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TN2009000312A1 - Fused ring compounds as partial agonists of ppar-gamma - Google Patents

Fused ring compounds as partial agonists of ppar-gamma

Info

Publication number
TN2009000312A1
TN2009000312A1 TNP2009000312A TN2009000312A TN2009000312A1 TN 2009000312 A1 TN2009000312 A1 TN 2009000312A1 TN P2009000312 A TNP2009000312 A TN P2009000312A TN 2009000312 A TN2009000312 A TN 2009000312A TN 2009000312 A1 TN2009000312 A1 TN 2009000312A1
Authority
TN
Tunisia
Prior art keywords
ppar
gamma
fused ring
partial agonists
ring compounds
Prior art date
Application number
TNP2009000312A
Other languages
English (en)
Inventor
Taisuko Tawaraishi
Hiroshi Imoto
Nobuo Cho
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39523585&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TN2009000312(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of TN2009000312A1 publication Critical patent/TN2009000312A1/fr

Links

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
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    • C07—ORGANIC CHEMISTRY
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10—Spiro-condensed systems
    • C07D491/113—Spiro-condensed systems with two or more oxygen atoms as ring hetero atoms in the oxygen-containing ring

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Biomedical Technology (AREA)
  • Rheumatology (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pain & Pain Management (AREA)
  • Oncology (AREA)
  • Otolaryngology (AREA)
  • Emergency Medicine (AREA)
  • Epidemiology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Psychology (AREA)
  • Dermatology (AREA)
  • Gastroenterology & Hepatology (AREA)
TNP2009000312A 2007-02-09 2009-07-30 Fused ring compounds as partial agonists of ppar-gamma TN2009000312A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2007031221 2007-02-09
PCT/JP2008/052217 WO2008099794A1 (fr) 2007-02-09 2008-02-05 Composés à cycles fusionnés utiles en tant qu'agonistes partiels de ppar-gamma

Publications (1)

Publication Number Publication Date
TN2009000312A1 true TN2009000312A1 (en) 2010-12-31

Family

ID=39523585

Family Applications (1)

Application Number Title Priority Date Filing Date
TNP2009000312A TN2009000312A1 (en) 2007-02-09 2009-07-30 Fused ring compounds as partial agonists of ppar-gamma

Country Status (21)

Country Link
US (2) US20110009384A1 (fr)
EP (1) EP2118066A1 (fr)
JP (1) JP2010517935A (fr)
KR (1) KR20090106660A (fr)
CN (1) CN101646653A (fr)
AR (1) AR065206A1 (fr)
AU (1) AU2008215490A1 (fr)
BR (1) BRPI0807014A2 (fr)
CA (1) CA2677736A1 (fr)
CL (1) CL2008000377A1 (fr)
CR (1) CR10991A (fr)
DO (1) DOP2009000202A (fr)
EA (1) EA200970746A1 (fr)
EC (1) ECSP099618A (fr)
IL (1) IL200114A0 (fr)
MA (1) MA31189B1 (fr)
MX (1) MX2009008103A (fr)
PE (1) PE20090068A1 (fr)
TN (1) TN2009000312A1 (fr)
TW (1) TW200838515A (fr)
WO (1) WO2008099794A1 (fr)

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EP2351743A4 (fr) 2008-10-27 2012-05-09 Takeda Pharmaceutical Composé bicyclique
EA020117B1 (ru) * 2008-11-14 2014-08-29 Консерт Фармасьютикалс Инк. Замещенные диоксопиперидинилфталимидные производные
US9045453B2 (en) 2008-11-14 2015-06-02 Concert Pharmaceuticals, Inc. Substituted dioxopiperidinyl phthalimide derivatives
WO2010076884A1 (fr) 2008-12-29 2010-07-08 武田薬品工業株式会社 Nouveau composé cyclique condensé et utilisation de celui-ci
JP5657578B2 (ja) 2009-06-09 2015-01-21 武田薬品工業株式会社 新規な縮合環化合物およびその用途
JP5732394B2 (ja) 2009-07-28 2015-06-10 武田薬品工業株式会社 錠剤
WO2011107494A1 (fr) 2010-03-03 2011-09-09 Sanofi Nouveaux dérivés aromatiques de glycoside, médicaments contenants ces composés, et leur utilisation
US8703758B2 (en) 2010-04-27 2014-04-22 Takeda Pharmaceutical Company Limited Bicyclic compound
WO2011158880A1 (fr) 2010-06-16 2011-12-22 武田薬品工業株式会社 Cristal de composé amide
EP2582709B1 (fr) 2010-06-18 2018-01-24 Sanofi Dérivés d'azolopyridin-3-one en tant qu'inhibiteurs de lipases et de phospholipases
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