GT199900019A - Formulas farmaceuticamente estables de solucion de oxaliplatino. - Google Patents
Formulas farmaceuticamente estables de solucion de oxaliplatino.Info
- Publication number
- GT199900019A GT199900019A GT199900019A GT199900019A GT199900019A GT 199900019 A GT199900019 A GT 199900019A GT 199900019 A GT199900019 A GT 199900019A GT 199900019 A GT199900019 A GT 199900019A GT 199900019 A GT199900019 A GT 199900019A
- Authority
- GT
- Guatemala
- Prior art keywords
- oxaliplatino
- solution
- pharmaceutically stable
- formulas
- stable formulas
- Prior art date
Links
- 206010028980 Neoplasm Diseases 0.000 abstract 2
- 201000011510 cancer Diseases 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/12—Carboxylic acids; Salts or anhydrides thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/28—Compounds containing heavy metals
- A61K31/282—Platinum compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/555—Heterocyclic compounds containing heavy metals, e.g. hemin, hematin, melarsoprol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Engineering & Computer Science (AREA)
- Dermatology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Abstract
LA INVENCIÒN SE RELACIONA CON FÒRMULAS FARMACEÙTICAMENTE ESTABLES DE SOLUCIÒN DE OXALIPLATINO, AL MÈTODO PARA USARLAS EN EL TRATAMIENTO DE TUMORES DE CÀNCER, A PROCESOS PARA LA PREPARACIÒN DE TALES FÒRMULAS Y A UN MÈTODO PARA ESTABILIZAR LAS SOLUCIONES DE OXALIPLATINO.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9804013.2A GB9804013D0 (en) | 1998-02-25 | 1998-02-25 | Formulations |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GT199900019A true GT199900019A (es) | 2000-08-04 |
Family
ID=10827600
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GT199900019A GT199900019A (es) | 1998-02-25 | 1999-02-11 | Formulas farmaceuticamente estables de solucion de oxaliplatino. |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US6306902B1 (es) |
| EP (1) | EP0943331B1 (es) |
| JP (1) | JP4430229B2 (es) |
| KR (1) | KR20010041182A (es) |
| CN (1) | CN1152718C (es) |
| AR (1) | AR015524A1 (es) |
| AT (1) | ATE202472T1 (es) |
| AU (1) | AU757101B2 (es) |
| BR (1) | BR9908273A (es) |
| CA (1) | CA2261500C (es) |
| CZ (1) | CZ302196B6 (es) |
| DE (1) | DE69900162T2 (es) |
| DK (1) | DK0943331T3 (es) |
| ES (1) | ES2161085T3 (es) |
| GB (1) | GB9804013D0 (es) |
| GR (1) | GR3036646T3 (es) |
| GT (1) | GT199900019A (es) |
| HU (1) | HU224611B1 (es) |
| IL (1) | IL137772A (es) |
| MX (1) | MXPA00008195A (es) |
| NO (1) | NO329900B1 (es) |
| PL (1) | PL197948B1 (es) |
| PT (1) | PT943331E (es) |
| RU (1) | RU2207857C2 (es) |
| UA (1) | UA70316C2 (es) |
| WO (1) | WO1999043355A2 (es) |
| ZA (1) | ZA991489B (es) |
Families Citing this family (44)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9804013D0 (en) | 1998-02-25 | 1998-04-22 | Sanofi Sa | Formulations |
| WO2000021527A2 (fr) * | 1998-10-14 | 2000-04-20 | Debiopharm S.A. | Conditionnement d'une preparation d'oxaliplatine |
| US7070796B1 (en) | 1999-08-30 | 2006-07-04 | Debiopharm S.A. | Pharmaceutically stable oxaliplatinum preparation for parenteral administration |
