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IN2003KO00001A - - Google Patents

Info

Publication number
IN2003KO00001A
IN2003KO00001A IN1KO2003A IN2003KO00001A IN 2003KO00001 A IN2003KO00001 A IN 2003KO00001A IN 1KO2003 A IN1KO2003 A IN 1KO2003A IN 2003KO00001 A IN2003KO00001 A IN 2003KO00001A
Authority
IN
India
Application number
Other languages
English (en)
Inventor
Mark R Schmitt
Donald R Kirsch
Jane E Harris
Carl F Beyer
Klaus-Juergen Pees
Paul Carter
Waldemar Pfrengle
Guido Albert
Original Assignee
American Home Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Home Prod filed Critical American Home Prod
Publication of IN2003KO00001A publication Critical patent/IN2003KO00001A/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IN1KO2003 2000-06-30 2003-01-01 IN2003KO00001A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US21558500P 2000-06-30 2000-06-30

Publications (1)

Publication Number Publication Date
IN2003KO00001A true IN2003KO00001A (fr) 2005-12-02

Family

ID=22803554

Family Applications (1)

Application Number Title Priority Date Filing Date
IN1KO2003 IN2003KO00001A (fr) 2000-06-30 2003-01-01

Country Status (24)

Country Link
US (1) US7329663B2 (fr)
EP (1) EP1307200A2 (fr)
JP (1) JP2004502691A (fr)
KR (1) KR20030013475A (fr)
CN (1) CN1592624A (fr)
AR (1) AR034553A1 (fr)
AU (2) AU7306201A (fr)
BG (1) BG107277A (fr)
BR (1) BR0112038A (fr)
CA (1) CA2413802A1 (fr)
CZ (1) CZ20024150A3 (fr)
EA (1) EA006483B1 (fr)
GE (1) GEP20053688B (fr)
HK (1) HK1052646A1 (fr)
HU (1) HUP0300798A3 (fr)
IL (1) IL152869A0 (fr)
IN (1) IN2003KO00001A (fr)
MX (1) MXPA02011913A (fr)
NO (1) NO20026195L (fr)
NZ (1) NZ523807A (fr)
PL (1) PL360027A1 (fr)
SK (1) SK18412002A3 (fr)
WO (1) WO2002002563A2 (fr)
ZA (1) ZA200300793B (fr)

Families Citing this family (49)

