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EE200300237A - Difenüülasetidinooni derivaadid, nende kasutamine, ravim ja selle valmistamismeetod - Google Patents

Difenüülasetidinooni derivaadid, nende kasutamine, ravim ja selle valmistamismeetod

Info

Publication number
EE200300237A
EE200300237A EEP200300237A EEP200300237A EE200300237A EE 200300237 A EE200300237 A EE 200300237A EE P200300237 A EEP200300237 A EE P200300237A EE P200300237 A EEP200300237 A EE P200300237A EE 200300237 A EE200300237 A EE 200300237A
Authority
EE
Estonia
Prior art keywords
drug
preparation
azetidinone derivatives
diphenyl azetidinone
diphenyl
Prior art date
Application number
EEP200300237A
Other languages
English (en)
Inventor
Glombik Heiner
Kramer Werner
Flohr Stefanie
Frick Wendelin
Heuer Hubert
Jaehne Gerhard
Lindenschmidt Andreas
Schaefer Hans-Ludwig
Original Assignee
Aventis Pharma Deutschland Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE10064402A external-priority patent/DE10064402A1/de
Priority claimed from DE2001154520 external-priority patent/DE10154520A1/de
Application filed by Aventis Pharma Deutschland Gmbh filed Critical Aventis Pharma Deutschland Gmbh
Publication of EE200300237A publication Critical patent/EE200300237A/et

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
EEP200300237A 2000-12-21 2001-12-11 Difenüülasetidinooni derivaadid, nende kasutamine, ravim ja selle valmistamismeetod EE200300237A (et)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10064402A DE10064402A1 (de) 2000-12-21 2000-12-21 Diphenylazetidinonderivate, Verfahren zu deren Herstellung, diese Verbindungen enthaltende Arzneimittel und deren Verwendung
DE2001154520 DE10154520A1 (de) 2001-11-07 2001-11-07 Diphenylazetidinonderivate, Verfahren zu deren Herstellung, diese Verbindungen enthaltende Arzneimittel und deren Verwendung
PCT/EP2001/014532 WO2002050068A1 (de) 2000-12-21 2001-12-11 Diphenylazetidinonderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung

Publications (1)

Publication Number Publication Date
EE200300237A true EE200300237A (et) 2003-08-15

Family

ID=26008045

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200300237A EE200300237A (et) 2000-12-21 2001-12-11 Difenüülasetidinooni derivaadid, nende kasutamine, ravim ja selle valmistamismeetod

Country Status (23)

Country Link
US (1) US6498156B2 (et)
EP (1) EP1345932B1 (et)
JP (1) JP2004516293A (et)
KR (1) KR20030061462A (et)
CN (1) CN1222522C (et)
AR (1) AR034282A1 (et)
AT (1) ATE342899T1 (et)
AU (2) AU1917302A (et)
BR (1) BR0116482A (et)
CA (1) CA2431985A1 (et)
CZ (1) CZ20031731A3 (et)
DE (1) DE50111293D1 (et)
EE (1) EE200300237A (et)
HR (1) HRP20030499A2 (et)
HU (1) HUP0401067A2 (et)
IL (1) IL156552A0 (et)
MX (1) MXPA03005018A (et)
NO (1) NO20032733L (et)
NZ (1) NZ526592A (et)
PL (1) PL362173A1 (et)
SK (1) SK7812003A3 (et)
WO (1) WO2002050068A1 (et)
YU (1) YU46903A (et)

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US7053080B2 (en) 2001-09-21 2006-05-30 Schering Corporation Methods and therapeutic combinations for the treatment of obesity using sterol absorption inhibitors
US7056906B2 (en) 2001-09-21 2006-06-06 Schering Corporation Combinations of hormone replacement therapy composition(s) and sterol absorption inhibitor(s) and treatments for vascular conditions in post-menopausal women
US20030119808A1 (en) * 2001-09-21 2003-06-26 Schering Corporation Methods of treating or preventing cardiovascular conditions while preventing or minimizing muscular degeneration side effects
DE60216300T2 (de) 2001-09-21 2007-06-28 Schering Corp. Behandlung von xanthom mittels azetidinon-derivate als hemmer der sterol absorption
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US7671047B2 (en) 2002-06-19 2010-03-02 Sanofi-Aventis Deutschland Gmbh Cationically substituted diphenylazetidinones, process for their preparation, medicaments comprising these compounds, and their use
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Also Published As

Publication number Publication date
JP2004516293A (ja) 2004-06-03
US6498156B2 (en) 2002-12-24
BR0116482A (pt) 2004-02-03
MXPA03005018A (es) 2003-09-25
AU2002219173B2 (en) 2006-06-22
CN1222522C (zh) 2005-10-12
EP1345932A1 (de) 2003-09-24
NO20032733L (no) 2003-08-14
WO2002050068A1 (de) 2002-06-27
ATE342899T1 (de) 2006-11-15
PL362173A1 (en) 2004-10-18
HRP20030499A2 (en) 2005-04-30
IL156552A0 (en) 2004-01-04
DE50111293D1 (de) 2006-11-30
EP1345932B1 (de) 2006-10-18
NZ526592A (en) 2004-11-26
NO20032733D0 (no) 2003-06-16
CZ20031731A3 (cs) 2003-09-17
HK1059936A1 (en) 2004-07-23
HUP0401067A2 (hu) 2004-09-28
AR034282A1 (es) 2004-02-18
SK7812003A3 (en) 2004-01-08
US20020128252A1 (en) 2002-09-12
AU1917302A (en) 2002-07-01
CA2431985A1 (en) 2002-06-27
KR20030061462A (ko) 2003-07-18
YU46903A (sh) 2006-05-25
CN1481381A (zh) 2004-03-10

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