| BRPI0013613B8 (pt) * | 1999-08-30 | 2021-05-25 | Debiopharm Sa | composição farmacêuticamente estável de oxaliplatina para administração parenteral. |
| EP1341555A2 (fr) * | 2000-12-12 | 2003-09-10 | Debiopharm S.A. | Preparation pharmaceutique d'oxaliplatine pour administration par voie parenterale et procede d'obtention de ladite preparation |
| DE60220766T2 (de) | 2001-03-02 | 2008-03-06 | Debiopharm S.A. | Verwendung eines eine oxaliplatinlösung beinhaltenden fläschchens |
| US20040186172A1 (en) | 2001-07-02 | 2004-09-23 | Houssam Ibrahim | Oxaliplatin active substance with a very low content of oxalic acid |
| US6476068B1 (en) * | 2001-12-06 | 2002-11-05 | Pharmacia Italia, S.P.A. | Platinum derivative pharmaceutical formulations |
| CA2388352A1 (en) * | 2002-05-31 | 2003-11-30 | Voiceage Corporation | A method and device for frequency-selective pitch enhancement of synthesized speed |
| DE10314377A1 (de) * | 2003-03-28 | 2004-10-07 | Stada Arzneimittel Ag | Gebrauchsfertige Oxaliplatin-Lösungen |
| US20050020556A1 (en) * | 2003-05-30 | 2005-01-27 | Kosan Biosciences, Inc. | Method for treating diseases using HSP90-inhibiting agents in combination with platinum coordination complexes |
| GB2441445B (en) * | 2003-08-28 | 2008-04-23 | Mayne Pharma Ltd | Acid containing oxaliplatin formulation |
| JP2007504098A (ja) | 2003-08-28 | 2007-03-01 | メイン・ファーマ・リミテッド | 酸を含むオキサリプラチン製剤 |
| CZ300795B6 (cs) * | 2003-09-02 | 2009-08-12 | Pliva-Lachema A. S. | Farmaceutická kompozice a zpusob její výroby |
| JP2007504177A (ja) * | 2003-09-02 | 2007-03-01 | プリヴァ−ラケマ,エー.エス. | 医薬組成物、その製造方法及び治療上の使用 |
| EP2330110A1 (en) | 2003-11-25 | 2011-06-08 | Platco Technologies (Proprietary) Limited | Platinum(II) complexes, preparation and use |
| WO2005056641A1 (ja) * | 2003-12-10 | 2005-06-23 | Toudai Tlo, Ltd. | ジアミノシクロヘキサン白金(ii)とポリ(カルボン酸)セグメント含有ブロック共重合体との配位錯体、その抗腫瘍剤 |
| CN100471493C (zh) * | 2003-12-17 | 2009-03-25 | 梅比欧法姆股份有限公司 | 含有奥沙利铂的脂质体制剂 |
| WO2005102312A1 (en) * | 2004-04-27 | 2005-11-03 | Mayne Pharma Limited | Concentrated oxaliplatin solutions |
| PL1789427T3 (pl) | 2004-09-01 | 2009-10-30 | Platco Tech Proprietary Limited | Otrzymywanie kompleksów platyny (II) |
| US20060063720A1 (en) * | 2004-09-22 | 2006-03-23 | Edgar Schridde | Oxaliplatin solution concentrate |
| US20060063833A1 (en) * | 2004-09-22 | 2006-03-23 | Edgar Schridde | Ready-to-use oxaliplatin solutions |
| DE102004052877B4 (de) * | 2004-11-02 | 2008-06-19 | Ebewe Pharma Ges.M.B.H. Nfg.Kg | Stabile wässrige Formulierungen eines Platin-Derivats |
| DE102004063764A1 (de) * | 2004-12-29 | 2006-07-13 | Hexal Ag | Kunststoff-Flasche für Oxaliplatin |
| JP2006248978A (ja) | 2005-03-10 | 2006-09-21 | Mebiopharm Co Ltd | 新規なリポソーム製剤 |
| AU2005329764B2 (en) * | 2005-03-28 | 2010-08-12 | Dabur Pharma Ltd. | Stable pharmaceutical compositions of platinum (II) antitumour agents |
| EP1874290A1 (en) * | 2005-04-09 | 2008-01-09 | Vuab Pharma A. S. | A process for the preparation of an oxaliplatin preparation |
