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AR065280A1 - Agentes antiparasitarios - Google Patents

Agentes antiparasitarios

Info

Publication number
AR065280A1
AR065280A1 ARP080100563A ARP080100563A AR065280A1 AR 065280 A1 AR065280 A1 AR 065280A1 AR P080100563 A ARP080100563 A AR P080100563A AR P080100563 A ARP080100563 A AR P080100563A AR 065280 A1 AR065280 A1 AR 065280A1
Authority
AR
Argentina
Prior art keywords
compounds
agents
tautomer
prodrug
antiparasitary
Prior art date
Application number
ARP080100563A
Other languages
English (en)
Inventor
Stuart Nicholas Comlay
Joanne Clare Hannam
William Howson
Christelle Lauret
Yogesh Anil Sabins
Original Assignee
Pfizer Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Ltd filed Critical Pfizer Ltd
Publication of AR065280A1 publication Critical patent/AR065280A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C381/00—Compounds containing carbon and sulfur and having functional groups not covered by groups C07C301/00 - C07C337/00
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N41/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a sulfur atom bound to a hetero atom
    • A01N41/12—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a sulfur atom bound to a hetero atom not containing sulfur-to-oxygen bonds, e.g. polysulfides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/166—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the carbon of a carboxamide group directly attached to the aromatic ring, e.g. procainamide, procarbazine, metoclopramide, labetalol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Agronomy & Crop Science (AREA)
  • Wood Science & Technology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pyridine Compounds (AREA)

Abstract

La presente se refiere a compuestos de formula (1) o un tautomero o profármaco de los mismos, o una sal farmacéuticamente aceptable de dicho compuesto, tautomero o profármaco, en la que R1, R2. R3, R4 y R5 se selecciona cada uno independientemente de H, halogeno, CN, CF3 y CONH2; composiciones que contienen dichos compuestos y a los usos de dichos compuestos como agentes antiparasitarios.
ARP080100563A 2007-02-09 2008-02-08 Agentes antiparasitarios AR065280A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US88904107P 2007-02-09 2007-02-09
US94682007P 2007-06-28 2007-06-28

Publications (1)

Publication Number Publication Date
AR065280A1 true AR065280A1 (es) 2009-05-27

Family

ID=39402647

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP080100563A AR065280A1 (es) 2007-02-09 2008-02-08 Agentes antiparasitarios

Country Status (21)

Country Link
US (2) US7608604B2 (es)
EP (1) EP2118055B1 (es)
JP (1) JP4592819B2 (es)
KR (2) KR20110098012A (es)
AR (1) AR065280A1 (es)
AU (1) AU2008212594C1 (es)
BR (1) BRPI0807137A2 (es)
CA (1) CA2676147C (es)
CL (1) CL2008000403A1 (es)
CO (1) CO6220853A2 (es)
CY (1) CY1114932T1 (es)
DK (1) DK2118055T3 (es)
ES (1) ES2435191T3 (es)
MX (1) MX2009007482A (es)
NZ (1) NZ578259A (es)
PL (1) PL2118055T3 (es)
PT (1) PT2118055E (es)
RU (1) RU2425825C2 (es)
TW (1) TWI352695B (es)
UY (1) UY30897A1 (es)
WO (1) WO2008096231A1 (es)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7361653B2 (en) * 2001-04-17 2008-04-22 Nihon Nohyaku Co., Ltd Pest control agent composition and method of using the same
NZ599754A (en) 2007-06-07 2013-10-25 Bayer Animal Health Gmbh Control of ectoparasites
MX2010001133A (es) * 2007-07-30 2010-03-01 Du Pont Metodo de control de pulgas.
JP5614853B2 (ja) 2008-10-21 2014-10-29 メリアル リミテッド チオアミド化合物、その製造方法及び使用方法
MY153715A (en) 2008-11-14 2015-03-13 Merial Ltd Enantiomerically enriched aryloazol-2-yl cyanoethylamino compounds, method of making and method of using thereof
CA2741338A1 (en) 2008-12-03 2010-06-10 Novartis Ag Amidoacetonitrile compounds and pesticidal composition thereof
GB0905365D0 (en) 2009-03-27 2009-05-13 Norbrook Lab Ltd A topical parasiticide composition
TWI510189B (zh) 2009-06-19 2015-12-01 Lilly Co Eli 殺外寄生蟲之方法及調配物
EP2314292A1 (en) * 2009-10-20 2011-04-27 Novartis AG Endoparasiticidal compositions
CN102711730B (zh) 2010-01-25 2015-06-17 伊莱利利公司 用于内部控制或治疗马类胃蝇幼虫的方法
TWI580442B (zh) * 2011-10-19 2017-05-01 傑特大學 醫藥毫微懸浮物
US8962681B2 (en) 2011-10-19 2015-02-24 Zoetis Llc Use of aminoacetonitrile derivatives against endoparasites
WO2013084860A1 (ja) * 2011-12-06 2013-06-13 宇部興産株式会社 ペンタフルオロスルファニル安息香酸の製造方法
US9539331B2 (en) * 2011-12-21 2017-01-10 Bayer Intellectual Property Gmbh Preparations containing amorphous emodepside
EP2796449A4 (en) * 2012-02-14 2015-11-18 Nippon Soda Co ARYLOXYACETAMIDE COMPOUND AND PESTICIDE THEREWITH
JP6220403B2 (ja) 2012-11-14 2017-10-25 イーライ リリー アンド カンパニー 有害外部寄生虫駆除方法及び製剤
WO2014146750A1 (de) 2013-03-22 2014-09-25 Merck Patent Gmbh Synthesebausteine für die herstellung von materialien für organische elektrolumineszenzvorrichtungen
CN104230743B (zh) * 2013-06-24 2017-02-08 海正药业南通有限公司 一种4-苄基-1-苯乙基哌嗪-2,6-二酮的制备方法
US20160368868A1 (en) * 2013-07-01 2016-12-22 Universite Zurich N-(1-cyano-2-hydroxy-1-methyl-ethyl)-4-(trifluoromethylsulfanyl)benzamide derivatives for use as nematocidal drugs
KR101960347B1 (ko) * 2015-02-12 2019-03-20 쯔지앙 하이썬 파머슈티컬 컴퍼니, 리미티드 프라지콴텔 및 이의 중간체 화합물의 제조방법
CN106018571A (zh) * 2015-11-09 2016-10-12 中华人民共和国淮安出入境检验检疫局 检测水生蔬菜中氯虫苯甲酰胺残留量的方法

