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SK1912004A3 - Nicotinic acetylcholine receptor agonists in the treatment of restless legs syndrome - Google Patents

Nicotinic acetylcholine receptor agonists in the treatment of restless legs syndrome Download PDF

Info

Publication number
SK1912004A3
SK1912004A3 SK191-2004A SK1912004A SK1912004A3 SK 1912004 A3 SK1912004 A3 SK 1912004A3 SK 1912004 A SK1912004 A SK 1912004A SK 1912004 A3 SK1912004 A3 SK 1912004A3
Authority
SK
Slovakia
Prior art keywords
carbon atoms
alkyl
group
tricyclo
aza
Prior art date
Application number
SK191-2004A
Other languages
English (en)
Slovak (sk)
Inventor
Mario David Saltarelli
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of SK1912004A3 publication Critical patent/SK1912004A3/sk

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
SK191-2004A 2001-10-31 2002-10-21 Nicotinic acetylcholine receptor agonists in the treatment of restless legs syndrome SK1912004A3 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US33481001P 2001-10-31 2001-10-31
US33585801P 2001-11-26 2001-11-26
PCT/IB2002/004379 WO2003037329A1 (fr) 2001-10-31 2002-10-21 Agonistes du recepteur d'acetylcholine nicotinique pour traiter les impatiences des membres inferieurs

Publications (1)

Publication Number Publication Date
SK1912004A3 true SK1912004A3 (en) 2004-09-08

Family

ID=26989404

Family Applications (1)

Application Number Title Priority Date Filing Date
SK191-2004A SK1912004A3 (en) 2001-10-31 2002-10-21 Nicotinic acetylcholine receptor agonists in the treatment of restless legs syndrome

Country Status (14)

Country Link
EP (1) EP1439836A1 (fr)
JP (1) JP2005507411A (fr)
KR (1) KR20050038583A (fr)
CN (1) CN1568184A (fr)
BR (1) BR0213696A (fr)
CA (1) CA2460118A1 (fr)
CZ (1) CZ2004524A3 (fr)
HU (1) HUP0401967A2 (fr)
IL (1) IL160967A0 (fr)
MX (1) MXPA04002539A (fr)
PL (1) PL370549A1 (fr)
SK (1) SK1912004A3 (fr)
TW (1) TW200300139A (fr)
WO (1) WO2003037329A1 (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2006528237A (ja) * 2003-05-20 2006-12-14 ファイザー・プロダクツ・インク バレニクリンの医薬組成物
MXPA06003043A (es) 2003-09-17 2006-05-31 Xenoport Inc Tratamiento o prevencion del sindrome piernas inquietas utilizando prodrogas de analogos gaba.
CA2622755C (fr) 2005-10-07 2017-01-31 Exelixis, Inc. Azetidines en tant qu'inhibiteurs de mek
EP2101759B1 (fr) 2006-12-14 2018-10-10 Exelixis, Inc. Procédés d'utilisation d'inhibiteurs de mek
ES2880399T3 (es) 2012-07-27 2021-11-24 Neurodyn Life Sciences Inc Biodisponibilidad cerebral mejorada de galantamina mediante formulaciones seleccionadas y administración transmucosa de profármacos lipofílicos
HK1206242A1 (en) * 2012-07-27 2016-01-08 神经动力生命科学公司 Enhanced brain bioavailability of galantamine by selected formulations and transmucosal administration of lipophilic prodrugs
GEP201706690B (en) 2012-10-12 2017-06-26 Exelixis Inc Novel process for making compounds for use in treatment of cancer
US10568852B2 (en) * 2015-05-22 2020-02-25 Helmholtz Zentrum Munchen - Deutsches Forschungszentrum Fur Gesundheit Und Umwelt (Gmbh) Combination compositions and their use in methods for treating obesity and obesity-related disorders
WO2018236957A1 (fr) * 2017-06-20 2018-12-27 Nexien Biopharma, Inc. Procédé et compositions permettant de traiter le syndrome des jambes sans repos

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6020335A (en) * 1997-02-06 2000-02-01 Pfizer Inc (N-(pyridinylmethyl)-heterocyclic)ylideneamine compounds as nicotinic acetylcholine receptor binding agents
US5977131A (en) * 1997-04-09 1999-11-02 Pfizer Inc. Azaindole-ethylamine derivatives as nicotinic acetylcholine receptor binding agents
US6605610B1 (en) * 1997-12-31 2003-08-12 Pfizer Inc Aryl fused azapolycyclic compounds
EP0955301A3 (fr) * 1998-04-27 2001-04-18 Pfizer Products Inc. Dérivés de 7-aza-bicyclo[2.2.1]-heptane, leur préparation et utilisation sur la base d'affinité pour les recepteurs de l'acetylcholine nicotinique neuronaux
KR100420423B1 (ko) * 1998-04-29 2004-03-04 화이자 프로덕츠 인코포레이티드 아릴 축합된 아자 다환식 화합물

Also Published As

Publication number Publication date
KR20050038583A (ko) 2005-04-27
IL160967A0 (en) 2004-08-31
PL370549A1 (en) 2005-05-30
HUP0401967A2 (hu) 2005-01-28
EP1439836A1 (fr) 2004-07-28
CA2460118A1 (fr) 2003-05-08
MXPA04002539A (es) 2004-05-31
CN1568184A (zh) 2005-01-19
TW200300139A (en) 2003-05-16
WO2003037329A1 (fr) 2003-05-08
CZ2004524A3 (cs) 2004-07-14
JP2005507411A (ja) 2005-03-17
BR0213696A (pt) 2004-10-26

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