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NO20026195D0 - Substituerte-triazolopyrimidiner som anticancer midler - Google Patents

Substituerte-triazolopyrimidiner som anticancer midler

Info

Publication number
NO20026195D0
NO20026195D0 NO20026195A NO20026195A NO20026195D0 NO 20026195 D0 NO20026195 D0 NO 20026195D0 NO 20026195 A NO20026195 A NO 20026195A NO 20026195 A NO20026195 A NO 20026195A NO 20026195 D0 NO20026195 D0 NO 20026195D0
Authority
NO
Norway
Prior art keywords
triazolopyrimidines
substituted
anticancer agents
anticancer
agents
Prior art date
Application number
NO20026195A
Other languages
English (en)
Other versions
NO20026195L (no
Inventor
Mark R Schmitt
Donald R Kirsch
Jane E Harris
Carl F Beyer
Klaus-Juergen Pees
Paul Carter
Waldemar Pfrengle
Guido Albert
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of NO20026195D0 publication Critical patent/NO20026195D0/no
Publication of NO20026195L publication Critical patent/NO20026195L/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
NO20026195A 2000-06-30 2002-12-23 Substituerte triazolpyrimidiner som anticancermidler NO20026195L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US21558500P 2000-06-30 2000-06-30
PCT/US2001/020672 WO2002002563A2 (en) 2000-06-30 2001-06-28 Substituted-triazolopyrimidines as anticancer agents

Publications (2)

Publication Number Publication Date
NO20026195D0 true NO20026195D0 (no) 2002-12-23
NO20026195L NO20026195L (no) 2003-02-27

Family

ID=22803554

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20026195A NO20026195L (no) 2000-06-30 2002-12-23 Substituerte triazolpyrimidiner som anticancermidler

Country Status (24)

Country Link
US (1) US7329663B2 (no)
EP (1) EP1307200A2 (no)
JP (1) JP2004502691A (no)
KR (1) KR20030013475A (no)
CN (1) CN1592624A (no)
AR (1) AR034553A1 (no)
AU (2) AU7306201A (no)
BG (1) BG107277A (no)
BR (1) BR0112038A (no)
CA (1) CA2413802A1 (no)
CZ (1) CZ20024150A3 (no)
EA (1) EA006483B1 (no)
GE (1) GEP20053688B (no)
HK (1) HK1052646A1 (no)
HU (1) HUP0300798A3 (no)
IL (1) IL152869A0 (no)
IN (1) IN2003KO00001A (no)
MX (1) MXPA02011913A (no)
NO (1) NO20026195L (no)
NZ (1) NZ523807A (no)
PL (1) PL360027A1 (no)
SK (1) SK18412002A3 (no)
WO (1) WO2002002563A2 (no)
ZA (1) ZA200300793B (no)