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1643766A1 (de) * 1967-01-06 1971-07-01 Allied Chem Perhalogenierte Jodide sowie Verfahren zu ihrer Herstellung
GB9801851D0 (en) * 1998-01-29 1998-03-25 Pfizer Ltd Parasiticidal agents
US6239077B1 (en) 1998-05-01 2001-05-29 Nihon Nohyaku Co., Ltd. Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof
AU2002224942A1 (en) 2000-12-20 2002-07-01 Syngenta Participations Ag N-acyl aminoacetonitriles having pesticidal properties
AU3458802A (en) 2000-12-20 2002-07-01 Novartis Ag Organic compounds
AR035531A1 (es) 2001-01-22 2004-06-02 Novartis Ag Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos
DE10222192A1 (de) * 2002-05-18 2003-11-27 Aventis Pharma Gmbh Pentafluorsulfuranyl-benzoylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament
GB0402677D0 (en) * 2003-11-06 2004-03-10 Novartis Ag Organic compounds
DE10353205A1 (de) * 2003-11-13 2005-06-16 Aventis Pharma Deutschland Gmbh Ortho-substituierte Pentafluorsulfuranyl-Benzole, Verfahren zu ihrer Herstellung sowie ihre Verwendung als wertvolle Synthese-Zwischenstufen
US7514464B2 (en) * 2003-12-18 2009-04-07 Pfizer Limited Substituted arylpyrazoles
US7425580B2 (en) 2004-05-19 2008-09-16 Wyeth (Diaryl-methyl)-malononitriles and their use as estrogen receptor ligands
AR049391A1 (es) 2004-06-10 2006-07-26 Novartis Ag Derivados de aminoacetonitrilo y su uso para controlar parasitos en animales de sangre caliente
WO2006043654A1 (ja) 2004-10-22 2006-04-27 Nihon Nohyaku Co., Ltd. アセトニトリル誘導体及び有害生物防除剤並びにその使用方法
KR100878824B1 (ko) 2005-04-01 2009-01-14 엘지전자 주식회사 스케일러블 비디오 신호 인코딩 및 디코딩 방법

Also Published As

Publication number Publication date
AU2008212594A1 (en) 2008-08-14
MX2009007482A (es) 2009-08-13
KR20110098012A (ko) 2011-08-31
AU2008212594C1 (en) 2013-04-11
TWI352695B (en) 2011-11-21
KR101136251B1 (ko) 2012-04-25
UY30897A1 (es) 2008-09-30
RU2425825C2 (ru) 2011-08-10
JP4592819B2 (ja) 2010-12-08
ES2435191T3 (es) 2013-12-16
KR20090104856A (ko) 2009-10-06
PT2118055E (pt) 2013-11-19
NZ578259A (en) 2011-12-22
CA2676147A1 (en) 2008-08-14
WO2008096231A8 (en) 2009-08-20
CY1114932T1 (el) 2016-12-14
AU2008212594B2 (en) 2012-10-04
US7608604B2 (en) 2009-10-27
DK2118055T3 (da) 2013-11-04
JP2010518067A (ja) 2010-05-27
PL2118055T3 (pl) 2014-01-31
TW200843728A (en) 2008-11-16
US20080194694A1 (en) 2008-08-14
HK1133871A1 (en) 2010-04-09
CA2676147C (en) 2012-03-13
WO2008096231A1 (en) 2008-08-14
CO6220853A2 (es) 2010-11-19
EP2118055A1 (en) 2009-11-18
BRPI0807137A2 (pt) 2014-04-15
EP2118055B1 (en) 2013-08-21
CL2008000403A1 (es) 2008-08-18
US20100010093A1 (en) 2010-01-14
RU2009127356A (ru) 2011-03-20

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