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PA8663901A1 - Derivados del (1,5-difenil-1h-pirazol-3-il)oxadiazol, su prepararacion y su aplicacion en terapéutica - Google Patents

Derivados del (1,5-difenil-1h-pirazol-3-il)oxadiazol, su prepararacion y su aplicacion en terapéutica

Info

Publication number
PA8663901A1
PA8663901A1 PA20068663901A PA8663901A PA8663901A1 PA 8663901 A1 PA8663901 A1 PA 8663901A1 PA 20068663901 A PA20068663901 A PA 20068663901A PA 8663901 A PA8663901 A PA 8663901A PA 8663901 A1 PA8663901 A1 PA 8663901A1
Authority
PA
Panama
Prior art keywords
difenil
pirazol
oxadiazol
therapeutics
derivatives
Prior art date
Application number
PA20068663901A
Other languages
English (en)
Inventor
Francis Barth
Christian Congy
Patrick Gueule
Murielle Rinaldi-Carmona
Broeck Didier Van
Original Assignee
Sanofi Aventis Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35079215&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PA8663901(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Aventis Sanofi Aventis filed Critical Sanofi Aventis Sanofi Aventis
Publication of PA8663901A1 publication Critical patent/PA8663901A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4245—Oxadiazoles
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Addiction (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Immunology (AREA)
  • Oncology (AREA)
  • Pulmonology (AREA)
  • Reproductive Health (AREA)
  • Obesity (AREA)
  • Communicable Diseases (AREA)
  • Vascular Medicine (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hospice & Palliative Care (AREA)
  • Child & Adolescent Psychology (AREA)

Abstract

LA PRESENTE INVENCION TINE COMO OBJETIVO COMPUESTOS QYE RESPONDEN A LA FORMULA: EN LA QUE: RI REPRESENTA UN RADICAL HETEROCICLICO ELEGIDO ENTRE: R2 REPRESENTA UN ALQUILO (C1-C5) O UN CIANO; R3 REPRESENTA UN FENILO NO SUSTITUIDO O SUSTITUIDO; R4 REPRESENTA UN FENILO NO SUSTITUIDO O SUSTITUIDO; ASI COMO SUS HIDRATOS O SUS SOLVATOS.
PA20068663901A 2005-02-21 2006-02-21 Derivados del (1,5-difenil-1h-pirazol-3-il)oxadiazol, su prepararacion y su aplicacion en terapéutica PA8663901A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0501860A FR2882365B1 (fr) 2005-02-21 2005-02-21 Derives de 2-(1,5-diphenyl-1h-pyrazol-3-yl)-1,3,4-oxadiazole leur preparation et leur application en therapeutique

Publications (1)

Publication Number Publication Date
PA8663901A1 true PA8663901A1 (es) 2006-12-07

Family

ID=35079215

Family Applications (1)

Application Number Title Priority Date Filing Date
PA20068663901A PA8663901A1 (es) 2005-02-21 2006-02-21 Derivados del (1,5-difenil-1h-pirazol-3-il)oxadiazol, su prepararacion y su aplicacion en terapéutica

Country Status (25)

Country Link
US (1) US7632852B2 (es)
EP (1) EP1853595A1 (es)
JP (1) JP4812778B2 (es)
KR (1) KR20070107053A (es)
CN (1) CN101119990A (es)
AR (1) AR055560A1 (es)
AU (1) AU2006215443A1 (es)
BR (1) BRPI0606845A2 (es)
CA (1) CA2597359A1 (es)
DO (1) DOP2006000045A (es)
EA (1) EA200701779A1 (es)
FR (1) FR2882365B1 (es)
GT (1) GT200600082A (es)
IL (1) IL185163A0 (es)
MA (1) MA29261B1 (es)
MX (1) MX2007009994A (es)
NO (1) NO20074763L (es)
NZ (1) NZ560790A (es)
PA (1) PA8663901A1 (es)
PE (1) PE20061038A1 (es)
SV (1) SV2007002422A (es)
TW (1) TW200640916A (es)
UY (1) UY29388A1 (es)
WO (1) WO2006087480A1 (es)
ZA (1) ZA200706953B (es)

