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PT82678B - Processo para a preparacao de compostos de cinolina - Google Patents

Processo para a preparacao de compostos de cinolina

Info

Publication number
PT82678B
PT82678B PT82678A PT8267886A PT82678B PT 82678 B PT82678 B PT 82678B PT 82678 A PT82678 A PT 82678A PT 8267886 A PT8267886 A PT 8267886A PT 82678 B PT82678 B PT 82678B
Authority
PT
Portugal
Prior art keywords
cyininine
compounds
preparation
cyininine compounds
Prior art date
Application number
PT82678A
Other languages
English (en)
Other versions
PT82678A (en
Original Assignee
Ici America Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ici America Inc filed Critical Ici America Inc
Publication of PT82678A publication Critical patent/PT82678A/pt
Publication of PT82678B publication Critical patent/PT82678B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/26Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings condensed with carbocyclic rings or ring systems
    • C07D237/28Cinnolines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/18Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804Compounds having Si-O-C linkages

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
PT82678A 1985-05-30 1986-05-30 Processo para a preparacao de compostos de cinolina PT82678B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB858513639A GB8513639D0 (en) 1985-05-30 1985-05-30 Cinnoline compounds

Publications (2)

Publication Number Publication Date
PT82678A PT82678A (en) 1986-06-01
PT82678B true PT82678B (pt) 1988-03-03

Family

ID=10579908

Family Applications (1)

Application Number Title Priority Date Filing Date
PT82678A PT82678B (pt) 1985-05-30 1986-05-30 Processo para a preparacao de compostos de cinolina

Country Status (25)

Country Link
US (1) US4886800A (pt)
EP (1) EP0205272B1 (pt)
JP (1) JPH0713062B2 (pt)
KR (1) KR900004402B1 (pt)
CN (1) CN1014060B (pt)
AR (1) AR242026A1 (pt)
AT (1) ATE66215T1 (pt)
AU (1) AU592086B2 (pt)
CA (1) CA1309406C (pt)
DE (1) DE3680828D1 (pt)
DK (1) DK162221C (pt)
ES (3) ES8801803A1 (pt)
FI (1) FI85584C (pt)
GB (2) GB8513639D0 (pt)
GR (1) GR861411B (pt)
HU (1) HU199433B (pt)
IE (1) IE58782B1 (pt)
IL (1) IL78992A0 (pt)
MW (1) MW4386A1 (pt)
NO (1) NO171592C (pt)
PH (1) PH23518A (pt)
PL (1) PL149227B1 (pt)
PT (1) PT82678B (pt)
SU (1) SU1500158A3 (pt)
ZA (1) ZA863664B (pt)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8702288D0 (en) * 1987-02-02 1987-03-11 Erba Farmitalia Cinnoline-carboxamides
ATE79540T1 (de) * 1988-02-09 1992-09-15 Ici America Inc Pharmazeutische zusammensetzung.
US4925844A (en) * 1988-02-09 1990-05-15 Ici Americas Inc. Antagonizing the pharmacological effects of a benzodiazepine receptor agonist
IL112235A (en) * 1994-01-03 2000-06-29 Acea Pharm Inc 1,4-dihydro-pyrido¬2,3-b¾pyrazine-2,3-dione (5 or 8) oxide derivatives and pharmaceutical compositions containing them
HK1054235A1 (zh) 2000-03-21 2003-11-21 法玛西雅厄普约翰美国公司 作为抗病毒药的4-氧-1,4-二氢[1,8]-二氮杂萘-3-甲酰胺类
BR0109391A (pt) 2000-03-21 2003-06-03 Upjohn Co 4-hidroxicinolina-3-carboxiamidas como agentes antivirais
ES2208581T3 (es) 2000-03-21 2004-06-16 PHARMACIA & UPJOHN COMPANY 4-oxo-1,4-dihydro-3-cinolincarboxamidas como agentes antivirales.
JP2003528102A (ja) 2000-03-21 2003-09-24 ファルマシア・アンド・アップジョン・カンパニー 抗ウイルス剤としての4−ヒドロキシ−1,8−ナフチリジン−3−カルボキサミド
US7465795B2 (en) * 2005-12-20 2008-12-16 Astrazeneca Ab Compounds and uses thereof
RU2008122405A (ru) 2005-12-20 2010-01-27 Астразенека Аб (Se) Замещенные производные циннолина в качестве модуляторов гамма-рецепторов и способ их синтеза
TW200911760A (en) * 2007-06-19 2009-03-16 Astrazeneca Ab Compounds and uses thereof
WO2010123441A1 (en) * 2009-04-21 2010-10-28 Astrazeneca Ab Crystalline form of 4-amino-8-(2-fluoro-6-methoxy-phenyl)-n-propylcinnoline-3- carboxamide hydrogen sulphate, for treatment of anxiety disorders
WO2010123443A1 (en) * 2009-04-21 2010-10-28 Astrazeneca Ab Pharmaceutical composition comprising 4-amino-8-(2-fluoro-6-methoxy-phenyl)-n- propylcinnoline-3-carboxamide hydrogen sulphate.
WO2010123440A1 (en) * 2009-04-21 2010-10-28 Astrazeneca Ab Pharmaceutical composition comprising 4-amino-8-(2-fluoro-6-methoxy-phenyl)-n- propylcinnoline-3-carboxamide hydrogen sulphate and rate-controlling polymer
AU2012258977A1 (en) * 2011-05-23 2014-01-16 Imago Pharmaceuticals, Inc. Inhibitors of LRRK2 kinase activity
CN111905828B (zh) * 2020-08-24 2022-04-19 万华化学集团股份有限公司 一种萘基配体mof活性炭复合催化剂及其制备方法和用途