* Cited by examiner, † Cited by third party
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US6255309B1 (en) 1999-03-19 2001-07-03 American Cyanomid Co. Fungicidal trifluoromethylalkylamino-triazolopyrimidines
AU2002221831A1 (en) * 2000-11-13 2002-05-21 Basf Aktiengesellschaft 7-(r)-amino-triazolopyrimidines, the production thereof and use of the same for combating phytopathogenic fungi
JP2004526767A (ja) * 2001-04-11 2004-09-02 ビーエーエスエフ アクチェンゲゼルシャフト ６−（２−クロロ−６−フルオロ−フェニル）−トリアゾロピリミジン類
NZ528745A (en) * 2001-04-11 2005-03-24 Basf Ag 5-halogen-6-phenyl-7-fluoralkylamino-triazolopyrimidines as fungicides and their preparation process
DE10121101A1 (de) * 2001-04-27 2002-10-31 Bayer Ag Triazolopyrimidine
DE10121162A1 (de) * 2001-04-30 2002-10-31 Bayer Ag Triazolopyrimidine
DE10124208A1 (de) † 2001-05-18 2002-11-21 Bayer Ag Verwendung von Triazolopyrimidin-Derivaten als Mikrobizide
WO2003008417A1 (fr) * 2001-07-18 2003-01-30 Basf Aktiengesellschaft 6-(2-tolyl)-triazolopyrimidines substituees comme fongicides
PL372978A1 (en) 2002-03-21 2005-08-08 Basf Aktiengesellschaft Fungicidal triazolopyrimidines, methods for producing the same, use thereof for combating harmful fungi and agents containing said substances
JPWO2004011467A1 (ja) * 2002-07-29 2005-12-15 北興化学工業株式会社 トリアゾロピリミジン誘導体および農園芸用殺菌剤
UA80304C2 (en) * 2002-11-07 2007-09-10 Basf Ag Substituted 6-(2-halogenphenyl)triazolopyrimidines
MXPA05009338A (es) * 2003-03-31 2005-11-04 Basf Ag 7-alquenilamino-triazolopirimidinas, procedimientos para su obtencion y el uso de las mismas para controlar hongos nocivos, asi como productos que los contienen.
US20070275961A1 (en) * 2003-06-04 2007-11-29 Vernalis (Cambridge) Limited. Triazolo ' 1, 5-A ! Pyrimidines and Their Use in Medicine
DE10325133A1 (de) * 2003-06-04 2004-12-23 Bayer Cropscience Ag Triazolopyrimidine
DE10328173A1 (de) * 2003-06-24 2005-01-13 Bayer Cropscience Ag Triazolopyrimidine
DE10328171A1 (de) * 2003-06-24 2005-01-13 Bayer Cropscience Ag Triazolopyrimidine
DE10328481A1 (de) * 2003-06-25 2005-01-13 Bayer Ag Triazolopyrimidine
US7419982B2 (en) 2003-09-24 2008-09-02 Wyeth Holdings Corporation Crystalline forms of 5-chloro-6-{2,6-difluoro-4-[3-(methylamino)propoxy]phenyl}-N-[(1S)-2,2,2-trifluoro-1-methylethyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine salts
DE602004014525D1 (de) * 2003-09-24 2008-07-31 Wyeth Corp 6-aryl-7-halo-imidazoä1,2-aüpyrimidine als mittel gegen krebs
WO2005030775A1 (fr) * 2003-09-24 2005-04-07 Wyeth Holdings Corporation 6-[(substitutees)phenyl]triazolopyrimidines utilisees en tant qu'agent anticancereux
EP1674454A4 (fr) * 2003-10-17 2006-12-27 Nippon Kayaku Kk Derive 2-amino- 1,2,4|triazolo 1,5-a|pyrimidine substitue et utilisation de ce derive
JP4606015B2 (ja) * 2003-11-25 2011-01-05 日本化薬株式会社 ［１，２，４］トリアゾロ［１，５−ａ］ピリミジン誘導体の新規医薬用途
MY179926A (en) 2003-12-08 2020-11-19 Wyeth Corp Process for the preparation of tubulin inhibitors
CN1890243A (zh) * 2003-12-17 2007-01-03 巴斯福股份公司 6－(2,4,6－三卤代苯基)三唑并嘧啶、其制备方法及其在防治病原性真菌中的用途以及包含所述物质的组合物
JP2007514678A (ja) * 2003-12-17 2007-06-07 ビーエーエスエフ　アクチェンゲゼルシャフト ６−（２，３，６−トリフルオロフェニル）トリアゾロピリミジン、その調製および有害真菌防除のためのその使用、ならびに当該化合物を含んでなる組成物
EP1732927A2 (fr) * 2004-03-30 2006-12-20 Basf Aktiengesellschaft 6-(2-fluorophenyl)-triazolopyrimidines, procede de production desdits composes, leur utilisation dans la lutte contre des champignons parasites et des agents contenant lesdits composes
JP2007538028A (ja) * 2004-05-17 2007-12-27 ビーエーエスエフ　アクチェンゲゼルシャフト トリアゾロピリミジン化合物および病原菌を制御するためのそれらの使用
WO2005120233A1 (fr) * 2004-06-09 2005-12-22 Basf Aktiengesellschaft Composes de triazolopyrimidine et leur utilisation pour lutter contre des champignons nocifs
JP2008503538A (ja) * 2004-06-25 2008-02-07 ビーエーエスエフ　アクチェンゲゼルシャフト トリアゾロピリミジン化合物およびそれらの病原性菌類を防除するための使用
EA013525B1 (ru) * 2005-05-20 2010-06-30 Алантос-Фармасьютикалз Холдинг, Инк. Гетеробициклические ингибиторы металлопротеазы и их применение
US20070155738A1 (en) * 2005-05-20 2007-07-05 Alantos Pharmaceuticals, Inc. Heterobicyclic metalloprotease inhibitors
WO2007011759A2 (fr) * 2005-07-15 2007-01-25 Kalypsys, Inc. Inhibiteurs de la kinesine mitotique
CN101370813A (zh) * 2005-12-16 2009-02-18 惠氏公司 用作抗癌药物的6-[(取代的)苯基]三唑并嘧啶类的二聚体和加合物
AR059649A1 (es) * 2006-02-28 2008-04-16 Basf Ag 6- fenil 7-amino - amino (1,2,4) -triazolo (1,5-a) pirimidinas y su su uso para el combate de hongos daninos
WO2007116011A2 (fr) * 2006-04-10 2007-10-18 Basf Se Triazolopyrimidines substituées, procédé de fabrication, utilisation dans la lutte contre des champignons parasites et agent contenant ces composés
JP5231829B2 (ja) 2007-02-15 2013-07-10 石原産業株式会社 ピリジル−トリアゾロピリミジン誘導体又はその塩、それらを含有する有害生物防除剤並びにそれらの製造方法
NZ583267A (en) 2007-08-14 2012-03-30 Bayer Schering Pharma Ag Fused bicyclic pyrimidines
CN103889428A (zh) * 2010-10-04 2014-06-25 肝炎与病毒研究所 乙型肝炎病毒抗原分泌的新型抑制剂
JP6311603B2 (ja) * 2012-06-22 2018-04-18 住友化学株式会社 縮合複素環化合物
CN103360398B (zh) * 2013-07-22 2015-03-25 山东大学 一种三唑并嘧啶类hiv-1逆转录酶抑制剂及其制备方法与应用
GB201504565D0 (en) 2015-03-18 2015-05-06 Takeda Pharmaceutical Novel compounds
KR101995533B1 (ko) * 2017-03-21 2019-07-02 한국화학연구원 [1,2,4]트리아졸로[4,3-a]퀴노잘린 아미노 페닐 유도체 또는 이의 약학적으로 허용가능한 염, 이의 제조방법 및 이를 유효성분으로 포함하는 BET 단백질 관련 질환의 예방 또는 치료용 약학적 조성물
US11390626B2 (en) 2019-01-29 2022-07-19 Tosk, Inc. Pyrazolopyrimidine modulators of RAS GTPase
US20230167121A1 (en) * 2020-04-14 2023-06-01 The Trustees Of The University Of Pennsylvania Substituted {1,2,4,} triazolo{1,5-a} pyrimidine compounds and use in stabilizing microtubules
AU2021264550A1 (en) * 2020-05-01 2022-11-17 Gilead Sciences, Inc. CD73 inhibiting 2,4-dioxopyrimidine compounds
US20230279006A1 (en) * 2020-07-08 2023-09-07 Klotho Therapeutics, Inc. Novel compounds and methods for increasing klotho gene expression
US12180220B2 (en) 2020-10-14 2024-12-31 Tosk, Inc. Heteroaryl modulators of RAS GTPase
US11919869B2 (en) 2021-10-29 2024-03-05 Gilead Sciences, Inc. CD73 compounds
CN118475581A (zh) * 2022-01-25 2024-08-09 瑞石生物医药有限公司 一种ccr4小分子拮抗剂及其用途

