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PE20081358A1 - Combinaciones farmacologicas para el tratamiento de enfermedades de la vias aereas - Google Patents

Combinaciones farmacologicas para el tratamiento de enfermedades de la vias aereas

Info

Publication number
PE20081358A1
PE20081358A1 PE2007001123A PE2007001123A PE20081358A1 PE 20081358 A1 PE20081358 A1 PE 20081358A1 PE 2007001123 A PE2007001123 A PE 2007001123A PE 2007001123 A PE2007001123 A PE 2007001123A PE 20081358 A1 PE20081358 A1 PE 20081358A1
Authority
PE
Peru
Prior art keywords
hydroxy
ethyl
alkyl
treatment
airway
Prior art date
Application number
PE2007001123A
Other languages
English (en)
Inventor
Ingo Konetzki
Thierry Bouyssou
Sabine Pestel
Andreas Schnapp
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of PE20081358A1 publication Critical patent/PE20081358A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/536Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with carbocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/06Antiabortive agents; Labour repressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/04Antipruritics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Cardiology (AREA)
  • Epidemiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Dermatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

SE REFIERE A UNA COMBINACION FARMACEUTICA QUE COMPRENDE A) UNO O VARIOS COMPUESTOS DE FORMULA (I), EN DONDE R1 Y R2 SON INDEPENDIENTEMENTE H, HALOGENO, ALQUILO(C1-C4) O JUNTOS SON ALQUILENO(C1-C6); R3 ES H, HALOGENO, OH, ALQUILO(C1-C4) U O-ALQUILO(C1-C4); SIENDO SELECCIONADOS: N-(5-{2-[1,1-DIMETIL-3-(4-METIL-2-OXO-4H-BENZO[d][1,3]OXAZIN-1-IL)-PROPILAMINO]-1-HIDROXI-ETIL}-2-HIDROXI-FENIL)-METANSULFONAMIDA, N-(5-{2-[3-(4-ETIL-2-OXO-4H-BENZO[d][1,3]OXAZIN-1-IL)-1,1-DIMETIL-PROPILAMINO]-1-HIDROXI-ETIL}-2-HIDROXI-FENIL)-METANSULFONAMIDA, ENTRE OTROS; Y B) UNO O VARIOS COMPUESTOS ACTIVOS SELECCIONADOS DE ANTICOLINERGICOS, INHIBIDORES DE PDE-IV, ESTEROIDES, ANTAGONISTAS LTD4 O INHIBIDORES DE EGFR. TAMBIEN SE REFIERE A UNA COMPOSICION FARMACEUTICA, BAJO UNA FORMA DE ADMINISTRACION SELECCIONADO DE POLVOS PARA INHALACION, AEROSOLES DOSIFICADORES CON GAS PROPELENTE, O SOLUCIONES O SUPENCIONES SIN GAS PROPELENTE PARA INHALACION, SIENDO UTILES EN EL TRATAMIENTO DE ENFERMEDADES OBSTRUCTIVAS E INFALMATORIAS DE LAS VIAS AEREAS
PE2007001123A 2006-08-22 2007-08-20 Combinaciones farmacologicas para el tratamiento de enfermedades de la vias aereas PE20081358A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP06119272 2006-08-22

Publications (1)

Publication Number Publication Date
PE20081358A1 true PE20081358A1 (es) 2008-10-31

Family

ID=38535607

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2007001123A PE20081358A1 (es) 2006-08-22 2007-08-20 Combinaciones farmacologicas para el tratamiento de enfermedades de la vias aereas

Country Status (20)

Country Link
US (1) US20080051392A1 (es)
EP (1) EP2094271A2 (es)
JP (1) JP2010501521A (es)
KR (1) KR20090047539A (es)
CN (1) CN101505757A (es)
AR (1) AR062475A1 (es)
AU (1) AU2007287536A1 (es)
BR (1) BRPI0715855A2 (es)
CA (1) CA2661496A1 (es)
CO (1) CO6150168A2 (es)
EA (1) EA200900269A1 (es)
EC (1) ECSP099080A (es)
IL (1) IL197125A0 (es)
MX (1) MX2009001355A (es)
NO (1) NO20090067L (es)
PE (1) PE20081358A1 (es)
TW (1) TW200817009A (es)
UY (1) UY30552A1 (es)
WO (1) WO2008023003A1 (es)
ZA (1) ZA200810828B (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102005008921A1 (de) * 2005-02-24 2006-08-31 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Arzneimittel zur Behandlung von Atemwegserkrankungen
US7423146B2 (en) * 2005-11-09 2008-09-09 Boehringer Ingelheim International Gmbh Process for the manufacturing of pharmaceutically active 3,1-benzoxazine-2-ones
PE20080610A1 (es) * 2006-08-22 2008-07-15 Boehringer Ingelheim Int Nuevos beta-agonistas enantiomericamente puros, procedimientos para su preparacion y uso como medicamentos
EP2093219A1 (de) 2008-02-22 2009-08-26 Boehringer Ingelheim International Gmbh Kristalline, enantiomerenreine Salzform eines Betamimetikums und dessen Verwendung als Arzneimittel
WO2011061527A1 (en) 2009-11-17 2011-05-26 Astrazeneca Ab Combinations comprising a glucocorticoid receptor modulator for the treatment of respiratory diseases
GB201016912D0 (en) 2010-10-07 2010-11-24 Astrazeneca Ab Novel combination

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3026534A1 (de) * 1980-07-12 1982-03-18 C.H. Boehringer Sohn, 6507 Ingelheim 3,1-benzoxazin-2-one, ihre herstellung und verwendung
US4570630A (en) * 1983-08-03 1986-02-18 Miles Laboratories, Inc. Medicament inhalation device
FI88112C (fi) * 1985-07-30 1993-04-13 Glaxo Group Ltd Anordning foer administrering av laekemedel till patienter
EP1651222A1 (en) * 2003-07-29 2006-05-03 Boehringer Ingelheim International Gmbh Medicaments comprising pde iv inhibitors and an anticholinergic for treating respiratory disorders
DE102004048390A1 (de) * 2004-10-01 2006-04-06 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Pulverinhalativa auf Basis modifizierter Laktosemischungen als Hilfsstoff
DE102005008921A1 (de) * 2005-02-24 2006-08-31 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Arzneimittel zur Behandlung von Atemwegserkrankungen
US7423146B2 (en) * 2005-11-09 2008-09-09 Boehringer Ingelheim International Gmbh Process for the manufacturing of pharmaceutically active 3,1-benzoxazine-2-ones

Also Published As

Publication number Publication date
UY30552A1 (es) 2008-03-31
CA2661496A1 (en) 2008-02-28
BRPI0715855A2 (pt) 2013-07-30
ECSP099080A (es) 2009-02-27
ZA200810828B (en) 2009-11-25
US20080051392A1 (en) 2008-02-28
EA200900269A1 (ru) 2009-08-28
WO2008023003A8 (de) 2008-05-22
CN101505757A (zh) 2009-08-12
AR062475A1 (es) 2008-11-12
EP2094271A2 (de) 2009-09-02
KR20090047539A (ko) 2009-05-12
MX2009001355A (es) 2009-02-13
JP2010501521A (ja) 2010-01-21
AU2007287536A1 (en) 2008-02-28
WO2008023003A1 (de) 2008-02-28
NO20090067L (no) 2009-03-17
IL197125A0 (en) 2009-11-18
TW200817009A (en) 2008-04-16
CO6150168A2 (es) 2010-04-20

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