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FR13C0037I2 - Solvat acetonique du dimethoxy docetaxel et son procede de preparation - Google Patents

Solvat acetonique du dimethoxy docetaxel et son procede de preparation

Info

Publication number
FR13C0037I2
FR13C0037I2 FR13C0037C FR13C0037C FR13C0037I2 FR 13C0037 I2 FR13C0037 I2 FR 13C0037I2 FR 13C0037 C FR13C0037 C FR 13C0037C FR 13C0037 C FR13C0037 C FR 13C0037C FR 13C0037 I2 FR13C0037 I2 FR 13C0037I2
Authority
FR
France
Prior art keywords
preparation process
dimethoxy docetaxel
acetonic
solvate
acetonic solvate
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
FR13C0037C
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharma SA
Original Assignee
Aventis Pharma SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34224354&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FR13C0037(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Aventis Pharma SA filed Critical Aventis Pharma SA
Publication of FR13C0037I1 publication Critical patent/FR13C0037I1/fr
Application granted granted Critical
Publication of FR13C0037I2 publication Critical patent/FR13C0037I2/fr
Active legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D305/00Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Epoxy Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Cephalosporin Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
FR13C0037C 2003-09-19 2013-07-04 Solvat acetonique du dimethoxy docetaxel et son procede de preparation Active FR13C0037I2 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0311016A FR2859996B1 (fr) 2003-09-19 2003-09-19 Solvat acetonique du dimethoxy docetaxel et son procede de preparation
PCT/FR2004/002344 WO2005028462A1 (fr) 2003-09-19 2004-09-16 Solvat acetonique du dimethoxy docetaxel et son procede de preparation

Publications (2)

Publication Number Publication Date
FR13C0037I1 FR13C0037I1 (fr) 2013-09-08
FR13C0037I2 true FR13C0037I2 (fr) 2015-11-20

Family

ID=34224354

Family Applications (2)

Application Number Title Priority Date Filing Date
FR0311016A Expired - Lifetime FR2859996B1 (fr) 2003-09-19 2003-09-19 Solvat acetonique du dimethoxy docetaxel et son procede de preparation
FR13C0037C Active FR13C0037I2 (fr) 2003-09-19 2013-07-04 Solvat acetonique du dimethoxy docetaxel et son procede de preparation

Family Applications Before (1)

Application Number Title Priority Date Filing Date
FR0311016A Expired - Lifetime FR2859996B1 (fr) 2003-09-19 2003-09-19 Solvat acetonique du dimethoxy docetaxel et son procede de preparation

Country Status (37)

Country Link
US (1) US7241907B2 (fr)
EP (1) EP1667986B1 (fr)
JP (1) JP5010279B2 (fr)
KR (1) KR101123588B1 (fr)
CN (1) CN100429207C (fr)
AR (1) AR045667A1 (fr)
AU (1) AU2004274212B2 (fr)
BE (1) BE2013C036I2 (fr)
BR (1) BRPI0414492A8 (fr)
CA (1) CA2539309A1 (fr)
CR (1) CR8292A (fr)
CY (2) CY1114575T1 (fr)
DK (1) DK1667986T3 (fr)
ES (1) ES2403149T4 (fr)
FR (2) FR2859996B1 (fr)
HR (1) HRP20130322T1 (fr)
HU (1) HUS1300025I1 (fr)
IL (1) IL174240A (fr)
LU (1) LU92172I2 (fr)
MA (1) MA28045A1 (fr)
ME (2) ME00054B (fr)
MX (1) MXPA06002639A (fr)
MY (1) MY136668A (fr)
NO (2) NO335997B1 (fr)
NZ (1) NZ545835A (fr)
PA (1) PA8612401A1 (fr)
PE (1) PE20050870A1 (fr)
PL (1) PL1667986T3 (fr)
PT (1) PT1667986E (fr)
RS (2) RS20060189A (fr)
RU (1) RU2342373C2 (fr)
SI (1) SI1667986T1 (fr)
TN (1) TNSN06086A1 (fr)
TW (1) TWI382022B (fr)
UA (1) UA87115C2 (fr)
WO (1) WO2005028462A1 (fr)
ZA (1) ZA200602255B (fr)