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US5994360A (en) * 1997-07-14 1999-11-30 American Cyanamid Company Fungicidal 5-alkyl-triazolopyrimidines
US6020338A (en) * 1998-02-11 2000-02-01 American Cyanamid Company Fungicidal 7-alkyl-triazolopyrimidines
US6380202B1 (en) * 1998-09-25 2002-04-30 Basf Aktiengesellschaft Fungicidal fluoro-substituted 7-heterocyclyl-triazolopyrimidines
FR2784380B1 (fr) * 1998-09-25 2002-09-06 American Cyanamid Co Triazolopyrimidines 7-oxy- et 7-thio-substituees fongicides
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MY125533A (en) * 1999-12-06 2006-08-30 Bristol Myers Squibb Co Heterocyclic dihydropyrimidine compounds
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DE10121101A1 (de) * 2001-04-27 2002-10-31 Bayer Ag Triazolopyrimidine
DE10121102A1 (de) * 2001-04-27 2002-11-07 Bayer Ag Triazolopyrimidine
DE10121162A1 (de) * 2001-04-30 2002-10-31 Bayer Ag Triazolopyrimidine
US7037902B2 (en) * 2002-07-03 2006-05-02 Receptron, Inc. Affinity small molecules for the EPO receptor
US7419982B2 (en) * 2003-09-24 2008-09-02 Wyeth Holdings Corporation Crystalline forms of 5-chloro-6-{2,6-difluoro-4-[3-(methylamino)propoxy]phenyl}-N-[(1S)-2,2,2-trifluoro-1-methylethyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine salts
WO2005030775A1 (fr) * 2003-09-24 2005-04-07 Wyeth Holdings Corporation 6-[(substitutees)phenyl]triazolopyrimidines utilisees en tant qu'agent anticancereux

Also Published As

Publication number Publication date
SK18412002A3 (sk) 2003-06-03
JP2004502691A (ja) 2004-01-29
NO20026195D0 (no) 2002-12-23
PL360027A1 (en) 2004-09-06
EA200300091A1 (ru) 2003-08-28
CA2413802A1 (fr) 2002-01-10
CN1592624A (zh) 2005-03-09
ZA200300793B (en) 2004-07-20
HK1052646A1 (zh) 2003-09-26
EA006483B1 (ru) 2005-12-29
IL152869A0 (en) 2003-06-24
KR20030013475A (ko) 2003-02-14
BR0112038A (pt) 2003-04-01
EP1307200A2 (fr) 2003-05-07
NO20026195L (no) 2003-02-27
US20020068744A1 (en) 2002-06-06
HUP0300798A3 (en) 2006-02-28
BG107277A (bg) 2004-01-30
HUP0300798A2 (hu) 2003-07-28
AU2001273062B2 (en) 2005-11-24
WO2002002563A2 (fr) 2002-01-10
GEP20053688B (en) 2005-12-12
MXPA02011913A (es) 2003-04-22
AR034553A1 (es) 2004-03-03
CZ20024150A3 (cs) 2003-09-17
US7329663B2 (en) 2008-02-12
NZ523807A (en) 2004-09-24
WO2002002563A3 (fr) 2003-01-03
AU7306201A (en) 2002-01-14

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