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AU2007283113A1 (en) 2006-08-08 2008-02-14 Sanofi-Aventis Arylaminoaryl-alkyl-substituted imidazolidine-2,4-diones, processes for preparing them, medicaments comprising these compounds, and their use
KR101100028B1 (ko) * 2006-09-29 2011-12-29 주식회사 녹십자 칸나비노이드 ｃｂ1 수용체 길항제로서의 헤테로아릴-피라졸 유도체
US7875647B2 (en) 2006-09-29 2011-01-25 Green Cross Corporation Heteroaryl-pyrazole derivatives as cannabinoid CB1 receptor antagonists
US20080207704A1 (en) * 2007-02-27 2008-08-28 The Green Cross Corporation Heteroaryl-imidazole derivatives as cannabinoid cb1 receptor antagonists
US7705024B2 (en) 2007-04-12 2010-04-27 National Health Research Institutes Oxadiazole compounds
EP2025674A1 (de) 2007-08-15 2009-02-18 sanofi-aventis Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
WO2009078498A1 (en) * 2007-12-17 2009-06-25 Green Cross Corporation Biarylpyrazole 4-carboxamides as cannabinoid cb1 receptor ligands
UY31968A (es) 2008-07-09 2010-01-29 Sanofi Aventis Nuevos derivados heterocíclicos, sus procesos para su preparación, y sus usos terapéuticos
US8309584B2 (en) * 2008-09-25 2012-11-13 Green Cross Corporation Sulfur containing pyrazole-heterocycle derivatives as cannabinoid CB1 receptor antagonists
WO2010068601A1 (en) 2008-12-08 2010-06-17 Sanofi-Aventis A crystalline heteroaromatic fluoroglycoside hydrate, processes for making, methods of use and pharmaceutical compositions thereof
BR112012003973A2 (pt) 2009-08-26 2015-09-08 Sanofi Sa hidratos de fluoroglicosídeo heteroaromático cristalinos, produtos farmacêuticos compreendendo estes compostos e seu uso
US8933024B2 (en) 2010-06-18 2015-01-13 Sanofi Azolopyridin-3-one derivatives as inhibitors of lipases and phospholipases
WO2012120056A1 (de) 2011-03-08 2012-09-13 Sanofi Tetrasubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
EP2683705B1 (de) 2011-03-08 2015-04-22 Sanofi Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
WO2012120053A1 (de) 2011-03-08 2012-09-13 Sanofi Verzweigte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
WO2012120052A1 (de) 2011-03-08 2012-09-13 Sanofi Mit carbozyklen oder heterozyklen substituierte oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung
US8710050B2 (en) 2011-03-08 2014-04-29 Sanofi Di and tri- substituted oxathiazine derivatives, method for the production, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof
CN109651350B (zh) * 2019-01-11 2022-05-24 贵州大学 一类杂环取代的1,3,4-噁(噻)二唑类化合物及其制备方法和用途
CN109942567B (zh) * 2019-04-30 2023-04-07 贵州大学 一种1,3,4-噁(噻)二唑基的咪唑类化合物及其制备方法和用途

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WO2006087480A1 (fr) 2006-08-24
JP4812778B2 (ja) 2011-11-09
ZA200706953B (en) 2009-03-25
DOP2006000045A (es) 2006-11-15
US7632852B2 (en) 2009-12-15
MA29261B1 (fr) 2008-02-01
FR2882365A1 (fr) 2006-08-25
JP2008530188A (ja) 2008-08-07
AR055560A1 (es) 2007-08-22
KR20070107053A (ko) 2007-11-06
AU2006215443A1 (en) 2006-08-24
NZ560790A (en) 2009-08-28
MX2007009994A (es) 2007-10-10
TW200640916A (en) 2006-12-01
IL185163A0 (en) 2007-12-03
UY29388A1 (es) 2006-10-02
NO20074763L (no) 2007-11-16
EP1853595A1 (fr) 2007-11-14
GT200600082A (es) 2006-10-19
PE20061038A1 (es) 2006-11-24
SV2007002422A (es) 2007-01-17
CN101119990A (zh) 2008-02-06
CA2597359A1 (fr) 2006-08-24
FR2882365B1 (fr) 2007-09-07
EA200701779A1 (ru) 2008-02-28
US20080039510A1 (en) 2008-02-14

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