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HUE049997T2 - Eljárás a diozmin elõállítására - Google Patents

Eljárás a diozmin elõállítására

Info

Publication number
HUE049997T2
HUE049997T2 HUE16702557A HUE16702557A HUE049997T2 HU E049997 T2 HUE049997 T2 HU E049997T2 HU E16702557 A HUE16702557 A HU E16702557A HU E16702557 A HUE16702557 A HU E16702557A HU E049997 T2 HUE049997 T2 HU E049997T2
Authority
HU
Hungary
Prior art keywords
diiodine
production
Prior art date
Application number
HUE16702557A
Other languages
English (en)
Inventor
Cremades Francisco Javier Lopez
Original Assignee
Healthtech Bio Actives S L U
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Healthtech Bio Actives S L U filed Critical Healthtech Bio Actives S L U
Publication of HUE049997T2 publication Critical patent/HUE049997T2/hu

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/06Benzopyran radicals
    • C07H17/065Benzo[b]pyrans
    • C07H17/07Benzo[b]pyran-4-ones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/14Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00Processes for the preparation of sugar derivatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Cardiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Saccharide Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
HUE16702557A 2015-02-03 2016-02-02 Eljárás a diozmin elõállítására HUE049997T2 (hu)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP15153537.4A EP3053930A1 (en) 2015-02-03 2015-02-03 Process for the preparation of diosmin

Publications (1)

Publication Number Publication Date
HUE049997T2 true HUE049997T2 (hu) 2020-11-30

Family

ID=52477555

Family Applications (1)

Application Number Title Priority Date Filing Date
HUE16702557A HUE049997T2 (hu) 2015-02-03 2016-02-02 Eljárás a diozmin elõállítására

Country Status (24)

Country Link
US (2) US10287310B2 (hu)
EP (2) EP3053930A1 (hu)
KR (2) KR102216702B1 (hu)
CN (1) CN107108675B (hu)
AR (1) AR103583A1 (hu)
BR (1) BR112017016430B1 (hu)
CA (1) CA2974860A1 (hu)
EA (1) EA032402B1 (hu)
ES (1) ES2803213T3 (hu)
HR (1) HRP20201102T1 (hu)
HU (1) HUE049997T2 (hu)
LT (1) LT3253772T (hu)
MA (1) MA40703B1 (hu)
MX (1) MX372637B (hu)
MY (1) MY183290A (hu)
PH (1) PH12017501244B1 (hu)
PL (1) PL3253772T3 (hu)
PT (1) PT3253772T (hu)
RS (1) RS60494B1 (hu)
SI (1) SI3253772T1 (hu)
TW (1) TWI715551B (hu)
UA (1) UA123046C2 (hu)
UY (1) UY36549A (hu)
WO (1) WO2016124585A1 (hu)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN106967138A (zh) * 2017-04-19 2017-07-21 成都百特万合医药科技有限公司 基于二甲亚砜体系的地奥司明生产方法
AR122887A1 (es) * 2020-07-09 2022-10-12 Servier Lab Procedimiento de preparación de la diosmina
AR126366A1 (es) 2021-07-06 2023-10-11 Servier Lab Procedimiento para la preparación de diosmina y de fracción flavonoica

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH602778A5 (hu) 1975-05-16 1978-07-31 Hommel Ag
ES440427A1 (es) 1975-08-25 1977-03-01 Espanola Prod Quimicos Un procedimiento de obtencion de flavonas.
DE2740950A1 (de) 1977-09-10 1979-03-22 Merck Patent Gmbh Verfahren zur herstellung von flavonen
IT1150612B (it) 1982-03-04 1986-12-17 Prophin Lab Spa Procedimento per la preparazione del 1',5,7-tridrossi-4'-metossiflavone-7-rutinoside (diosmina)
DE3514123C2 (de) 1985-04-19 1994-12-08 Kabelmetal Ag Verfahren zur Herstellung von Durchlaufkokillen für Stranggießmaschinen
IT1191620B (it) 1985-05-30 1988-03-23 Edmond Pharma Srl Procedimento per la preparazione della diosmina
GB9717629D0 (en) * 1997-08-21 1997-10-22 Johnson Matthey Plc Removal of residual organic solvents
FR2782518A1 (fr) 1998-08-19 2000-02-25 Innokem Sarl Procede de fabrication industrielle de diosmine a partir de l'hesperidine par reaction avec de l'iode et de la pyridine
CN102653549A (zh) * 2011-12-28 2012-09-05 长沙富能生物技术有限公司 一种符合ep7版质量标准的地奥司明原料药合成方法

Also Published As

Publication number Publication date
PH12017501244A1 (en) 2017-10-30
PH12017501244B1 (en) 2017-10-30
UA123046C2 (uk) 2021-02-10
EP3053930A1 (en) 2016-08-10
ES2803213T3 (es) 2021-01-25
KR102216702B1 (ko) 2021-02-18
EP3253772B8 (en) 2020-07-15
EA032402B1 (ru) 2019-05-31
MX2017010026A (es) 2017-12-18
EA201791280A1 (ru) 2017-11-30
CN107108675A (zh) 2017-08-29
WO2016124585A1 (en) 2016-08-11
BR112017016430B1 (pt) 2022-11-29
PL3253772T3 (pl) 2020-12-28
TW201629078A (zh) 2016-08-16
SI3253772T1 (sl) 2020-09-30
CA2974860A1 (en) 2016-08-11
US10711025B2 (en) 2020-07-14
KR20170108005A (ko) 2017-09-26
EP3253772B1 (en) 2020-04-22
TWI715551B (zh) 2021-01-11
CN107108675B (zh) 2020-10-27
MX372637B (es) 2020-06-12
KR20200131334A (ko) 2020-11-23
KR102309525B1 (ko) 2021-10-07
EP3253772A1 (en) 2017-12-13
AR103583A1 (es) 2017-05-17
BR112017016430A2 (pt) 2018-04-10
RS60494B1 (sr) 2020-08-31
US20180016292A1 (en) 2018-01-18
US20190225639A1 (en) 2019-07-25
HRP20201102T1 (hr) 2020-11-13
UY36549A (es) 2016-08-31
PT3253772T (pt) 2020-07-01
MA40703B1 (fr) 2019-07-31
US10287310B2 (en) 2019-05-14
MA40703A1 (fr) 2017-12-29
LT3253772T (lt) 2020-09-25
MY183290A (en) 2021-02-18

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