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DE10121162A1 (de) * 2001-04-30 2002-10-31 Bayer Ag Triazolopyrimidine
DE10124208A1 (de) † 2001-05-18 2002-11-21 Bayer Ag Verwendung von Triazolopyrimidin-Derivaten als Mikrobizide
IL159606A0 (en) * 2001-07-18 2004-06-01 Basf Ag Substituted 6-(2-tolyl)-triazolopyrimidines as fungicides
WO2003080615A1 (de) * 2002-03-21 2003-10-02 Basf Aktiengesellschaft Fungizide triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
WO2004011467A1 (ja) * 2002-07-29 2004-02-05 Hokko Chemical Industry Co., Ltd. トリアゾロピリミジン誘導体および農園芸用殺菌剤
UA80304C2 (en) * 2002-11-07 2007-09-10 Basf Ag Substituted 6-(2-halogenphenyl)triazolopyrimidines
MXPA05009338A (es) * 2003-03-31 2005-11-04 Basf Ag 7-alquenilamino-triazolopirimidinas, procedimientos para su obtencion y el uso de las mismas para controlar hongos nocivos, asi como productos que los contienen.
DE10325133A1 (de) * 2003-06-04 2004-12-23 Bayer Cropscience Ag Triazolopyrimidine
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DE10328171A1 (de) * 2003-06-24 2005-01-13 Bayer Cropscience Ag Triazolopyrimidine
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DE602004014525D1 (de) 2003-09-24 2008-07-31 Wyeth Corp 6-aryl-7-halo-imidazoä1,2-aüpyrimidine als mittel gegen krebs
AU2004276240A1 (en) 2003-09-24 2005-04-07 Wyeth Holdings Corporation 6-[(substituted)phenyl]triazolopyrimidines as anticancer agents
EP1674454A4 (en) * 2003-10-17 2006-12-27 Nippon Kayaku Kk SUBSTITUTED 2-AMINO-1,2,4-TRIAZOLO 1,5-A-PYRIMIDINE DERIVATIVE AND THE USE THEREOF
JP4606015B2 (ja) * 2003-11-25 2011-01-05 日本化薬株式会社 ［１，２，４］トリアゾロ［１，５−ａ］ピリミジン誘導体の新規医薬用途
MY179926A (en) 2003-12-08 2020-11-19 Wyeth Corp Process for the preparation of tubulin inhibitors
EP1697373A1 (de) * 2003-12-17 2006-09-06 Basf Aktiengesellschaft 6-(2,4,6-trihalogenphenyl)-triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bek mpfung von schadpil zen sowie sie enthaltende mittel
CN1894254A (zh) * 2003-12-17 2007-01-10 巴斯福股份公司 用于防治病原性真菌的6－(2,3,6－三氟苯基)三唑并嘧啶
US20070208038A1 (en) * 2004-03-30 2007-09-06 Basf Aktiengesellschaft 6-(2-Fluorophenyl)-Triazolopyrimidines, Method for Producing Them, Their use for Controlling Parasitic Fungi and Agents Containing the Same
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WO2007099092A1 (de) * 2006-02-28 2007-09-07 Basf Se Substituierte 6-phenyl-7-amino-[1,2,4]-triazolo[1,5-a]pyrimidine und deren verwendung zur bekämpfung von schadpilzen
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CN103360398B (zh) * 2013-07-22 2015-03-25 山东大学 一种三唑并嘧啶类hiv-1逆转录酶抑制剂及其制备方法与应用
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KR101995533B1 (ko) * 2017-03-21 2019-07-02 한국화학연구원 [1,2,4]트리아졸로[4,3-a]퀴노잘린 아미노 페닐 유도체 또는 이의 약학적으로 허용가능한 염, 이의 제조방법 및 이를 유효성분으로 포함하는 BET 단백질 관련 질환의 예방 또는 치료용 약학적 조성물
WO2020159942A1 (en) * 2019-01-29 2020-08-06 Tosk, Inc. Pyrazolopyrimidine modulators of ras gtpase
AU2021255495A1 (en) * 2020-04-14 2022-12-15 The Regents Of The University Of California Substituted {1,2,4,} triazolo{1,5-a} pyrimidine compounds and use in stabilizing microtubules
MX2022013619A (es) 2020-05-01 2022-11-16 Gilead Sciences Inc Compuestos de 2,4-dioxopirimidina que inhiben cd73.
US20230279006A1 (en) * 2020-07-08 2023-09-07 Klotho Therapeutics, Inc. Novel compounds and methods for increasing klotho gene expression
US12180220B2 (en) 2020-10-14 2024-12-31 Tosk, Inc. Heteroaryl modulators of RAS GTPase
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CN118475581A (zh) * 2022-01-25 2024-08-09 瑞石生物医药有限公司 一种ccr4小分子拮抗剂及其用途

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Also Published As

Publication number Publication date
NO20026195L (no) 2003-02-27
CA2413802A1 (en) 2002-01-10
CN1592624A (zh) 2005-03-09
EA200300091A1 (ru) 2003-08-28
PL360027A1 (en) 2004-09-06
HUP0300798A3 (en) 2006-02-28
HK1052646A1 (zh) 2003-09-26
GEP20053688B (en) 2005-12-12
CZ20024150A3 (cs) 2003-09-17
SK18412002A3 (sk) 2003-06-03
HUP0300798A2 (hu) 2003-07-28
KR20030013475A (ko) 2003-02-14
US20020068744A1 (en) 2002-06-06
NZ523807A (en) 2004-09-24
US7329663B2 (en) 2008-02-12
JP2004502691A (ja) 2004-01-29
ZA200300793B (en) 2004-07-20
AR034553A1 (es) 2004-03-03
BG107277A (bg) 2004-01-30
EP1307200A2 (en) 2003-05-07
WO2002002563A3 (en) 2003-01-03
AU2001273062B2 (en) 2005-11-24
EA006483B1 (ru) 2005-12-29
IL152869A0 (en) 2003-06-24
MXPA02011913A (es) 2003-04-22
BR0112038A (pt) 2003-04-01
IN2003KO00001A (no) 2005-12-02
WO2002002563A2 (en) 2002-01-10
AU7306201A (en) 2002-01-14

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