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PE20061363A1 - Derivados de 4-fenil-5-oxo-1,4,5,6,7,8-hexahidroquinolina como agonistas del receptor fsh - Google Patents

Derivados de 4-fenil-5-oxo-1,4,5,6,7,8-hexahidroquinolina como agonistas del receptor fsh

Info

Publication number
PE20061363A1
PE20061363A1 PE2006000464A PE2006000464A PE20061363A1 PE 20061363 A1 PE20061363 A1 PE 20061363A1 PE 2006000464 A PE2006000464 A PE 2006000464A PE 2006000464 A PE2006000464 A PE 2006000464A PE 20061363 A1 PE20061363 A1 PE 20061363A1
Authority
PE
Peru
Prior art keywords
oxo
phenyl
alkyl
bromo
propyl
Prior art date
Application number
PE2006000464A
Other languages
English (en)
Inventor
Poveda Pedro Manuel Grima
Karstens Willem Frederik Johan
Cornelis Marius Timmers
Original Assignee
Organon Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Organon Nv filed Critical Organon Nv
Publication of PE20061363A1 publication Critical patent/PE20061363A1/es

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Diabetes (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

SE REFIERE A UN COMPUESTO DE FORMULA I, DONDE R1 ES ALQUILO C1-C6, ALQUENILO C2-C6, ALQUINILO C2-C6, ENTRE OTROS; R2 Y R3 SON CADA UNO HALOGENO, ALQUILO C1-C4, ALQUENILO C2-C4, ALQUINILOXI C3-C4, ENTRE OTROS; R4 ES FENILO O HETEROARILO C2-C5, AMBOS SUSTITUIDOS CON R7 Y SUSTITUIDO O NO EN EL ANILLO HETEROAROMATICO CON 1 O MAS AMINO, HIDROXI, HALOGENO, NITRO, ENTRE OTROS; R7 ES H, ALQUILTIO C1-C4, ALQUILSULFONILO C1-C4, TRIFLUOROMETILSULFONILO, AMINOIMINOMETILO, ENTRE OTROS; X ES O, NH, AMINOALQUIL C1-C4, ENTRE OTROS; Y ES CH2, CO, SO2; Z ES CN, NO2. SON COMPUESTOS PREFERIDOS: N-{3-[2-BROMO-4-(3-CIANO-2-METIL-5-OXO-7-PROPIL-1,4,5,6,7,8-HEXAHIDROQUINOLIN-4-IL)-6-ETOXIFENOXIMETIL]-FENIL}-3,4,5-TRIMETOXIBENZAMIDA; 4-{3-BROMO-4-[3-(3,6-DIHIDRO-2H-PIRIDINA-1-CARBONIL)-BENCILOXI]-5-ETOXIFENIL}-2METIL-5-OXO-7-PROPIL-1,4,5,6,7,8-HEXAHIDRO-QUINOLINA-3-CARBONITRILO; N-{2-[2-BROMO-4-(3-CIANO-2-METIL-5-OXO-7-PROPIL-1,4,5,6,7,8-HEXAHIDROQUINOLIN-4-IL)-6-ETOXIMETOXIFENIL]-FENIL}-AMIDA DEL ACIDO FURANO-2-CARBOXILICO; ENTRE OTROS. REFERIDA TAMBIEN A UNA COMPOSICION FARMACEUTICA Y A UN PROCEDIMIENTO DE PREPARACION. DICHOS COMPUESTOS SON AGONISTAS DEL RECEPTOR DE FSH, UTILES EN EL TRATAMIENTO DE TRASTORNOS DE LA FERTILIDAD
PE2006000464A 2005-05-04 2006-05-03 Derivados de 4-fenil-5-oxo-1,4,5,6,7,8-hexahidroquinolina como agonistas del receptor fsh PE20061363A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP05103735 2005-05-04

Publications (1)

Publication Number Publication Date
PE20061363A1 true PE20061363A1 (es) 2007-01-15

Family

ID=34939693

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2006000464A PE20061363A1 (es) 2005-05-04 2006-05-03 Derivados de 4-fenil-5-oxo-1,4,5,6,7,8-hexahidroquinolina como agonistas del receptor fsh

Country Status (29)

Country Link
US (1) US8022218B2 (es)
EP (1) EP1881830B1 (es)
JP (1) JP5129737B2 (es)
KR (1) KR20080010426A (es)
CN (1) CN101212973B (es)
AR (1) AR057005A1 (es)
AT (1) ATE410166T1 (es)
AU (1) AU2006243868B2 (es)
BR (1) BRPI0611120A2 (es)
CA (1) CA2606683C (es)
CY (1) CY1108632T1 (es)
DE (1) DE602006003094D1 (es)
DK (1) DK1881830T3 (es)
ES (1) ES2314908T3 (es)
HR (1) HRP20080667T3 (es)
IL (1) IL186748A (es)
MX (1) MX2007013751A (es)
NO (1) NO20075617L (es)
NZ (1) NZ562686A (es)
PE (1) PE20061363A1 (es)
PL (1) PL1881830T3 (es)
PT (1) PT1881830E (es)
RS (1) RS50707B (es)
RU (1) RU2412170C2 (es)
SI (1) SI1881830T1 (es)
TW (1) TW200719894A (es)
UA (1) UA92007C2 (es)
WO (1) WO2006117368A1 (es)
ZA (1) ZA200709090B (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA92009C2 (ru) * 2005-05-04 2010-09-27 Н.В. Органон Производные 4-фенил-5-оксо-1,4,5,6,7,8-гексагидрохинолина для лечения бесплодия
JP4869336B2 (ja) * 2005-05-04 2012-02-08 ナームローゼ・フエンノートチヤツプ・オルガノン ジヒドロピリジン誘導体
UA92008C2 (en) * 2005-05-04 2010-09-27 Н.В. Органон 4-PHENYL-5-OXO-l,4,5,6,7,8-HEXAHYDROQUINOLINE DERIVATIVES AS MEDICAMENTS FOR THE TREATMENT OF INFERTILITY
TW200944523A (en) 2008-02-08 2009-11-01 Organon Nv (Dihydro)pyrrolo[2,1-a]isoquinolines
US8071587B2 (en) 2009-05-27 2011-12-06 N. V. Organon (Dihydro)imidazoiso[5,1-A]quinolines
TW201116531A (en) 2009-07-29 2011-05-16 Organon Nv Ring-annulated dihydropyrrolo[2,1-a]isoquinolines
US8431564B2 (en) 2009-07-29 2013-04-30 Merck Sharp & Dohme B.V. Ring-annulated dihydropyrrolo[2,1-α]isoquinolines
TW201116515A (en) 2009-07-31 2011-05-16 Organon Nv Dihydrobenzoindazoles
EP2694472B1 (en) 2011-04-05 2020-03-11 Takeda Pharmaceutical Company Limited Sulfonamide derivative and use thereof
US20150296779A1 (en) * 2012-11-28 2015-10-22 Stichting Dienst Landbouwkundig Onderzoek Substituted dihydropyridines for somatic embryogenesis in plants

