DZ3327A1 - Derives de benzimidazole nouveaux utiles comme agents antiproliferatifs. - Google Patents

Derives de benzimidazole nouveaux utiles comme agents antiproliferatifs.

Info

Publication number: DZ3327A1
Authority: DZ; Algeria
Prior art keywords: benzimidazole derivatives; derivatives useful; antiproliferative agents; new benzimidazole; new
Prior art date: 1999-11-30

Application number

DZ003327A

Other languages

English (en)

Inventor

Wayne Ernest Barth

Michael Joseph Luzzio

Joseph Peter Lyssikatos

Original Assignee

Pfizer Prod Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-11-30

Filing date

2000-11-10

Publication date

2001-06-07

2000-11-10 Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc

2001-06-07 Application granted granted Critical

2001-06-07 Publication of DZ3327A1 publication Critical patent/DZ3327A1/fr

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
- A—HUMAN NECESSITIES
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61P9/08—Vasodilators for multiple indications
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/10—Spiro-condensed systems

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Immunology (AREA)
Urology & Nephrology (AREA)
Dermatology (AREA)
Diabetes (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Pulmonology (AREA)
Neurology (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Rheumatology (AREA)
Hematology (AREA)
Endocrinology (AREA)
Transplantation (AREA)
Psychiatry (AREA)
Vascular Medicine (AREA)
Emergency Medicine (AREA)
Oncology (AREA)
Ophthalmology & Optometry (AREA)
Hospice & Palliative Care (AREA)
Pain & Pain Management (AREA)
Obesity (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

DZ003327A 1999-11-30 2000-11-10 Derives de benzimidazole nouveaux utiles comme agents antiproliferatifs. DZ3327A1 (fr)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US16821799P	1999-11-30	1999-11-30
PCT/IB2000/001636 WO2001040217A1 (fr)	1999-11-30	2000-11-10	Nouveaux derives benzoimidazole convenant comme agents antiproliferatifs

Publications (1)

Publication Number	Publication Date
DZ3327A1 true DZ3327A1 (fr)	2001-06-07

Family

ID=22610585

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DZ003327A DZ3327A1 (fr)	1999-11-30	2000-11-10	Derives de benzimidazole nouveaux utiles comme agents antiproliferatifs.

Country Status (47)

Country	Link
US (1)	US7019147B1 (fr)
EP (1)	EP1235825B1 (fr)
JP (2)	JP4522635B2 (fr)
KR (1)	KR100479401B1 (fr)
CN (2)	CN101289442A (fr)
AP (1)	AP1895A (fr)
AR (1)	AR026633A1 (fr)
AT (1)	ATE316528T1 (fr)
AU (1)	AU782077B2 (fr)
BG (1)	BG65862B1 (fr)
BR (1)	BR0015911A (fr)
CA (1)	CA2392973C (fr)
CO (1)	CO5251455A1 (fr)
CR (1)	CR6643A (fr)
CU (1)	CU23132A3 (fr)
CZ (1)	CZ300789B6 (fr)
DE (1)	DE60025747T2 (fr)
DK (1)	DK1235825T3 (fr)
DZ (1)	DZ3327A1 (fr)
EA (1)	EA005407B1 (fr)
EE (1)	EE05350B1 (fr)
EG (1)	EG24433A (fr)
ES (1)	ES2256052T3 (fr)
GE (1)	GEP20033141B (fr)
GT (1)	GT200000198A (fr)
HR (1)	HRP20020475B1 (fr)
HU (1)	HU230829B1 (fr)
IL (2)	IL149841A0 (fr)
IS (1)	IS2209B (fr)
MA (1)	MA26847A1 (fr)
MX (1)	MXPA02005343A (fr)
MY (1)	MY128765A (fr)
NO (1)	NO324043B1 (fr)
NZ (1)	NZ518280A (fr)
PA (1)	PA8507601A1 (fr)
PE (1)	PE20010899A1 (fr)
PL (1)	PL201784B1 (fr)
RS (1)	RS50800B (fr)
SI (1)	SI1235825T1 (fr)
SK (1)	SK286773B6 (fr)
SV (1)	SV2002000232A (fr)
TN (1)	TNSN00228A1 (fr)
TR (1)	TR200201430T2 (fr)
TW (1)	TWI258475B (fr)
UA (1)	UA75055C2 (fr)
WO (1)	WO2001040217A1 (fr)
ZA (1)	ZA200204244B (fr)

