DK2776034T3 - Farmaceutiske sammensætninger omfattende (s)-(+)-7-(1h-imidazol-4-ylmethyl)-5,6,7,8-tetrahydro-quinolin til behandling af hudsygdomme og -tilstande - Google Patents
Farmaceutiske sammensætninger omfattende (s)-(+)-7-(1h-imidazol-4-ylmethyl)-5,6,7,8-tetrahydro-quinolin til behandling af hudsygdomme og -tilstande Download PDFInfo
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- DK2776034T3 DK2776034T3 DK12784857.0T DK12784857T DK2776034T3 DK 2776034 T3 DK2776034 T3 DK 2776034T3 DK 12784857 T DK12784857 T DK 12784857T DK 2776034 T3 DK2776034 T3 DK 2776034T3
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- skin
- dermatitis
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-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/14—Decongestants or antiallergics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
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- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Dermatology (AREA)
- Ophthalmology & Optometry (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cosmetics (AREA)
- Medicinal Preparation (AREA)
Claims (11)
1. Farmaceutisk sammensætning til anvendelse i en fremgangsmåde til behandling af hudtilstande hos en patient, der lider deraf, hvor den farmaceutiske sammensætning omfatter en terapeutisk effektiv mængde af (S)-(+)-7-(lH-Imidazol-4-ylmethyl)-5,6,7,8-tetrahydro-quinolin, eller de individuelle tautomerer deraf, eller et farmaceutisk acceptabelt salt deraf.
2. Den farmaceutiske sammensætning til anvendelse i en fremgangsmåde ifølge krav 1, hvor den behandlede tilstand er valgt fra: rosacea, rosacea fulminans, solskoldning, psoriasis, menopause-associerede hedeture, rødmen og rødhed associeret med hedeture, erytem associeret med hedeture, hedeture som resultat af orchiektomyatopisk dermatitis, behandling af rødhed og kløe fra insektbid, fotoaldring, seboroisk dermatitis, akne, allergisk dermatitis, ansigtstelangiektasi (udvidelser af allerede eksisterende små blodkar), angioektasi, rhinophyma (hypertrofi af næsen med follikulær udvidelse), akne-lignende hududslæt (kan sive ud eller danne skorpe), brændende eller sviende fornemmelse, huderytem, kutan hyperaktivitet med udvidelse af blodkar i huden, Lyells syndrom, Stevens-Johnson syndrom, lokal kløe og ubehag associeret med hæmorroider, hæmorroider, erytem multiform minor, erytem multiform major, erytem nodosum, hævede øjne, urticaria, pruritis, purpura, åreknuder, kontaktdermatitis, atopisk dermatitis, nummulat dermatitis, generaliseret exfoliativ dermatitis, stasedermatitis, lichen simplex chronicus, perioral dermatitis, pseudofolliculitis barbae, granuloma annulare, aktinisk keratose, basal celle karcinom, pladeepithelkarcinomer, og eksem.
3. Den farmaceutiske sammensætning til anvendelse i en fremgangsmåde ifølge krav 1, hvor tilstanden er rosacea.
4. Den farmaceutiske sammensætning til anvendelse i en fremgangsmåde ifølge krav 1, hvor tilstanden er psoriasis.
5. Den farmaceutiske sammensætning til anvendelse i en fremgangsmåde ifølge krav 1, hvor tilstanden er rosacea fulminans.
6. Den farmaceutiske sammensætning til anvendelse i en fremgangsmåde ifølge krav 1, hvor tilstanden er ansigtstelangiektasi.
7. Den farmaceutiske sammensætning til anvendelse i en fremgangsmåde ifølge krav 1, hvor tilstanden er huderytem.
8. Den farmaceutiske sammensætning til anvendelse i en fremgangsmåde ifølge krav 1, hvor tilstanden er solskoldning.
9. Den farmaceutiske sammensætning til anvendelse i en fremgangsmåde ifølge krav 1, hvor tilstanden er kutan hyperaktivitet med udvidelse af blodkar i huden.
