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SV2007002007A - Compuestos de quinolina sustituidos ref. pc 25932a - Google Patents

Compuestos de quinolina sustituidos ref. pc 25932a

Info

Publication number
SV2007002007A
SV2007002007A SV2005002007A SV2005002007A SV2007002007A SV 2007002007 A SV2007002007 A SV 2007002007A SV 2005002007 A SV2005002007 A SV 2005002007A SV 2005002007 A SV2005002007 A SV 2005002007A SV 2007002007 A SV2007002007 A SV 2007002007A
Authority
SV
El Salvador
Prior art keywords
substituted quinoline
quinoline compounds
compounds ref
compounds
ref
Prior art date
Application number
SV2005002007A
Other languages
English (en)
Inventor
Peter Bertinato
Michel Andre Couturier
Ernest Seiichi Hamanaka
Marcus Douglas Ewing
Ralph Pelton Robinson Jr
Derek Lawrence Tickner
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of SV2007002007A publication Critical patent/SV2007002007A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)

Abstract

ESTA INVENCIÓN SE REFIERE A INHIBIDORES DE LA SECRECIÓN DE MTP/APO-B DE FORMULA (I) VER FORMULA DONDE R1-R7, X1, M Y N SON COMO SE HAN DEFINIDO EN LA MEMORIA DESCRIPTIVA, ASÍ COMO COMPOSICIONES FARMACÉUTICAS QUE COMPRENDEN LOS COMPUESTOS, A PROCEDIMIENTOS DE USO DE LOS COMPUESTO Y COMPOSICIONES. LOS COMPUESTOS DE LA INVENCIÓN SON ÚTILES EN EL TRATAMIENTO DE LA OBESIDAD Y ENFERMEDADES, AFECCIONES O TRASTORNOS ASOCIADOS
SV2005002007A 2004-02-04 2005-02-04 Compuestos de quinolina sustituidos ref. pc 25932a SV2007002007A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US54167804P 2004-02-04 2004-02-04
US63376304P 2004-12-06 2004-12-06

Publications (1)

Publication Number Publication Date
SV2007002007A true SV2007002007A (es) 2007-03-20

Family

ID=34890449

Family Applications (1)

Application Number Title Priority Date Filing Date
SV2005002007A SV2007002007A (es) 2004-02-04 2005-02-04 Compuestos de quinolina sustituidos ref. pc 25932a

Country Status (25)

Country Link
US (3) US7468378B2 (es)
EP (1) EP1716137A1 (es)
JP (1) JP2007520543A (es)
KR (1) KR100799802B1 (es)
AP (1) AP2006003685A0 (es)
AR (1) AR047529A1 (es)
AU (1) AU2005214159A1 (es)
BR (1) BRPI0507462A (es)
CA (1) CA2555133A1 (es)
CO (1) CO5700721A2 (es)
CR (1) CR8544A (es)
EA (1) EA010369B1 (es)
EC (1) ECSP066717A (es)
GE (1) GEP20084360B (es)
IL (2) IL176715A0 (es)
MA (1) MA28347A1 (es)
NL (1) NL1028192C2 (es)
NO (1) NO20063928L (es)
OA (1) OA13365A (es)
PA (1) PA8623001A1 (es)
PE (1) PE20050773A1 (es)
SV (1) SV2007002007A (es)
TW (2) TW200906800A (es)
UY (1) UY28734A1 (es)
WO (1) WO2005080373A1 (es)

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Also Published As

Publication number Publication date
AR047529A1 (es) 2006-01-25
IL208963A0 (en) 2011-07-31
US20070093525A1 (en) 2007-04-26
ECSP066717A (es) 2006-10-31
CO5700721A2 (es) 2006-11-30
OA13365A (en) 2007-04-13
KR20060127123A (ko) 2006-12-11
KR100799802B1 (ko) 2008-01-31
NL1028192A1 (nl) 2005-08-08
TW200906800A (en) 2009-02-16
US7468378B2 (en) 2008-12-23
US20050234099A1 (en) 2005-10-20
US7368573B2 (en) 2008-05-06
EA200601239A1 (ru) 2007-02-27
EP1716137A1 (en) 2006-11-02
MA28347A1 (fr) 2006-12-01
JP2007520543A (ja) 2007-07-26
US7393958B2 (en) 2008-07-01
PE20050773A1 (es) 2005-10-26
IL176715A0 (en) 2006-10-31
WO2005080373A1 (en) 2005-09-01
US20060223851A1 (en) 2006-10-05
NO20063928L (no) 2006-10-31
NL1028192C2 (nl) 2006-05-30
TW200533354A (en) 2005-10-16
AP2006003685A0 (en) 2006-08-31
UY28734A1 (es) 2005-09-30
AU2005214159A1 (en) 2005-09-01
TWI306454B (en) 2009-02-21
CR8544A (es) 2006-11-30
PA8623001A1 (es) 2006-03-24
BRPI0507462A (pt) 2007-07-10
GEP20084360B (en) 2008-04-29
EA010369B1 (ru) 2008-08-29
CA2555133A1 (en) 2005-09-01

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