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GT200800199A - Compuestos nuevos - Google Patents

Compuestos nuevos

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Publication number
GT200800199A
GT200800199A GT200800199A GT200800199A GT200800199A GT 200800199 A GT200800199 A GT 200800199A GT 200800199 A GT200800199 A GT 200800199A GT 200800199 A GT200800199 A GT 200800199A GT 200800199 A GT200800199 A GT 200800199A
Authority
GT
Guatemala
Prior art keywords
new compounds
compounds
dgat1
humans
animals
Prior art date
Application number
GT200800199A
Other languages
English (en)
Inventor
Michael H Serrano-Wu
Kwak Young-Shin
Liu Wenming
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38564569&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=GT200800199(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of GT200800199A publication Critical patent/GT200800199A/es

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/421—1,3-Oxazoles, e.g. pemoline, trimethadione
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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Abstract

LA PRESENTE INVENCIÓN PROPORCIONA COMPUESTOS ORGÁNICOS DE LA SIGUIENTE ESTRUCTURA: A-L1-B-C-D-L2-E, DONDE A, L1, L2, B, C, D Y E SE ENCUENTRAN EXPLICADOS EN LA MEMORIA DESCRIPTIVA. ESTOS COMPUESTOS SON ÚTILES PARA TRATAR O PREVENIR CONDICIONES O TRASTORNOS ASOCIADOS CON LA ACTIVIDAD DE LA DGAT1 EN LOS ANIMALES, EN PARTICULAR EN LOS HUMANOS. T2008
GT200800199A 2006-03-31 2008-09-29 Compuestos nuevos GT200800199A (es)

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