10. Den farmaceutiske sammensætning til anvendelse i en fremgangsmåde ifølge krav 1, hvor den farmaceutiske sammensætning er i en formulering egnet til topikal dermatologisk administration.
11. Den farmaceutiske sammensætning til anvendelse i en fremgangsmåde ifølge krav 1, hvor den farmaceutiske sammensætning administreres som en form valgt fra suspensioner, geler, opløsninger, cremer, lotions, salver, skum, emulsioner, mikroemulsioner, mælk, serummer, aerosoler, sprays, dispersioner, mikrokapsler, vesikler, mikropartikler, våde klude, tørre klude, ansigtsklude eller direkte injektion.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161558104P | 2011-11-10 | 2011-11-10 | |
| PCT/US2012/064075 WO2013070861A1 (en) | 2011-11-10 | 2012-11-08 | Pharmaceutical compositions comprising 7-(1h-imidazol-4-ylmethyl)-5,6,7,8-tetrahydro-quinoline for treating skin diseases and conditions |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK2776034T3 true DK2776034T3 (da) | 2017-07-10 |
Family
ID=47178364
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK12784857.0T DK2776034T3 (da) | 2011-11-10 | 2012-11-08 | Farmaceutiske sammensætninger omfattende (s)-(+)-7-(1h-imidazol-4-ylmethyl)-5,6,7,8-tetrahydro-quinolin til behandling af hudsygdomme og -tilstande |
Country Status (22)
| Country | Link |
|---|---|
| US (4) | US20130123303A1 (da) |
| EP (3) | EP3184110B1 (da) |
| JP (2) | JP6359456B2 (da) |
| KR (1) | KR102004563B1 (da) |
| CN (1) | CN104136029A (da) |
| AR (1) | AR088845A1 (da) |
| AU (2) | AU2012335803B2 (da) |
| BR (1) | BR112014011336A2 (da) |
| CA (1) | CA2855005C (da) |
| CL (1) | CL2014001242A1 (da) |
| DK (1) | DK2776034T3 (da) |
| ES (1) | ES2635421T3 (da) |
| IL (3) | IL232483B (da) |
| MX (1) | MX350662B (da) |
| MY (1) | MY182553A (da) |
| PH (1) | PH12014501051A1 (da) |
| RU (2) | RU2630978C2 (da) |
| SG (3) | SG11201402246RA (da) |
| TW (3) | TW202014189A (da) |
| UA (1) | UA109359C2 (da) |
| WO (1) | WO2013070861A1 (da) |
| ZA (1) | ZA201403396B (da) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9283217B2 (en) | 2011-11-10 | 2016-03-15 | Allergan, Inc. | Pharmaceutical compositions comprising 7-(1 H-imidazol-4-ylmethyl)-5,6,7,8-tetrahydro-quinoline for treating skin diseases and conditions |
| CN105188691A (zh) * | 2013-05-06 | 2015-12-23 | 阿勒根公司 | 用于治疗组织创伤的α-肾上腺素能激动剂 |
| FR3061434B1 (fr) * | 2017-01-04 | 2019-07-12 | Pierre Fabre Dermo-Cosmetique | Composition cosmetique comprenant une association d'huile de pongamia et de pentylene glycol 4-t-butylcyclohexanol pour lutter contre la rosacee |
| RU2727695C1 (ru) * | 2020-02-13 | 2020-07-22 | Мурад Умарович Магомедов | Способ комплексного лечения ринофимы |
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| ATE319456T1 (de) * | 1998-05-08 | 2006-03-15 | Univ Miami | Verwendung von tetracyclinen zur behandlung von störungen der meibomschen drüsen |
| US6242442B1 (en) * | 1998-12-17 | 2001-06-05 | Alcon Laboratories, Inc. | Brinzolamide and brimonidine for treating ocular conditions |
| US20010049369A1 (en) * | 2000-02-10 | 2001-12-06 | Jablonski Monica M. | Brimonidine compositions and methods for retinal degeneration |