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FR2945211A1 (fr) * 2009-05-06 2010-11-12 Sanofi Aventis Combinaison antitumorale comprenant la cabazitaxel et la capecitabine
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CN102675257B (zh) * 2012-05-10 2014-07-02 上海金和生物技术有限公司 一种卡巴他赛晶体及其制备方法
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EP2884963B1 (fr) 2012-08-15 2017-12-27 Yung Shin Pharm. Ind. Co. Ltd. Formulation pharmaceutique stable de cabazitaxel
CN103664836B (zh) * 2012-09-20 2016-04-20 齐鲁制药有限公司 7β,10β-二甲氧基多西紫杉醇氘代丙酮合物的晶型A及其制备方法
WO2014055493A1 (fr) 2012-10-02 2014-04-10 Cerulean Pharma Inc. Procédés et systèmes s'appliquant à la précipitation de polymères et à la génération de particules
CN103804323A (zh) * 2012-11-14 2014-05-21 上海希迈医药科技有限公司 一种卡巴他赛溶剂化物及其制备方法和应用
CN103058960B (zh) * 2012-12-12 2014-12-10 江苏奥赛康药业股份有限公司 卡巴他赛多晶型形式及其制备方法
EP2743264A1 (fr) 2012-12-13 2014-06-18 INDENA S.p.A. Nouvelle forme cristalline de cabazitaxel, procédé de préparation et ses compositions pharmaceutiques
CN103910696B (zh) * 2012-12-30 2016-01-20 上海医药工业研究院 卡巴他赛异丙醚合物及其结晶
CN103910698B (zh) * 2012-12-30 2016-01-20 上海医药工业研究院 卡巴他赛丙酮合物及其结晶
EP2777691A1 (fr) 2013-03-14 2014-09-17 Pharmachemie B.V. Taxoïde - purification des excipients liquides
EP2815749A1 (fr) 2013-06-20 2014-12-24 IP Gesellschaft für Management mbH Forme solide de 4-amino-2-(2,6-dioxopiperidine-3-yl)isoindoline-1,3-dione ayant un réseau de diffraction de rayons X spécifique
WO2015000165A1 (fr) * 2013-07-04 2015-01-08 北京新天宇科技开发有限公司 Produit de transformation stable du mono-acétonate de dimethoxy docetaxel et ses formes cristallines, et leurs procédés de préparation
CN104277014A (zh) * 2013-07-04 2015-01-14 北京新天宇科技开发有限公司 二甲氧基多西紫杉醇一丙酮化物的稳定转化物及其结晶形式、以及它们的制备方法
EP2865674A1 (fr) 2013-10-23 2015-04-29 INDENA S.p.A. Formes dissoutes cristallines de Cabazitaxel
EP2865675A1 (fr) * 2013-10-23 2015-04-29 INDENA S.p.A. Forme cristalline anhydre de Cabazitaxel, procédé de préparation et ses compositions pharmaceutiques
CN103601704B (zh) * 2013-11-22 2015-05-06 石家庄智恒医药科技有限公司 无定形卡巴他赛的制备
ES2904505T3 (es) 2015-01-12 2022-04-05 Emcure Pharmaceuticals Ltd Formulación líquida de cabazitaxel
EP3258931B1 (fr) * 2015-02-17 2020-08-12 Erasmus University Medical Center Rotterdam Utilisation de cabazitaxel pour le traitement du cancer de la prostate
EP3093014A1 (fr) 2015-05-13 2016-11-16 Aventis Pharma S.A. Cabazitaxel et son utilisation pour le traitement du cancer
US10188626B2 (en) 2015-11-03 2019-01-29 Cipla Limited Stabilized cabazitaxel formulations
CN110312721A (zh) 2016-11-29 2019-10-08 显莎制药公司 墨蝶呤的多晶型物
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Also Published As

Publication number Publication date
BRPI0414492A (pt) 2006-11-14
JP5010279B2 (ja) 2012-08-29
AU2004274212B2 (en) 2010-03-04
BRPI0414492A8 (pt) 2019-01-15
UA87115C2 (ru) 2009-06-25
US7241907B2 (en) 2007-07-10
CY2013016I2 (el) 2018-01-10
PA8612401A1 (es) 2005-08-04
ME00054B (me) 2011-02-10
NO20061714L (no) 2006-04-19
MEP11708A (en) 2010-06-10
EP1667986A1 (fr) 2006-06-14
NZ545835A (en) 2009-10-30
CN1849311A (zh) 2006-10-18
KR101123588B1 (ko) 2012-03-22
RS20060189A (sr) 2008-06-05
LU92172I9 (fr) 2019-01-03
MXPA06002639A (es) 2006-06-05
ES2403149T3 (es) 2013-05-14
FR2859996B1 (fr) 2006-02-03
KR20060072147A (ko) 2006-06-27
CN100429207C (zh) 2008-10-29
HUS1300025I1 (hu) 2016-08-29
PE20050870A1 (es) 2005-11-21
PL1667986T3 (pl) 2013-06-28
TWI382022B (zh) 2013-01-11
DK1667986T3 (da) 2013-05-06
HRP20130322T1 (en) 2013-07-31
TW200524891A (en) 2005-08-01
RU2342373C2 (ru) 2008-12-27
AR045667A1 (es) 2005-11-02
CA2539309A1 (fr) 2005-03-31
PT1667986E (pt) 2013-04-24
CR8292A (es) 2008-10-15
ZA200602255B (en) 2007-07-25
FR2859996A1 (fr) 2005-03-25
BE2013C036I2 (fr) 2023-12-14
HK1093340A1 (zh) 2007-03-02
FR13C0037I1 (fr) 2013-09-08
NO2015013I2 (no) 2015-04-22
MY136668A (en) 2008-11-28
AU2004274212A1 (en) 2005-03-31
IL174240A (en) 2010-12-30
TNSN06086A1 (en) 2007-10-03
ES2403149T4 (es) 2013-06-24
RS54614B1 (sr) 2016-08-31
US20050065138A1 (en) 2005-03-24
EP1667986B1 (fr) 2013-01-16
NO2015013I1 (no) 2015-05-04
LU92172I2 (fr) 2013-05-21
IL174240A0 (en) 2006-08-01
RU2006113122A (ru) 2006-08-27
MA28045A1 (fr) 2006-07-03
CY1114575T1 (el) 2016-10-05
CY2013016I1 (el) 2018-01-10
JP2007505866A (ja) 2007-03-15
NO335997B1 (no) 2015-04-20
SI1667986T1 (sl) 2013-05-31
WO2005028462A1 (fr) 2005-03-31

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