CY1113719T1 - Φαρμακευτικο σκευασμα για τη θεραπεια του ανωτερου πεπτικου σωληνα - Google Patents
Φαρμακευτικο σκευασμα για τη θεραπεια του ανωτερου πεπτικου σωληναInfo
- Publication number
- CY1113719T1 CY1113719T1 CY20131100174T CY131100174T CY1113719T1 CY 1113719 T1 CY1113719 T1 CY 1113719T1 CY 20131100174 T CY20131100174 T CY 20131100174T CY 131100174 T CY131100174 T CY 131100174T CY 1113719 T1 CY1113719 T1 CY 1113719T1
- Authority
- CY
- Cyprus
- Prior art keywords
- treatment
- pharmaceutical preparation
- upper dental
- dental tube
- tube
- Prior art date
Links
- 239000000825 pharmaceutical preparation Substances 0.000 title 1
- VOVIALXJUBGFJZ-KWVAZRHASA-N Budesonide Chemical compound C1CC2=CC(=O)C=C[C@]2(C)[C@@H]2[C@@H]1[C@@H]1C[C@H]3OC(CCC)O[C@@]3(C(=O)CO)[C@@]1(C)C[C@@H]2O VOVIALXJUBGFJZ-KWVAZRHASA-N 0.000 abstract 1
- 230000003110 anti-inflammatory effect Effects 0.000 abstract 1
- 229960004436 budesonide Drugs 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 239000007938 effervescent tablet Substances 0.000 abstract 1
- 230000001506 immunosuppresive effect Effects 0.000 abstract 1
- 230000010534 mechanism of action Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
- A61K9/0007—Effervescent
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
- A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Plant Substances (AREA)
Abstract
Προσφέρεται ένα αναβράζον δισκίο για την παρασκευή ενός στοματικού διαλύματος, όπου το αναβράζον δισκίο εμφανίζει μεγάλο ρυθμό αποδέσμευσης της βουδεσονίδης. Έτσι επιτυγχάνεται μεγάλη διαθεσιμότητα της δραστικής ουσίας κατά τη χρήση ως στοματικού διαλύματος στον φλεγμένοντα βλεννογόνο του ανώτερου πεπτικού σωλήνα. Το πλεονέκτημα του σύμφωνου με την εφεύρεση σκευάσματος βρίσκεται στη συγκρίσιμη βιοδιαθεσιμότητα με τις από του στόματος μορφές χορήγησης, η οποία καθιστά δυνατή την ασφαλή χρήση για μεγάλο χρονικό διάστημα.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP08013091A EP2151235B1 (de) | 2008-07-21 | 2008-07-21 | Pharmazeutische Formulierung zur Behandlung des oberen Verdauungstraktes |
| EP09800023A EP2306988B1 (de) | 2008-07-21 | 2009-07-02 | Pharmazeutische formulierung zur behandlung des oberen verdauungstraktes |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CY1113719T1 true CY1113719T1 (el) | 2016-06-22 |
Family
ID=39951664
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CY20111100274T CY1111878T1 (el) | 2008-07-21 | 2011-03-11 | Φαρμακευτικο σκευασμα για τη θεραπεια του ανωτερoy πεπτικου σωληνα |
| CY20131100174T CY1113719T1 (el) | 2008-07-21 | 2013-02-26 | Φαρμακευτικο σκευασμα για τη θεραπεια του ανωτερου πεπτικου σωληνα |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CY20111100274T CY1111878T1 (el) | 2008-07-21 | 2011-03-11 | Φαρμακευτικο σκευασμα για τη θεραπεια του ανωτερoy πεπτικου σωληνα |
Country Status (23)
| Country | Link |
|---|---|
| US (2) | US8580300B2 (el) |
| EP (2) | EP2151235B1 (el) |
| JP (2) | JP5616889B2 (el) |
| CN (1) | CN102159196B (el) |
| AT (1) | ATE498396T1 (el) |
| AU (1) | AU2009273361B2 (el) |
| CA (1) | CA2731312C (el) |
| CY (2) | CY1111878T1 (el) |
| DE (1) | DE502008002621D1 (el) |
| DK (2) | DK2151235T3 (el) |
| EA (1) | EA018465B1 (el) |
| ES (2) | ES2358158T3 (el) |
| HR (2) | HRP20130171T1 (el) |
| IL (1) | IL210779A (el) |