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EP2281901B1 (fr)	2005-08-02	2013-11-27	Eisai R&D Management Co., Ltd.	Composition pharmaceutique anti-tumeur avec des inhibiteurs d'angiogénèse
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CN101511793B (zh)	2006-08-28	2011-08-03	卫材R&D管理有限公司	针对未分化型胃癌的抗肿瘤剂
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EA005407B1 (ru)	2005-02-24
NO20022556D0 (no)	2002-05-29
AP1895A (en)	2008-10-08
TWI258475B (en)	2006-07-21
CU23132A3 (es)	2006-05-22
TNSN00228A1 (fr)	2005-11-10
PL201784B1 (pl)	2009-05-29
WO2001040217A1 (fr)	2001-06-07
TR200201430T2 (tr)	2003-01-21
JP2003515603A (ja)	2003-05-07
YU30702A (sh)	2005-06-10
CN1402721A (zh)	2003-03-12
HRP20020475B1 (en)	2007-06-30
MA26847A1 (fr)	2004-12-20
ATE316528T1 (de)	2006-02-15
MY128765A (en)	2007-02-28
ZA200204244B (en)	2003-05-28
DE60025747D1 (de)	2006-04-13
EP1235825B1 (fr)	2006-01-25
CA2392973C (fr)	2007-05-15
US7019147B1 (en)	2006-03-28
HUP0203725A3 (en)	2004-05-28
DE60025747T2 (de)	2006-08-31
ES2256052T3 (es)	2006-07-16
EA200200509A1 (ru)	2002-10-31
GEP20033141B (en)	2003-12-25
CR6643A (es)	2003-11-07
NO324043B1 (no)	2007-07-30
HU230829B1 (en)	2018-08-28
CN101289442A (zh)	2008-10-22
SI1235825T1 (sl)	2006-06-30
AU1048001A (en)	2001-06-12
GT200000198A (es)	2002-05-23
JP4522635B2 (ja)	2010-08-11
BG106812A (bg)	2003-01-31
CZ20021759A3 (cs)	2003-06-18
IS2209B (is)	2007-02-15
SK286773B6 (sk)	2009-05-07
AR026633A1 (es)	2003-02-19
NZ518280A (en)	2004-05-28
KR100479401B1 (ko)	2005-03-28
RS50800B (sr)	2010-08-31
KR20020059827A (ko)	2002-07-13
JP2007126468A (ja)	2007-05-24
HRP20020475A2 (en)	2005-10-31
EP1235825A1 (fr)	2002-09-04
IL149841A0 (en)	2002-11-10
MXPA02005343A (es)	2002-12-11
UA75055C2 (uk)	2006-03-15
PL355917A1 (en)	2004-05-31
PA8507601A1 (es)	2003-02-14
CZ300789B6 (cs)	2009-08-12
AP2002002529A0 (en)	2002-06-30
PE20010899A1 (es)	2001-09-05
CO5251455A1 (es)	2003-02-28
NO20022556L (no)	2002-07-29
EG24433A (en)	2009-06-25
CA2392973A1 (fr)	2001-06-07
IS6341A (is)	2002-04-12
EE200200276A (et)	2003-06-16
HUP0203725A2 (hu)	2003-02-28
AU782077B2 (en)	2005-06-30
DK1235825T3 (da)	2006-05-15
IL149841A (en)	2008-07-08
EE05350B1 (et)	2010-10-15
BR0015911A (pt)	2002-08-06
SK7172002A3 (en)	2004-07-07
BG65862B1 (bg)	2010-03-31
SV2002000232A (es)	2002-06-07

Publication	Publication Date	Title
DZ3327A1 (fr)	2001-06-07	Derives de benzimidazole nouveaux utiles comme agents antiproliferatifs.
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PT1177185E (pt)	2005-08-31	Derivados de 4, 5, 6, 7-tetra-hidroindazole como agentes antitumorais
MA26832A1 (fr)	2004-12-20	Derives de benzodiazepine.
TR200000520A3 (tr)	2001-06-21	4-Fenil-piridin türevleri.
DZ3159A1 (fr)	2001-04-19	Derives de purine.
MA26831A1 (fr)	2004-12-20	Derives de benzodiazepine."
MA26932A1 (fr)	2004-12-20	Derives d'imidazole.
MA26794A1 (fr)	2004-12-20	Derives de 5-phenyl-pyrimidine.
PT1218378E (pt)	2003-09-30	Derivados de terc-butil-(7-metil-imidazo-¬1,2-a\|-piridin-3-il)-amina
MA26846A1 (fr)	2004-12-20	Derives de 2,4-diaminopyrimidine utiles comme agents immunosuppresseurs.
MA26816A1 (fr)	2004-12-20	Derives d'amino-triazolopyridine
ATE263748T1 (de)	2004-04-15	Admantan-derivate
IT1316230B1 (it)	2003-04-03	Complesso di essiccazione.
BR0013417B1 (pt)	2013-07-16	composiÇço aquosa.
DE60009154D1 (de)	2004-04-22	Phenylpiperazinyl-derivate
ATE257148T1 (de)	2004-01-15	Propargyletherderivate
ATE219157T1 (de)	2002-06-15	Gleitlager
PT1154988E (pt)	2004-12-31	Derivados de mevinolina
EE200200204A (et)	2003-04-15	Asendatud bensimidasooli preparaat
MA26793A1 (fr)	2004-12-20	Derives de 4-phenyl-pyrimidine.
ATE293592T1 (de)	2005-05-15	Resorcinderivate
DE60025958D1 (de)	2006-04-20	14,15-beta-methylen substituierte androgene
MA26844A1 (fr)	2004-12-20	Nouveaux derives de la thiazolidinedione comme agents antidiabetiques
PT1088818E (pt)	2005-03-31	Derivados de quinolin-4-ilo