| US6468989B1 (en) | 2000-07-13 | 2002-10-22 | Dow Pharmaceutical Sciences | Gel compositions containing metronidazole |
| US6387383B1 (en) | 2000-08-03 | 2002-05-14 | Dow Pharmaceutical Sciences | Topical low-viscosity gel composition |
| US20020198209A1 (en) | 2001-05-03 | 2002-12-26 | Allergan Sales Inc. | Compositions having enhanced pharmacokinetic characteristics |
| US6680062B2 (en) | 2001-10-05 | 2004-01-20 | Color Access, Inc. | Anti-irritating rosacea treatment |
| US7030149B2 (en) * | 2002-04-19 | 2006-04-18 | Allergan, Inc. | Combination of brimonidine timolol for topical ophthalmic use |
| US20040146539A1 (en) * | 2003-01-24 | 2004-07-29 | Gupta Shyam K. | Topical Nutraceutical Compositions with Selective Body Slimming and Tone Firming Antiaging Benefits |
| US7439241B2 (en) * | 2003-05-27 | 2008-10-21 | Galderma Laboratories, Inc. | Compounds, formulations, and methods for treating or preventing rosacea |
| US20050020600A1 (en) * | 2003-07-23 | 2005-01-27 | Scherer Warren J. | Methods of treating cutaneous flushing using selective alpha-2-adrenergic receptor agonists |
| EP1689397A4 (en) * | 2003-11-20 | 2007-06-20 | Othera Pharmaceuticals Inc | IMPROVING MACULAR DEGENERATION AND OTHER OPHTHALMIC DISEASES |
| US7812049B2 (en) | 2004-01-22 | 2010-10-12 | Vicept Therapeutics, Inc. | Method and therapeutic/cosmetic topical compositions for the treatment of rosacea and skin erythema using α1-adrenoceptor agonists |
| KR101257046B1 (ko) * | 2004-05-25 | 2013-04-22 | 산스로사 파마슈티칼 디벨로프먼트, 인코포레이티드 | 염증성 피부 질환을 치료하거나 예방하기 위한 화합물,제형 및 방법 |
| US20070203144A1 (en) * | 2006-01-17 | 2007-08-30 | Allergan, Inc. | Use of Memantine and Brimonidine to Attenuate Vitreoretinal Vascular Endothelial Growth Factor (VEGF) Protein Levels in Animals |
| US7323477B2 (en) * | 2006-02-02 | 2008-01-29 | Allergan, Inc. | 7-((1H-imidazol-4-yl)methyl)-5,6,7,8-tetrahydroquinoline |
| RU2321399C1 (ru) * | 2006-06-01 | 2008-04-10 | Федеральное государственное учреждение "Нижегородский научно-исследовательский кожно-венерологический институт Федерального агентства по здравоохранению и социальному развитию" | Способ лечения больных розацеа |
| US20090005450A1 (en) * | 2007-04-09 | 2009-01-01 | Belinda Tsao Nivaggioli | Use of creatine compounds for the treatment of eye disorders |
| US20090061020A1 (en) * | 2007-08-31 | 2009-03-05 | Theobald Klaus P | Brimonidine Compositions for Treating Erythema |
| US8455548B2 (en) * | 2007-10-18 | 2013-06-04 | Allergan, Inc. | Method of treating sensorimotor disorders with alpha-2 adrenergic receptor agonists |
| WO2010014552A1 (en) * | 2008-08-01 | 2010-02-04 | Alpha Synergy Development, Inc. | Vasoconstriction compositions and methods of use |
| US20100203165A1 (en) * | 2008-08-01 | 2010-08-12 | Gerald Horn | Compositions and methods for treatment of disorders or conditions of the eye |
| FR2942138A1 (fr) * | 2009-02-16 | 2010-08-20 | Galderma Res & Dev | Association de composes pour le traitement ou la prevention des affections dermatologiques |
| RU2012122983A (ru) * | 2009-10-26 | 2014-01-27 | Галдерма Фарма С.А. | Способ лечения и профилактики острой эритемы |