| ME (2) | ME01256B (el) |
| NZ (1) | NZ590593A (el) |
| PL (2) | PL2151235T3 (el) |
| PT (2) | PT2151235E (el) |
| RS (2) | RS51649B (el) |
| SI (2) | SI2151235T1 (el) |
| UA (1) | UA100759C2 (el) |
| WO (1) | WO2010009961A1 (el) |
| ZA (1) | ZA201100283B (el) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8895064B2 (en) | 1999-06-14 | 2014-11-25 | Cosmo Technologies Limited | Controlled release and taste masking oral pharmaceutical composition |
| RU2246293C2 (ru) | 1999-06-14 | 2005-02-20 | Космо С.П.А. | Фармацевтические композиции для перорального введения с регулируемым высвобождением активного ингредиента и маскируемым вкусом |
| US8497258B2 (en) | 2005-11-12 | 2013-07-30 | The Regents Of The University Of California | Viscous budesonide for the treatment of inflammatory diseases of the gastrointestinal tract |
| SI2151235T1 (sl) * | 2008-07-21 | 2011-04-29 | Falk Pharma Gmbh | Farmacevtska formulacija za zdravljenje zgornjega prebavnega trakta |
| EP2440210A4 (en) | 2009-06-12 | 2014-01-29 | Meritage Pharma Inc | METHOD FOR THE TREATMENT OF STOMACH DARM DISEASES |
| EP3403654B1 (en) | 2009-10-01 | 2019-07-31 | Adare Development I, L.P. | Orally administered corticosteroid compositions |
| US10154964B2 (en) | 2011-09-07 | 2018-12-18 | Cosmo Technologies Limited | Controlled release and taste masking oral pharmaceutical composition |
| WO2015034678A2 (en) | 2013-09-06 | 2015-03-12 | Aptalis Pharmatech, Inc. | Corticosteroid containing orally disintegrating tablet compositions for eosinophilic esophagitis |
| SI2886108T2 (sl) * | 2013-12-23 | 2023-02-28 | Dr. Falk Pharma Gmbh | Optimizirana farmacevtska formulacija za zdravljenje vnetnih sprememb požiralnika |
| TWI777515B (zh) | 2016-08-18 | 2022-09-11 | 美商愛戴爾製藥股份有限公司 | 治療嗜伊紅性食道炎之方法 |
Family Cites Families (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE4332394A1 (de) | 1993-09-23 | 1995-03-30 | Falk Pharma Gmbh | Budesonid-Pellets mit kontrolliertem Freigabeprofil und Verfahren zu ihrer Herstellung |
| US5639475A (en) * | 1995-02-03 | 1997-06-17 | Eurand America, Incorporated | Effervescent microcapsules |
| US5607697A (en) * | 1995-06-07 | 1997-03-04 | Cima Labs, Incorporated | Taste masking microparticles for oral dosage forms |
| US5807577A (en) * | 1995-11-22 | 1998-09-15 | Lab Pharmaceutical Research International Inc. | Fast-melt tablet and method of making same |
| US5807578A (en) * | 1995-11-22 | 1998-09-15 | Lab Pharmaceutical Research International Inc. | Fast-melt tablet and method of making same |
| GB9611364D0 (en) * | 1996-05-31 | 1996-08-07 | Smithkline Beecham Plc | Composition |
| US6350470B1 (en) * | 1998-04-29 | 2002-02-26 | Cima Labs Inc. | Effervescent drug delivery system for oral administration |
| JP3818789B2 (ja) * | 1999-02-18 | 2006-09-06 | 三菱化学フーズ株式会社 | 易崩壊性錠剤 |
| WO2003006629A1 (en) | 2001-07-11 | 2003-01-23 | Toshirou Sekine | Culturing method and device for photosynthetic microbes |
| JP2005519865A (ja) * | 2001-09-25 | 2005-07-07 | ランバクシー ラボラトリーズ リミテッド | 急速溶解性投薬形態物の製造方法 |
| JP2005517636A (ja) * | 2001-11-20 | 2005-06-16 | ディーエムアイ バイオサイエンシズ インコーポレイテッド | オーラル・ケアのための方法および製品 |
| CA2479735C (en) * | 2002-03-20 | 2011-05-17 | Elan Pharma International Ltd. | Fast dissolving dosage forms having reduced friability |
