EP2258357A3 - Neurogenese mit Acetylcholinesterasehemmer - Google Patents
Neurogenese mit Acetylcholinesterasehemmer Download PDFInfo
- Publication number
- EP2258357A3 EP2258357A3 EP10009738A EP10009738A EP2258357A3 EP 2258357 A3 EP2258357 A3 EP 2258357A3 EP 10009738 A EP10009738 A EP 10009738A EP 10009738 A EP10009738 A EP 10009738A EP 2258357 A3 EP2258357 A3 EP 2258357A3
- Authority
- EP
- European Patent Office
- Prior art keywords
- neurogenesis
- acetylcholinesterase inhibitor
- ache
- stimulate
- stimulating
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 230000004766 neurogenesis Effects 0.000 title abstract 2
- 229940100578 Acetylcholinesterase inhibitor Drugs 0.000 title 1
- 239000000544 cholinesterase inhibitor Substances 0.000 title 1
- 108090000371 Esterases Proteins 0.000 abstract 1
- 102000014415 Muscarinic acetylcholine receptor Human genes 0.000 abstract 1
- 108050003473 Muscarinic acetylcholine receptor Proteins 0.000 abstract 1
- OIPILFWXSMYKGL-UHFFFAOYSA-N acetylcholine Chemical compound CC(=O)OCC[N+](C)(C)C OIPILFWXSMYKGL-UHFFFAOYSA-N 0.000 abstract 1
- 229960004373 acetylcholine Drugs 0.000 abstract 1
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- 210000003169 central nervous system Anatomy 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 230000005764 inhibitory process Effects 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 230000001272 neurogenic effect Effects 0.000 abstract 1
- 210000002569 neuron Anatomy 0.000 abstract 1
- 210000001428 peripheral nervous system Anatomy 0.000 abstract 1
- 230000004936 stimulating effect Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/325—Carbamic acids; Thiocarbamic acids; Anhydrides or salts thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/473—Quinolines; Isoquinolines ortho- or peri-condensed with carbocyclic ring systems, e.g. acridines, phenanthridines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US71184605P | 2005-08-26 | 2005-08-26 | |
| US72712705P | 2005-10-14 | 2005-10-14 | |
| US73813305P | 2005-11-17 | 2005-11-17 | |
| US80382606P | 2006-06-02 | 2006-06-02 | |
| EP06813787A EP1928437A2 (de) | 2005-08-26 | 2006-08-25 | Neurogenese mittels muscarinrezeptormodulation |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EP06813787.6 Division | 2006-08-25 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| EP2258357A2 EP2258357A2 (de) | 2010-12-08 |
| EP2258357A3 true EP2258357A3 (de) | 2011-04-06 |
Family
ID=43084447
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EP10009738A Withdrawn EP2258357A3 (de) | 2005-08-26 | 2006-08-25 | Neurogenese mit Acetylcholinesterasehemmer |
| EP10009740A Withdrawn EP2258359A3 (de) | 2005-08-26 | 2006-08-25 | Neurogenese durch Modulation des Muscarinrezeptors mit Sabcomelin |
| EP10009739A Withdrawn EP2258358A3 (de) | 2005-08-26 | 2006-08-25 | Neurogenese mit Acetylcholinesterasehemmer |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EP10009740A Withdrawn EP2258359A3 (de) | 2005-08-26 | 2006-08-25 | Neurogenese durch Modulation des Muscarinrezeptors mit Sabcomelin |
| EP10009739A Withdrawn EP2258358A3 (de) | 2005-08-26 | 2006-08-25 | Neurogenese mit Acetylcholinesterasehemmer |
Country Status (1)
| Country | Link |
|---|---|
| EP (3) | EP2258357A3 (de) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2013044123A1 (en) * | 2011-09-23 | 2013-03-28 | Neupyramid Biotechnology Llc | Uses of bis(3)-cognitin and related compounds |
| WO2013158837A1 (en) * | 2012-04-18 | 2013-10-24 | Concourse Health Sciences Llc | Methods and compositions for treatment of attention deficit hyperactivity disorder |
| BR112017025664A2 (pt) | 2015-06-22 | 2018-08-07 | Nestec Sa | composições e métodos para aumentar a neurogênese em animais |
Citations (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20010036949A1 (en) * | 2000-05-09 | 2001-11-01 | Coe Jotham Wadsworth | Pharmaceutical composition and method of treatment of diseases of cognitive dysfunction in a mammal |
| WO2004034963A2 (en) * | 2002-05-17 | 2004-04-29 | Eisai Co., Ltd. | Methods and compositions using cholinesterase inhibitors |
| WO2004101603A1 (en) * | 2003-05-13 | 2004-11-25 | Boehringer Ingelheim International Gmbh | Statine derivatives for the treatment of alzheimer's disease |
| WO2005005439A1 (en) * | 2003-07-09 | 2005-01-20 | Suven Life Sciences Limited | Benzothiazino indoles |
| EP1541197A1 (de) * | 2003-12-02 | 2005-06-15 | B&B Beheer NV | Verwendung von D4 und 5-HT2A Antagonisten, inverse Agonisten oder partielle Agonisten |
| WO2005072713A2 (en) * | 2004-01-27 | 2005-08-11 | The Feinstein Institute For Medical Research | Cholinesterase inhibitors for treating inflammation |
| WO2006048294A1 (en) * | 2004-11-05 | 2006-05-11 | Novartis Ag | Combinations of nicotinic acetylcholine alpha 7 receptor agonists |
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Also Published As
| Publication number | Publication date |
|---|---|
| EP2258359A3 (de) | 2011-04-06 |
| EP2258359A2 (de) | 2010-12-08 |
| EP2258357A2 (de) | 2010-12-08 |
| EP2258358A2 (de) | 2010-12-08 |
| EP2258358A3 (de) | 2011-09-07 |
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