| RU2292210C1 (ru) * | 2005-05-03 | 2007-01-27 | Институт химии и химической технологии СО РАН (ИХХТ СО РАН) | Способ получения стерилизованной микрокристаллической цис-дихлородиамминплатины (ii) |
| DE102005038347A1 (de) * | 2005-08-11 | 2007-02-15 | Hexal Ag | Herstellung einer Oxaliplatin-Lösung und Behälter sowie Behälter-Set mit der Lösung |
| WO2007029268A2 (en) * | 2005-09-05 | 2007-03-15 | Dabur Pharma Limited | Stable oxaliplatin formulation |
| JP2009525273A (ja) | 2006-01-30 | 2009-07-09 | プラットコー テクノロジーズ (プロプライエタリー) リミテッド | 白金(ii)錯体の調製 |
| KR100913063B1 (ko) | 2006-09-13 | 2009-08-21 | 주식회사유한양행 | 옥살리플라틴-함유 주사용 용액 |
| MX2009007801A (es) * | 2007-01-22 | 2009-10-08 | Pliva Lachema As | Composicion farmaceutica de oxaliplatino con regulador basado en azucar alcoholico. |
| RU2340347C2 (ru) * | 2007-01-24 | 2008-12-10 | Институт химии и химической технологии СО РАН (ИХХТ СО РАН) | Способ получения стерилизованной микрокристаллической соли цис-дихлороамминизопропиламинплатины (ii) |
| US20100267824A1 (en) * | 2007-11-12 | 2010-10-21 | Intas Pharmaceuticals Limited | Stable oxaliplatin composition for parenteral administration |
| US20090130017A1 (en) * | 2007-11-19 | 2009-05-21 | Searete Llc | Targeted short-lived drug delivery |
| TW201021855A (en) * | 2008-11-13 | 2010-06-16 | Taigen Biotechnology Co Ltd | Lyophilization formulation |
| CN101461801B (zh) * | 2008-12-26 | 2013-05-15 | 辰欣药业股份有限公司 | 一种奥沙利铂药物组合物及其制备方法 |
| AU2010296180B2 (en) | 2009-09-21 | 2016-05-05 | Bio-Synectics, Inc | Oxaliplatin nanoparticles and method for preparing same |
| CN102274171A (zh) * | 2011-08-04 | 2011-12-14 | 上海希迪制药有限公司 | 一种奥沙利铂注射剂 |
| CN104523674B (zh) * | 2014-12-11 | 2017-10-24 | 广州市上为医药科技有限公司 | 一种以奥沙利铂为主药成分的注射用组合物 |
| KR101683635B1 (ko) * | 2014-12-29 | 2016-12-09 | 가천대학교 산학협력단 | 락테이트 금속염을 포함하는 암 치료용 약학 조성물 |
| CN104829653B (zh) * | 2015-05-06 | 2016-03-23 | 山东罗欣药业集团股份有限公司 | 一种奥沙利铂水合物晶体及其冻干粉针剂 |
| KR102868782B1 (ko) | 2018-01-12 | 2025-10-13 | (주)메티메디제약 | 만성 염증성 질환의 치료 방법 |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS6041077B2 (ja) * | 1976-09-06 | 1985-09-13 | 喜徳 喜谷 | 1,2‐ジアミノシクロヘキサン異性体のシス白金(2)錯体 |
| PT93772A (pt) | 1989-04-17 | 1991-01-08 | Searle & Co | Processo para a preparacao de composicoes para o tratamento de neoplasias, contendo um agente anti-neoplastico, por exemplo doxorubicina e um agente protector para reduzir os efeitos secundarios, por exemplo carbetimer |
| EP0464210A4 (en) | 1989-12-15 | 1992-11-25 | Tsumura & Co. | Novel platinum complex and antitumor drug containing the same as active ingredient |
| JPH04185601A (ja) | 1990-11-20 | 1992-07-02 | Unitika Ltd | 白金抗癌剤徐放性製剤 |
| MX9206577A (es) | 1991-11-15 | 1993-05-01 | Smithkline Beecham Corp | COMPOSICIóN FARMACEUTICA PARA INHIBIR EL CRECIMIENTO DE CELULAS TUMORALES |
| JPH0776230B2 (ja) * | 1992-01-13 | 1995-08-16 | 田中貴金属工業株式会社 | 白金化合物の製造方法 |
| JPH05238936A (ja) | 1992-02-27 | 1993-09-17 | Dainippon Pharmaceut Co Ltd | カルシトリオールの水性液剤 |
| JPH06287021A (ja) * | 1992-04-22 | 1994-10-11 | Tanaka Kikinzoku Kogyo Kk | 光学活性な白金錯化合物の光学的分割方法 |