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| CA2792649A1 (en) * | 2010-03-26 | 2011-09-29 | Michael Graeber | Improved methods and compositions for safe and effective treatment of telangiectasia |
| MX2012010824A (es) * | 2010-03-26 | 2012-10-10 | Galderma Res & Dev | Metodos y composiciones mejoradas para tratamiento seguro y efectivo del eritema. |
| KR20130128375A (ko) * | 2010-08-06 | 2013-11-26 | 갈데르마 리서치 & 디벨로프먼트 | 피부 질환을 치료 또는 예방하기 위한 화합물들의 배합물 |
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2012
- 2012-08-11 UA UAA201406109A patent/UA109359C2/ru unknown
- 2012-11-08 JP JP2014541225A patent/JP6359456B2/ja active Active
- 2012-11-08 AU AU2012335803A patent/AU2012335803B2/en not_active Ceased
- 2012-11-08 RU RU2014122758A patent/RU2630978C2/ru active
- 2012-11-08 CN CN201280065945.0A patent/CN104136029A/zh active Pending
- 2012-11-08 EP EP17156230.9A patent/EP3184110B1/en active Active
- 2012-11-08 EP EP12784857.0A patent/EP2776034B1/en active Active
- 2012-11-08 ES ES12784857.0T patent/ES2635421T3/es active Active
- 2012-11-08 SG SG11201402246RA patent/SG11201402246RA/en unknown
- 2012-11-08 MY MYPI2014001376A patent/MY182553A/en unknown
- 2012-11-08 MX MX2014005640A patent/MX350662B/es active IP Right Grant
- 2012-11-08 KR KR1020147015533A patent/KR102004563B1/ko not_active Expired - Fee Related
- 2012-11-08 RU RU2017131492A patent/RU2667645C1/ru active
- 2012-11-08 WO PCT/US2012/064075 patent/WO2013070861A1/en not_active Ceased
- 2012-11-08 US US13/672,475 patent/US20130123303A1/en not_active Abandoned
- 2012-11-08 SG SG10201609145PA patent/SG10201609145PA/en unknown
- 2012-11-08 CA CA2855005A patent/CA2855005C/en active Active
- 2012-11-08 BR BR112014011336A patent/BR112014011336A2/pt not_active Application Discontinuation
- 2012-11-08 PH PH1/2014/501051A patent/PH12014501051A1/en unknown
- 2012-11-08 EP EP20193075.7A patent/EP3763370A1/en not_active Withdrawn
- 2012-11-08 DK DK12784857.0T patent/DK2776034T3/da active
- 2012-11-08 SG SG10201809506TA patent/SG10201809506TA/en unknown
- 2012-11-09 TW TW108123351A patent/TW202014189A/zh unknown
- 2012-11-09 TW TW106103338A patent/TWI708604B/zh not_active IP Right Cessation
- 2012-11-09 TW TW101141967A patent/TWI580424B/zh active
- 2012-11-12 AR ARP120104260A patent/AR088845A1/es unknown
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2014
- 2014-05-07 IL IL232483A patent/IL232483B/en active IP Right Grant
- 2014-05-12 CL CL2014001242A patent/CL2014001242A1/es unknown
- 2014-05-12 ZA ZA2014/03396A patent/ZA201403396B/en unknown
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2015
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2016
- 2016-08-17 AU AU2016216627A patent/AU2016216627B2/en not_active Ceased
- 2016-11-16 US US15/353,262 patent/US20170095466A1/en not_active Abandoned
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2017
- 2017-05-08 JP JP2017092572A patent/JP6526737B2/ja active Active
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2018
- 2018-08-21 IL IL261269A patent/IL261269A/en unknown
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2019
- 2019-08-18 IL IL26875719A patent/IL268757A/en unknown
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