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FI943799L - Fenoksifenyylisyklopentenyylihydroksiureoita - Google Patents

Fenoksifenyylisyklopentenyylihydroksiureoita Download PDF

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Publication number
FI943799L
FI943799L FI943799A FI943799A FI943799L FI 943799 L FI943799 L FI 943799L FI 943799 A FI943799 A FI 943799A FI 943799 A FI943799 A FI 943799A FI 943799 L FI943799 L FI 943799L
Authority
FI
Finland
Prior art keywords
phenoxyphenylcyclopentenylhydroxyureas
Prior art date
Application number
FI943799A
Other languages
English (en)
Swedish (sv)
Other versions
FI943799A0 (fi
FI114466B (fi
Inventor
Akiyoshi Kawai
Rodney W Stevens
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI943799A0 publication Critical patent/FI943799A0/fi
Publication of FI943799L publication Critical patent/FI943799L/fi
Application granted granted Critical
Publication of FI114466B publication Critical patent/FI114466B/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C275/00Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C275/64Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups singly-bound to oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/17Amides, e.g. hydroxamic acids having the group >N—C(O)—N< or >N—C(S)—N<, e.g. urea, thiourea, carmustine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/06Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/10Systems containing only non-condensed rings with a five-membered ring the ring being unsaturated

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Immunology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Polyurethanes Or Polyureas (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
FI943799A 1993-08-19 1994-08-18 Menetelmä terapeuttisesti käyttökelpoisten fenoksifenyylisyklopentenyylihydroksiureayhdisteiden valmistamiseksi FI114466B (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP20545393 1993-08-19
JP20545393 1993-08-19

Publications (3)

Publication Number Publication Date
FI943799A0 FI943799A0 (fi) 1994-08-18
FI943799L true FI943799L (fi) 1995-02-20
FI114466B FI114466B (fi) 2004-10-29

Family

ID=16507136

Family Applications (1)

Application Number Title Priority Date Filing Date
FI943799A FI114466B (fi) 1993-08-19 1994-08-18 Menetelmä terapeuttisesti käyttökelpoisten fenoksifenyylisyklopentenyylihydroksiureayhdisteiden valmistamiseksi

Country Status (27)

Country Link
US (1) US5792882A (fi)
EP (1) EP0720598B1 (fi)
JP (1) JP2794343B2 (fi)
KR (1) KR0170623B1 (fi)
CN (1) CN1077568C (fi)
AT (1) ATE171939T1 (fi)
AU (1) AU674776B2 (fi)
BR (1) BR9407314A (fi)
CA (1) CA2169066C (fi)
CO (1) CO4230229A1 (fi)
CZ (1) CZ288358B6 (fi)
DE (1) DE69413831T2 (fi)
DK (1) DK0720598T3 (fi)
EC (1) ECSP941144A (fi)
EG (1) EG20530A (fi)
ES (1) ES2121218T3 (fi)
FI (1) FI114466B (fi)
IL (1) IL110628A (fi)
MY (1) MY111140A (fi)
NO (1) NO305595B1 (fi)
NZ (1) NZ269849A (fi)
PE (1) PE57194A1 (fi)
PL (1) PL176223B1 (fi)
RU (1) RU2125987C1 (fi)
TW (2) TW418089B (fi)
WO (1) WO1995005360A1 (fi)
ZA (1) ZA946253B (fi)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL317873A1 (en) * 1994-06-27 1997-04-28 Cytomed Inc Compounds for and method of treating cardiovascular, inflammatory and immunological disorders
ATE184272T1 (de) * 1994-11-10 1999-09-15 Pfizer Aryloxycycloalkenyl- und aryloxyiminocycloalkenyl-hydroxyharnstoffe mit 5-lipoxygenase inhibierender wirkung
WO1996016054A1 (en) * 1994-11-18 1996-05-30 Pfizer Pharmaceuticals Inc. Cycloalkenyl-n-hydroxyureas
EP1741424B1 (en) 1997-08-11 2018-10-03 Pfizer Products Inc. Solid pharmaceutical dispersions with enhanced bioavailabilty
US6121323A (en) * 1997-12-03 2000-09-19 3M Innovative Properties Company Bishydroxyureas
KR100879423B1 (ko) 2004-12-02 2009-01-19 (주)아모레퍼시픽 Tnf-알파의 생산을 저해하는 2-사이클로펜텐-1-온 옥심유도체
KR101494488B1 (ko) 2007-12-03 2015-02-24 (주)아모레퍼시픽 2-사이클로펜텐-1-온 옥심 유도체를 유효성분으로 포함하는 지방대사질환 예방 및 치료용 약학 조성물
MX2011008303A (es) 2009-04-03 2011-11-29 Plexxikon Inc Composiciones del acido propano-1-sulfonico {3-[5-(4-cloro-fenil)- 1h-pirrolo [2,3-b]-piridina-3-carbonil]-2,4-difluoro-fenil}-amida y el uso de las mismas.
US8512464B2 (en) * 2009-12-02 2013-08-20 3M Innovative Properties Company Functionalized zirconia nanoparticles and high index films made therefrom