| JP2673331B2 (ja) * | 1993-01-12 | 1997-11-05 | 田中貴金属工業 株式会社 | 光学的に高純度なシス―オキザラート(トランス―1―1,2―シクロヘキサンジアミン)白金(▲ii▼) |
| AU5416394A (en) * | 1992-11-24 | 1994-06-22 | Debiopharm S.A. | Cisplatinum/oxaliplatinum combination |
| JP3025602B2 (ja) * | 1993-05-21 | 2000-03-27 | デビオファーム エス.アー. | 光学的に高純度なシス−オキザラート(トランス−l−1,2−シクロヘキサンジアミン)白金(II)錯体の製造方法 |
| US5455270A (en) * | 1993-08-11 | 1995-10-03 | Bristol-Myers Squibb Co. | Stabilized solutions of platinum(II) antitumor agents |
| KR100365171B1 (ko) | 1994-08-08 | 2003-02-19 | 드바이오팜 에스.아. | 약학적으로안정한옥살리플라티늄제제 |
| DE69531722T2 (de) * | 1994-11-11 | 2004-07-01 | Debiopharm S.A. | Karzinostatische Zusammensetzungen, welche Cis-Oxaliplatin und eine oder mehrere andere verträgliche Karzinostatika enthalten |
| FR2740686B1 (fr) * | 1995-11-03 | 1998-01-16 | Sanofi Sa | Formulation pharmaceutique lyophilisee stable |
| EP0801070B1 (en) | 1996-04-10 | 2003-04-16 | Debiopharm S.A. | Process of preparing platinum compound |
| JPH09294809A (ja) | 1996-05-07 | 1997-11-18 | Terumo Corp | 薬液注入器具 |
| GB9804013D0 (en) | 1998-02-25 | 1998-04-22 | Sanofi Sa | Formulations |
-
1998
- 1998-02-25 GB GBGB9804013.2A patent/GB9804013D0/en not_active Ceased
-
1999
- 1999-02-11 CA CA002261500A patent/CA2261500C/en not_active Expired - Lifetime
- 1999-02-11 GT GT199900019A patent/GT199900019A/es unknown
- 1999-02-22 US US09/255,087 patent/US6306902B1/en not_active Expired - Lifetime
- 1999-02-24 AR ARP990100774A patent/AR015524A1/es active IP Right Grant
- 1999-02-24 ZA ZA9901489A patent/ZA991489B/xx unknown
- 1999-02-25 PT PT99301412T patent/PT943331E/pt unknown
- 1999-02-25 ES ES99301412T patent/ES2161085T3/es not_active Expired - Lifetime
- 1999-02-25 EP EP99301412A patent/EP0943331B1/en not_active Expired - Lifetime
- 1999-02-25 DE DE69900162T patent/DE69900162T2/de not_active Ceased
- 1999-02-25 PL PL343021A patent/PL197948B1/pl unknown
- 1999-02-25 AT AT99301412T patent/ATE202472T1/de active
- 1999-02-25 DK DK99301412T patent/DK0943331T3/da active
- 1999-02-25 HU HU0103707A patent/HU224611B1/hu active IP Right Grant
- 1999-02-25 MX MXPA00008195A patent/MXPA00008195A/es active IP Right Grant
- 1999-02-25 CN CNB99803276XA patent/CN1152718C/zh not_active Expired - Lifetime
- 1999-02-25 CZ CZ20003089A patent/CZ302196B6/cs not_active IP Right Cessation
- 1999-02-25 RU RU2000121254/14A patent/RU2207857C2/ru active
- 1999-02-25 JP JP2000533150A patent/JP4430229B2/ja not_active Expired - Lifetime
- 1999-02-25 UA UA2000095450A patent/UA70316C2/uk unknown
- 1999-02-25 WO PCT/GB1999/000572 patent/WO1999043355A2/en not_active Ceased
- 1999-02-25 AU AU26324/99A patent/AU757101B2/en not_active Expired
- 1999-02-25 KR KR1020007009239A patent/KR20010041182A/ko not_active Ceased
- 1999-02-25 BR BR9908273-0A patent/BR9908273A/pt not_active Application Discontinuation
-
2000
- 2000-08-09 IL IL137772A patent/IL137772A/en not_active IP Right Cessation
- 2000-08-24 NO NO20004240A patent/NO329900B1/no not_active IP Right Cessation
-
2001
- 2001-09-18 GR GR20010401504T patent/GR3036646T3/el unknown
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