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DZ2826A1 - Formulaons intranasales de mésylate de sildénafil et procédé pour leur préparation. - Google Patents

Formulaons intranasales de mésylate de sildénafil et procédé pour leur préparation.

Info

Publication number
DZ2826A1
DZ2826A1 DZ990126A DZ990126A DZ2826A1 DZ 2826 A1 DZ2826 A1 DZ 2826A1 DZ 990126 A DZ990126 A DZ 990126A DZ 990126 A DZ990126 A DZ 990126A DZ 2826 A1 DZ2826 A1 DZ 2826A1
Authority
DZ
Algeria
Prior art keywords
intranasal
formulas
preparation
sildenafil mesylate
sildenafil
Prior art date
Application number
DZ990126A
Other languages
English (en)
Inventor
Anne Billotte
Brian Thomas Henry
Joanna Jayne Woods
Peter James Dunn
Peter Vallance Marshall
Original Assignee
Pfizer Res & Dev Company Nv I
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9813452.1A external-priority patent/GB9813452D0/en
Priority claimed from GBGB9820837.4A external-priority patent/GB9820837D0/en
Priority claimed from GBGB9903177.5A external-priority patent/GB9903177D0/en
Application filed by Pfizer Res & Dev Company Nv I filed Critical Pfizer Res & Dev Company Nv I
Application granted granted Critical
Publication of DZ2826A1 publication Critical patent/DZ2826A1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0043Nose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Reproductive Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Endocrinology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Otolaryngology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DZ990126A 1998-06-22 1999-06-21 Formulaons intranasales de mésylate de sildénafil et procédé pour leur préparation. DZ2826A1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9813452.1A GB9813452D0 (en) 1998-06-22 1998-06-22 Pharmaceutical formulations
GBGB9820837.4A GB9820837D0 (en) 1998-09-24 1998-09-24 Pharmaceutical formulations
GBGB9903177.5A GB9903177D0 (en) 1999-02-13 1999-02-13 Pharmaceutical formulations

Publications (1)

Publication Number Publication Date
DZ2826A1 true DZ2826A1 (fr) 2003-12-01

Family

ID=27269368

Family Applications (1)

Application Number Title Priority Date Filing Date
DZ990126A DZ2826A1 (fr) 1998-06-22 1999-06-21 Formulaons intranasales de mésylate de sildénafil et procédé pour leur préparation.

Country Status (40)

Country Link
US (2) US20020040139A1 (fr)
EP (1) EP0967214B1 (fr)
JP (1) JP3263379B2 (fr)
KR (1) KR100345824B1 (fr)
AP (1) AP1178A (fr)
AR (1) AR016993A1 (fr)
AT (1) ATE269866T1 (fr)
AU (1) AU746865B2 (fr)
BG (1) BG64372B1 (fr)
BR (1) BR9903273A (fr)
CA (1) CA2275554C (fr)
CZ (1) CZ294856B6 (fr)
DE (1) DE69918222T2 (fr)
DK (1) DK0967214T3 (fr)
DZ (1) DZ2826A1 (fr)
EA (1) EA001903B1 (fr)
ES (1) ES2221733T3 (fr)
GT (1) GT199900095A (fr)
HN (1) HN1999000096A (fr)
HR (1) HRP990195B1 (fr)
HU (1) HUP9902076A3 (fr)
ID (1) ID23554A (fr)
IL (1) IL130539A0 (fr)
IS (1) IS5085A (fr)
MA (1) MA25089A1 (fr)
MY (1) MY117967A (fr)
NO (1) NO317365B1 (fr)
NZ (1) NZ336382A (fr)
OA (1) OA11069A (fr)
PA (1) PA8476301A1 (fr)
PE (1) PE20000702A1 (fr)
PT (1) PT967214E (fr)
SG (1) SG77246A1 (fr)
SI (1) SI0967214T1 (fr)
SK (1) SK284574B6 (fr)
TN (1) TNSN99129A1 (fr)
TR (1) TR199901444A2 (fr)
TW (1) TWI223598B (fr)
UA (1) UA59385C2 (fr)
YU (1) YU29699A (fr)

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Also Published As

Publication number Publication date
CZ9902257A3 (cs) 2000-11-15
EA001903B1 (ru) 2001-10-22
DK0967214T3 (da) 2004-09-27
EA199900487A3 (ru) 2000-04-24
JP2000034232A (ja) 2000-02-02
SG77246A1 (en) 2000-12-19
NO993051D0 (no) 1999-06-21
NZ336382A (en) 1999-11-29
EP0967214A1 (fr) 1999-12-29
TR199901444A2 (xx) 2000-01-21
BG64372B1 (bg) 2004-12-30
HRP990195A2 (en) 2000-02-29
HN1999000096A (es) 2000-12-03
IS5085A (is) 1999-12-23
DE69918222D1 (de) 2004-07-29
MA25089A1 (fr) 2000-12-31
YU29699A (sh) 2003-02-28
CA2275554C (fr) 2003-06-03
BR9903273A (pt) 2000-05-09
KR20000006310A (ko) 2000-01-25
PE20000702A1 (es) 2000-08-16
TNSN99129A1 (fr) 2005-11-10
JP3263379B2 (ja) 2002-03-04
UA59385C2 (uk) 2003-09-15
HUP9902076A2 (hu) 2000-05-28
HRP990195B1 (en) 2003-04-30
AP9901585A0 (en) 1999-06-30
SK284574B6 (sk) 2005-06-02
TWI223598B (en) 2004-11-11
SK81999A3 (en) 2001-01-18
NO993051L (no) 1999-12-23
AR016993A1 (es) 2001-08-01
ID23554A (id) 2000-05-04
NO317365B1 (no) 2004-10-18
OA11069A (en) 2002-03-13
US20020040139A1 (en) 2002-04-04
CA2275554A1 (fr) 1999-12-22
ATE269866T1 (de) 2004-07-15
KR100345824B1 (ko) 2002-07-24
HUP9902076A3 (en) 2002-03-28
IL130539A0 (en) 2000-06-01
GT199900095A (es) 2000-12-13
AU746865B2 (en) 2002-05-02
PT967214E (pt) 2004-08-31
US20030158206A1 (en) 2003-08-21
EP0967214B1 (fr) 2004-06-23
SI0967214T1 (en) 2004-10-31
AU3579499A (en) 2000-01-06
MY117967A (en) 2004-08-30
AP1178A (en) 2003-06-30
EA199900487A2 (ru) 1999-12-29
CZ294856B6 (cs) 2005-03-16
BG103510A (en) 2000-01-31
HU9902076D0 (en) 1999-08-30
PA8476301A1 (es) 2000-09-29
DE69918222T2 (de) 2005-07-28
ES2221733T3 (es) 2005-01-01

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