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3657241A (en) * 1970-03-12 1972-04-18 Dow Chemical Co Substituted cinnoline compounds
GB1306839A (en) * 1970-10-16 1973-02-14 Ici Ltd Pharmaceutical compositions
GB1474399A (en) * 1974-08-19 1977-05-25 Ici Ltd Cinnolin-3-yl carboxylic acids and derivatives thereof
US4085103A (en) * 1974-11-07 1978-04-18 Imperial Chemical Industries Limited 6-Substituted-4-hydroxycinnolin-3-yl-carboxylic acids and esters thereof
GB1472766A (en) * 1974-11-07 1977-05-04 Ici Ltd Hydroxycinnoline derivatives processes for their preparation and their use in pharmaceutical compositions
DD123525A1 (pt) * 1976-02-10 1977-01-05
US4379929A (en) * 1981-03-19 1983-04-12 Eli Lilly And Company 4(1H)-Oxocinnoline-3-carboxylic acid derivatives
US4729782A (en) * 1983-09-14 1988-03-08 Lafarge Coppee Pollen suppressant comprising a fused pyridazinone
GB8702288D0 (en) * 1987-02-02 1987-03-11 Erba Farmitalia Cinnoline-carboxamides

Also Published As

Publication number Publication date
NO171592B (no) 1992-12-28
IE861267L (en) 1986-11-30
NO171592C (no) 1993-04-07
AU5781986A (en) 1986-12-04
ES557790A0 (es) 1988-10-01
IL78992A0 (en) 1986-09-30
FI862315A7 (fi) 1986-12-01
GB8611419D0 (en) 1986-06-18
DK256386A (da) 1986-12-01
PH23518A (en) 1989-08-16
US4886800A (en) 1989-12-12
ES8801803A1 (es) 1988-02-16
ES8801903A1 (es) 1988-03-01
SU1500158A3 (ru) 1989-08-07
ES557522A0 (es) 1988-03-01
KR900004402B1 (ko) 1990-06-25
EP0205272A2 (en) 1986-12-17
EP0205272B1 (en) 1991-08-14
DK162221C (da) 1992-03-02
PT82678A (en) 1986-06-01
IE58782B1 (en) 1993-11-17
ZA863664B (en) 1987-03-25
HUT41012A (en) 1987-03-30
DK256386D0 (da) 1986-05-30
FI85584C (fi) 1992-05-11
HU199433B (en) 1990-02-28
DE3680828D1 (de) 1991-09-19
FI862315A0 (fi) 1986-05-30
GB8513639D0 (en) 1985-07-03
ATE66215T1 (de) 1991-08-15
PL149227B1 (en) 1990-01-31
CN86104358A (zh) 1987-04-01
CA1309406C (en) 1992-10-27
AR242026A1 (es) 1993-02-26
MW4386A1 (en) 1987-06-19
GR861411B (en) 1986-08-28
JPS61280483A (ja) 1986-12-11
NO862141L (no) 1986-12-01
CN1014060B (zh) 1991-09-25
DK162221B (da) 1991-09-30
KR860008986A (ko) 1986-12-19
ES8802611A1 (es) 1988-10-01
ES555546A0 (es) 1988-02-16
FI85584B (fi) 1992-01-31
EP0205272A3 (en) 1987-11-19
JPH0713062B2 (ja) 1995-02-15
AU592086B2 (en) 1990-01-04

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