EE05195B1 - Kinoliini ja kinolinooni derivaadid glutamaatretseptori antagonistidena, nende saamine ja kasutamine ravimite valmistamiseks ning neid sisaldav farmatseutiline kompositsioon - Google Patents
Kinoliini ja kinolinooni derivaadid glutamaatretseptori antagonistidena, nende saamine ja kasutamine ravimite valmistamiseks ning neid sisaldav farmatseutiline kompositsioonInfo
- Publication number
- EE05195B1 EE05195B1 EEP200300126A EEP200300126A EE05195B1 EE 05195 B1 EE05195 B1 EE 05195B1 EE P200300126 A EEP200300126 A EE P200300126A EE P200300126 A EEP200300126 A EE P200300126A EE 05195 B1 EE05195 B1 EE 05195B1
- Authority
- EE
- Estonia
- Prior art keywords
- preparation
- quinoline
- pharmaceuticals
- pharmaceutical composition
- composition containing
- Prior art date
Links
- SMWDFEZZVXVKRB-UHFFFAOYSA-N Quinoline Chemical compound N1=CC=CC2=CC=CC=C21 SMWDFEZZVXVKRB-UHFFFAOYSA-N 0.000 title 2
- 239000003814 drug Substances 0.000 title 1
- 239000003825 glutamate receptor antagonist Substances 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- LISFMEBWQUVKPJ-UHFFFAOYSA-N quinolin-2-ol Chemical class C1=CC=C2NC(=O)C=CC2=C1 LISFMEBWQUVKPJ-UHFFFAOYSA-N 0.000 title 1
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- C07D215/04—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to the ring carbon atoms
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- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP00203419 | 2000-10-02 | ||
| PCT/EP2001/011135 WO2002028837A1 (en) | 2000-10-02 | 2001-09-25 | Metabotropic glutamate receptor antagonists |
Publications (2)
| Publication Number | Publication Date |
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| EE200300126A EE200300126A (et) | 2005-04-15 |
| EE05195B1 true EE05195B1 (et) | 2009-08-17 |
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| Application Number | Title | Priority Date | Filing Date |
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| EEP200300126A EE05195B1 (et) | 2000-10-02 | 2001-09-25 | Kinoliini ja kinolinooni derivaadid glutamaatretseptori antagonistidena, nende saamine ja kasutamine ravimite valmistamiseks ning neid sisaldav farmatseutiline kompositsioon |
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| EP (1) | EP1332133B1 (et) |
| JP (1) | JP2004510764A (et) |
| KR (1) | KR100818965B1 (et) |
| CN (1) | CN1703403A (et) |
| AR (1) | AR035065A1 (et) |
| AT (1) | ATE400558T1 (et) |
| AU (2) | AU2001293847B2 (et) |
| BG (1) | BG107672A (et) |
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| DE (1) | DE60134762D1 (et) |
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| US5475007A (en) * | 1993-05-28 | 1995-12-12 | The Regents Of The University Of California | 1,2,3,4-tetrahydroquinoline-2,3,4-trione-3 or 4-oximes and the use thereof |
| JPH0733743A (ja) * | 1993-07-22 | 1995-02-03 | Kyorin Pharmaceut Co Ltd | 2−アリール−4−キノリノール誘導体 |
| JPH08295690A (ja) * | 1995-04-26 | 1996-11-12 | Tokuyama Corp | クロメン化合物 |
| JP2000511532A (ja) * | 1996-05-20 | 2000-09-05 | メルク エンド カンパニー インコーポレーテッド | 性腺刺激ホルモン放出ホルモンのアンタゴニスト |
| WO1999003822A1 (en) | 1997-07-18 | 1999-01-28 | Georgetown University | Bicyclic metabotropic glutamate receptor ligands |
| EP1037878A2 (en) | 1997-11-21 | 2000-09-27 | Nps Pharmaceuticals, Inc. | Metabotropic glutamate receptor antagonists for treating central nervous system diseases |
| BR9913315A (pt) * | 1998-08-27 | 2001-05-22 | Pfizer Prod Inc | Derivados de quinolin-2-ona úteis como agentes anticâncer |
| JP2000169450A (ja) | 1998-09-30 | 2000-06-20 | Kyorin Pharmaceut Co Ltd | 6―アリ―ルキノリンカルボン酸誘導体とその付加塩及びそれらの製造方法 |
| HU229404B1 (en) * | 1998-12-23 | 2013-12-30 | Janssen Pharmaceutica Nv | 1,2-annelated quinoline derivatives |
| DE19859750A1 (de) | 1998-12-23 | 2000-06-29 | Henkel Kgaa | Mittel zum Färben von keratinhaltigen Fasern |
| ID29584A (id) * | 1999-02-11 | 2001-09-06 | Pfizer Prod Inc | Turunan-turunan kuinolin-2-on tersubstitusi heteroaril yang bermanfaat sebagai zat-zat anti kanker |
| CA2402096A1 (en) | 2000-03-07 | 2001-09-13 | Takeda Chemical Industries, Ltd. | Vasoactive agents |
| EA007464B1 (ru) * | 2000-10-02 | 2006-10-27 | Янссен Фармацевтика Н.В. | Антагонисты метаботропных рецепторов глутамата |
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