| SE0401031D0 (sv) * | 2004-04-22 | 2004-04-22 | Duocort Ab | A new glucocorticoid replacement therapy |
| US20060013873A1 (en) * | 2004-07-16 | 2006-01-19 | Chih-Chiang Yang | Bioadhesive dosage form of steroids |
| US20070071817A1 (en) * | 2005-09-26 | 2007-03-29 | Phyzz, Inc. | Effervescent oral care compositions and method of use |
| WO2007095342A2 (en) * | 2006-02-15 | 2007-08-23 | Tika Läkemedel Ab | Stable corticosteroid mixtures |
| PL2170348T3 (pl) * | 2007-06-22 | 2017-01-31 | Dompé Farmaceutici S.P.A. | Tabletki musujące do zastosowania wziewnego |
| EP2572705B1 (en) * | 2007-10-01 | 2017-09-13 | Laboratorios Lesvi, S.L. | Orodispersible tablets |
| SI2151235T1 (sl) * | 2008-07-21 | 2011-04-29 | Falk Pharma Gmbh | Farmacevtska formulacija za zdravljenje zgornjega prebavnega trakta |
| EP2440210A4 (en) * | 2009-06-12 | 2014-01-29 | Meritage Pharma Inc | METHOD FOR THE TREATMENT OF STOMACH DARM DISEASES |
-
2008
- 2008-07-21 SI SI200830187T patent/SI2151235T1/sl unknown
- 2008-07-21 AT AT08013091T patent/ATE498396T1/de active
- 2008-07-21 DK DK08013091.7T patent/DK2151235T3/da active
- 2008-07-21 PL PL08013091T patent/PL2151235T3/pl unknown
- 2008-07-21 EP EP08013091A patent/EP2151235B1/de active Active
- 2008-07-21 RS RS20110100A patent/RS51649B/sr unknown
- 2008-07-21 ES ES08013091T patent/ES2358158T3/es active Active
- 2008-07-21 PT PT08013091T patent/PT2151235E/pt unknown
- 2008-07-21 ME MEP-2011-46A patent/ME01256B/me unknown
- 2008-07-21 DE DE502008002621T patent/DE502008002621D1/de active Active
-
2009
- 2009-02-07 UA UAA201101686A patent/UA100759C2/uk unknown
- 2009-07-02 EP EP09800023A patent/EP2306988B1/de not_active Revoked
- 2009-07-02 SI SI200930502T patent/SI2306988T1/sl unknown
- 2009-07-02 WO PCT/EP2009/058320 patent/WO2010009961A1/de not_active Ceased
- 2009-07-02 AU AU2009273361A patent/AU2009273361B2/en not_active Ceased
- 2009-07-02 PT PT98000235T patent/PT2306988E/pt unknown
- 2009-07-02 NZ NZ590593A patent/NZ590593A/en unknown
- 2009-07-02 HR HRP20130171AT patent/HRP20130171T1/hr unknown
- 2009-07-02 EA EA201100229A patent/EA018465B1/ru not_active IP Right Cessation
- 2009-07-02 RS RS20130071A patent/RS52662B/sr unknown
- 2009-07-02 ES ES09800023T patent/ES2399321T3/es active Active
- 2009-07-02 ME MEP-2013-22A patent/ME01494B/me unknown
- 2009-07-02 DK DK09800023.5T patent/DK2306988T3/da active
- 2009-07-02 US US13/054,844 patent/US8580300B2/en not_active Expired - Fee Related
- 2009-07-02 CN CN2009801358800A patent/CN102159196B/zh not_active Expired - Fee Related
- 2009-07-02 CA CA2731312A patent/CA2731312C/en not_active Expired - Fee Related
- 2009-07-02 JP JP2011519101A patent/JP5616889B2/ja not_active Expired - Fee Related
- 2009-07-02 PL PL09800023T patent/PL2306988T3/pl unknown
-
2011
- 2011-01-11 ZA ZA2011/00283A patent/ZA201100283B/en unknown
- 2011-01-20 IL IL210779A patent/IL210779A/en active IP Right Grant
- 2011-03-11 CY CY20111100274T patent/CY1111878T1/el unknown
- 2011-03-23 HR HR20110208T patent/HRP20110208T1/hr unknown
-
2013
- 2013-02-26 CY CY20131100174T patent/CY1113719T1/el unknown
- 2013-10-23 US US14/061,578 patent/US20140079646A1/en not_active Abandoned
-
2014
- 2014-07-30 JP JP2014155149A patent/JP6209495B2/ja not_active Expired - Fee Related
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