000-02-16 Antiinflamatuar ajanlar olarak faydalı bileşikler

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US (5) US6358945B1 (tr)
EP (1) EP1165516B1 (tr)
JP (1) JP4820488B2 (tr)
KR (1) KR100709497B1 (tr)
CN (2) CN1511830A (tr)
AR (1) AR028473A1 (tr)
AT (1) ATE278674T1 (tr)
AU (1) AU771273B2 (tr)
BG (1) BG65159B1 (tr)
BR (1) BR0008922A (tr)
CA (1) CA2362003C (tr)
CO (1) CO5251387A1 (tr)
CZ (1) CZ20013289A3 (tr)
DE (1) DE60014603T2 (tr)
DK (1) DK1165516T3 (tr)
EE (1) EE04799B1 (tr)
ES (1) ES2225095T3 (tr)
HK (1) HK1043127B (tr)
HR (1) HRP20010665A2 (tr)
HU (1) HUP0202248A3 (tr)
ID (1) ID30176A (tr)
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PT (1) PT1165516E (tr)
RU (1) RU2242474C2 (tr)
SG (1) SG142120A1 (tr)
SI (1) SI1165516T1 (tr)
SK (1) SK12832001A3 (tr)
TR (1) TR200102817T2 (tr)
UY (1) UY26058A1 (tr)
WO (1) WO2000055139A2 (tr)
YU (1) YU64701A (tr)

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