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EE200300145A - Asa- ja polüasanaftalenüülkarboksamiidid ja farmatseutiline kompositsioon - Google Patents

Asa- ja polüasanaftalenüülkarboksamiidid ja farmatseutiline kompositsioon

Info

Publication number
EE200300145A
EE200300145A EEP200300145A EEP200300145A EE200300145A EE 200300145 A EE200300145 A EE 200300145A EE P200300145 A EEP200300145 A EE P200300145A EE P200300145 A EEP200300145 A EE P200300145A EE 200300145 A EE200300145 A EE 200300145A
Authority
EE
Estonia
Prior art keywords
polyazanaphthalenylcarboxamides
aza
pharmaceutical composition
pharmaceutical
composition
Prior art date
Application number
EEP200300145A
Other languages
English (en)
Inventor
J. Anthony Neville
P. Gomez Robert
D. Young Steven
Egbertson Melissa
S. Wai John
Zhuang Linghang
Embrey Mark
Tran Lekhanh
Y. Melamed Jeffrey
Marie Langford H.
P. Guare James
E. Fisher Thorsten
M. Jolly Samson
S. Kuo Michelle
S. Perlow Debra
J. Bennett Jennifer
W. Funk Timothy
Original Assignee
Merck & Co., Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co., Inc. filed Critical Merck & Co., Inc.
Publication of EE200300145A publication Critical patent/EE200300145A/et

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Virology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
EEP200300145A 2000-10-12 2001-10-09 Asa- ja polüasanaftalenüülkarboksamiidid ja farmatseutiline kompositsioon EE200300145A (et)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US23970700P 2000-10-12 2000-10-12
US28165601P 2001-04-05 2001-04-05
PCT/US2001/042564 WO2002030931A2 (en) 2000-10-12 2001-10-09 Aza- and polyaza-naphthalenyl carboxamides useful as hiv integrase inhibitors

Publications (1)

Publication Number Publication Date
EE200300145A true EE200300145A (et) 2003-06-16

Family

ID=26932782

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200300145A EE200300145A (et) 2000-10-12 2001-10-09 Asa- ja polüasanaftalenüülkarboksamiidid ja farmatseutiline kompositsioon

Country Status (26)

Country Link
US (2) US6921759B2 (et)
EP (1) EP1326865B1 (et)
JP (1) JP4252797B2 (et)
KR (1) KR20030036922A (et)
CN (1) CN1469878A (et)
AR (1) AR033845A1 (et)
AT (1) ATE430745T1 (et)
AU (3) AU2002211527B2 (et)
BG (1) BG107677A (et)
BR (1) BR0114610A (et)
CA (1) CA2425440C (et)
CZ (1) CZ20031028A3 (et)
DE (1) DE60138635D1 (et)
EA (1) EA200300449A1 (et)
EE (1) EE200300145A (et)
HU (1) HUP0302367A2 (et)
IL (1) IL155089A0 (et)
IS (1) IS6760A (et)
MX (1) MXPA03003263A (et)
NO (1) NO20031672L (et)
NZ (1) NZ525088A (et)
PE (1) PE20020509A1 (et)
PL (1) PL360944A1 (et)
SK (1) SK4322003A3 (et)
WO (2) WO2002030931A2 (et)
YU (1) YU27903A (et)

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CN115710249B (zh) * 2022-11-14 2024-11-19 广东工业大学 一种多取代异喹啉和1,6-萘啶化合物的制备方法及光电材料常见分子骨架
CN119841471B (zh) * 2025-03-24 2025-06-03 杭州汇能实业有限公司 一种热镀锌冷却循环水的处理方法

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Also Published As

Publication number Publication date
US20050176718A1 (en) 2005-08-11
MXPA03003263A (es) 2003-06-06
IS6760A (is) 2003-03-27
WO2002030930A2 (en) 2002-04-18
JP4252797B2 (ja) 2009-04-08
ATE430745T1 (de) 2009-05-15
BG107677A (bg) 2003-11-28
PE20020509A1 (es) 2002-06-20
JP2004511483A (ja) 2004-04-15
CA2425440A1 (en) 2002-04-18
EP1326865A2 (en) 2003-07-16
NO20031672L (no) 2003-06-05
IL155089A0 (en) 2003-10-31
AU1152702A (en) 2002-04-22
EP1326865B1 (en) 2009-05-06
CA2425440C (en) 2010-04-13
PL360944A1 (en) 2004-09-20
WO2002030931A2 (en) 2002-04-18
WO2002030930A3 (en) 2002-08-29
CZ20031028A3 (cs) 2003-08-13
SK4322003A3 (en) 2003-09-11
DE60138635D1 (de) 2009-06-18
KR20030036922A (ko) 2003-05-09
YU27903A (sh) 2006-05-25
US20030055071A1 (en) 2003-03-20
NO20031672D0 (no) 2003-04-11
AU2002211527B2 (en) 2006-08-24
HUP0302367A2 (hu) 2003-11-28
NZ525088A (en) 2004-11-26
AR033845A1 (es) 2004-01-07
WO2002030931A3 (en) 2002-10-24
EA200300449A1 (ru) 2003-10-30
AU2002211874A1 (en) 2002-04-22
BR0114610A (pt) 2005-12-13
CN1469878A (zh) 2004-01-21
US6921759B2 (en) 2005-07-26

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