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1070162B (de) 1959-12-03 Farbwerke Hoechst Aktiengesellschaft vormals Meister Lucius &. Brüning, Frankfurt/M Verfahren zur Herstellung von 5 - Brom - 3 - nitro - 4 - hydroxybenzaldehyd bzw. 5 - Chlor - 3 - nitro - 4 - hydroxybenzaldehyd
GB9318935D0 (en) * 1992-10-20 1993-10-27 Zeneca Ltd Heterocyclic derivatives
US5455253A (en) * 1992-10-20 1995-10-03 Zeneca Limited Heterocyclic derivatives
DE4430639A1 (de) 1994-08-29 1996-03-07 Bayer Ag Verwendung von 5-substituierten Pyridin- und Hexahydrochinolin-3-carbonsäurederivaten
GB9515445D0 (en) 1995-07-27 1995-09-27 Pharmacia Spa Dihydropyridine and pyridine derivatives and process for their preparation
WO1997014682A1 (en) * 1995-10-19 1997-04-24 Takeda Chemical Industries, Ltd. Quinoline derivatives as gnrh antagonists
US6593335B1 (en) * 1997-12-18 2003-07-15 Abbott Laboratories Potassium channel openers
US6235755B1 (en) 1998-08-07 2001-05-22 Applied Research Systems Ars Holding N.A. FSH mimetics for the treatment of infertility
EP1307193A1 (en) 2000-07-27 2003-05-07 Affymax Research Institute Agonists of follicle stimulating hormone activity
IL159288A0 (en) 2001-07-02 2004-06-01 Akzo Nobel Nv Tetrahydroquinoline derivatives
JP2003026630A (ja) 2001-07-13 2003-01-29 Taoka Chem Co Ltd カラーカプラー中間体用カルボン酸クロリド類の製造法
TWI322012B (en) 2002-12-20 2010-03-21 Organon Nv Tetrahydroquinoline derivatives
UA92009C2 (ru) 2005-05-04 2010-09-27 Н.В. Органон Производные 4-фенил-5-оксо-1,4,5,6,7,8-гексагидрохинолина для лечения бесплодия
JP4869336B2 (ja) 2005-05-04 2012-02-08 ナームローゼ・フエンノートチヤツプ・オルガノン ジヒドロピリジン誘導体
UA92008C2 (en) 2005-05-04 2010-09-27 Н.В. Органон 4-PHENYL-5-OXO-l,4,5,6,7,8-HEXAHYDROQUINOLINE DERIVATIVES AS MEDICAMENTS FOR THE TREATMENT OF INFERTILITY

Also Published As

Publication number Publication date
ES2314908T3 (es) 2009-03-16
CY1108632T1 (el) 2014-04-09
RU2007144989A (ru) 2009-06-10
JP2008540376A (ja) 2008-11-20
NO20075617L (no) 2007-12-03
ZA200709090B (en) 2008-09-25
DK1881830T3 (da) 2009-01-26
SI1881830T1 (sl) 2009-04-30
JP5129737B2 (ja) 2013-01-30
EP1881830B1 (en) 2008-10-08
CA2606683A1 (en) 2006-11-09
CN101212973A (zh) 2008-07-02
PL1881830T3 (pl) 2009-04-30
AU2006243868A1 (en) 2006-11-09
BRPI0611120A2 (pt) 2010-11-09
US20080275042A1 (en) 2008-11-06
RU2412170C2 (ru) 2011-02-20
PT1881830E (pt) 2008-12-10
MX2007013751A (es) 2008-01-24
NZ562686A (en) 2009-12-24
HK1110025A1 (en) 2008-07-04
AR057005A1 (es) 2007-11-07
AU2006243868B2 (en) 2011-06-16
CN101212973B (zh) 2011-11-16
UA92007C2 (ru) 2010-09-27
IL186748A0 (en) 2008-02-09
RS50707B (sr) 2010-06-30
DE602006003094D1 (de) 2008-11-20
KR20080010426A (ko) 2008-01-30
US8022218B2 (en) 2011-09-20
CA2606683C (en) 2013-11-12
IL186748A (en) 2011-08-31
EP1881830A1 (en) 2008-01-30
WO2006117368A1 (en) 2006-11-09
HRP20080667T3 (en) 2009-01-31
ATE410166T1 (de) 2008-10-15
TW200719894A (en) 2007-06-01

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