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ222168A (en) * 1986-10-20 1991-05-28 Oncogene Science Inc Tumour growth inhibiting protein related to tgf-#b#1 and tgf-#b#2, preparation by genetic engineering methods, antibodies and pharmaceutical compositions
US5026729A (en) * 1987-02-10 1991-06-25 Abbott Laboratories Lipoxygenase inhibiting compounds
FI900536A7 (fi) * 1989-02-03 1990-08-04 The Wellcome Foundation Ltd Tulehdusta ehkäiseviä aryyliyhdisteitä
US5120752A (en) * 1989-12-28 1992-06-09 Abbott Laboratories Cyclopropyl derivative lipoxygenase inhibitors
US5037853A (en) * 1989-12-28 1991-08-06 Abbott Laboratories Cyclopropyl derivative lipoxygenase inhibitors
GB9025514D0 (en) * 1990-11-23 1991-01-09 Wellcome Found Anti-inflammatory compounds
JP3007138B2 (ja) * 1990-11-27 2000-02-07 ファイザー製薬株式会社 新規なヒドロキサム酸とn―ヒドロキシ尿素誘導体およびそれらの組成物
JPH06256285A (ja) * 1990-12-11 1994-09-13 Pfizer Pharmaceut Co Ltd ヒドロキサム酸誘導体およびその用途
US5130485A (en) * 1991-04-23 1992-07-14 Eli Lilly And Company N-hydroxy-N-(3-(2-substituted phenyl)prop-2-enyl)ureas and thioureas useful as 5-lipoxygenase inhibiting agents
US5149097A (en) * 1991-05-01 1992-09-22 Tonello John H Crossword puzzle aid
JPH05163229A (ja) * 1991-12-13 1993-06-29 Pfizer Pharmaceut Co Ltd 新規なシクロプロピル誘導体
JPH05294921A (ja) * 1992-04-17 1993-11-09 Pfizer Pharmaceut Co Ltd 新規なフェニル置換シクロアルキル尿素誘導体および組成物

Also Published As

Publication number Publication date
NO305595B1 (no) 1999-06-28
US5792882A (en) 1998-08-11
WO1995005360A1 (en) 1995-02-23
CZ48396A3 (en) 1996-07-17
CA2169066A1 (en) 1995-02-23
BR9407314A (pt) 1996-04-16
PL176223B1 (pl) 1999-05-31
JPH08511031A (ja) 1996-11-19
AU674776B2 (en) 1997-01-09
DE69413831T2 (de) 1999-02-25
CN1077568C (zh) 2002-01-09
ECSP941144A (es) 1995-02-27
JP2794343B2 (ja) 1998-09-03
IL110628A (en) 1998-12-27
EG20530A (en) 1999-07-31
NZ269849A (en) 1997-10-24
PL313037A1 (en) 1996-05-27
CO4230229A1 (es) 1995-10-19
CZ288358B6 (en) 2001-05-16
TW418089B (en) 2001-01-11
PE57194A1 (es) 1995-02-07
CN1129440A (zh) 1996-08-21
ZA946253B (en) 1996-02-19
FI943799A0 (fi) 1994-08-18
EP0720598A1 (en) 1996-07-10
CA2169066C (en) 1999-06-22
FI114466B (fi) 2004-10-29
TW448144B (en) 2001-08-01
AU7350994A (en) 1995-03-14
NO960631L (no) 1996-02-16
DE69413831D1 (de) 1998-11-12
ES2121218T3 (es) 1998-11-16
ATE171939T1 (de) 1998-10-15
KR960703845A (ko) 1996-08-31
KR0170623B1 (ko) 1999-03-30
DK0720598T3 (da) 1999-06-21
EP0720598B1 (en) 1998-10-07
NO960631D0 (no) 1996-02-16
MY111140A (en) 1999-08-30
IL110628A0 (en) 1994-11-11
RU2125987C1 (ru) 1999-02-10

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