CY1107711T1 - Υπογλωσσια χορηγηση φαρμακευτικης συνθεσης ως αγωγη εναντι οξεων διαταραχων - Google Patents
Υπογλωσσια χορηγηση φαρμακευτικης συνθεσης ως αγωγη εναντι οξεων διαταραχωνInfo
- Publication number
- CY1107711T1 CY1107711T1 CY20071101054T CY071101054T CY1107711T1 CY 1107711 T1 CY1107711 T1 CY 1107711T1 CY 20071101054 T CY20071101054 T CY 20071101054T CY 071101054 T CY071101054 T CY 071101054T CY 1107711 T1 CY1107711 T1 CY 1107711T1
- Authority
- CY
- Cyprus
- Prior art keywords
- pharmaceutical composition
- particles
- treatment against
- composition
- against acid
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 239000002253 acid Substances 0.000 title 1
- 239000000203 mixture Substances 0.000 abstract 4
- 239000002245 particle Substances 0.000 abstract 4
- 239000013543 active substance Substances 0.000 abstract 2
- 230000001154 acute effect Effects 0.000 abstract 2
- 239000003795 chemical substances by application Substances 0.000 abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 208000035475 disorder Diseases 0.000 abstract 2
- 238000000034 method Methods 0.000 abstract 1
- 210000004877 mucosa Anatomy 0.000 abstract 1
- 230000001737 promoting effect Effects 0.000 abstract 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 abstract 1
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/136—Amines having aromatic rings, e.g. ketamine, nortriptyline having the amino group directly attached to the aromatic ring, e.g. benzeneamine
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- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
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- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/196—Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
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Abstract
Περιγράφεται φαρμακευτική σύνθεση προς αγωγή έναντι οξέων διαταραχών. Η σύνθεση περιλαμβάνει ουσιωδώς ελεύθερο ύδατος, διατεταγμένο μείγμα τουλάχιστον ενός φαρμακευτικώς δραστικού παράγοντα υπό τη μορφή μικροσκοπικών σωματιδίων τα οποία προσκολλώνται στις επιφάνειες σωματιδιών ενός φορέα τα οποία σωματίδια του φορέα είναι ουσιωδώς πιο ευμεγέθη από τα σωματίδια του δραστικού παράγοντα ή των δραστικών παραγόντων, και τα οποία είναι ουσιωδώς υδατοδυαλυτά, σε συνδυασμό με παράγοντα προαγωγής της προσκόλλησης σε βιολογικές επιφάνειες και/ή σε βλεννογόνο. Η εφεύρεση επίσης σχετίζεται με μέθοδο παρασκευής της σύνθεσης και με τη χρήση της σύνθεσης προς αγωγή έναντι οξέων διαταραχών.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE9803240A SE9803240D0 (sv) | 1998-09-24 | 1998-09-24 | A pharmaceutical composition having a rapid action |
| EP99952867A EP1115383B1 (en) | 1998-09-24 | 1999-09-24 | Treatment of acute disorders by sublingual administration of a pharmaceutical composition |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CY1107711T1 true CY1107711T1 (el) | 2013-04-18 |
Family
ID=20412702
Family Applications (5)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
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| CY20131100974T CY1114620T1 (el) | 1998-09-24 | 2013-11-04 | Φαρμακευτικη συνθεση προς υπογλωσσια χορηγηση |
| CY20141100588T CY1115685T1 (el) | 1998-09-24 | 2014-08-04 | Φαρμακευτικη συνθεση προς αγωγη εναντι αϋπνιας μεσω υπογλωσσιας χορηγησης |
| CY20141100730T CY1115688T1 (el) | 1998-09-24 | 2014-09-10 | Φαρμακευτικη συνθεση που περιλαμβανει φεντανυλη προς αγωγη εναντι οξεος ή παροξυσμικου πονου μεσω υπογλωσσιας χορηγησης |
| CY20171101261T CY1119644T1 (el) | 1998-09-24 | 2017-11-30 | Φαρμακευτικη συνθεση ταχειας δρασης που περιλαμβανει βουπρενορφινη |
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| CY20141100588T CY1115685T1 (el) | 1998-09-24 | 2014-08-04 | Φαρμακευτικη συνθεση προς αγωγη εναντι αϋπνιας μεσω υπογλωσσιας χορηγησης |
| CY20141100730T CY1115688T1 (el) | 1998-09-24 | 2014-09-10 | Φαρμακευτικη συνθεση που περιλαμβανει φεντανυλη προς αγωγη εναντι οξεος ή παροξυσμικου πονου μεσω υπογλωσσιας χορηγησης |
| CY20171101261T CY1119644T1 (el) | 1998-09-24 | 2017-11-30 | Φαρμακευτικη συνθεση ταχειας δρασης που περιλαμβανει βουπρενορφινη |
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| AU (1) | AU764346B2 (el) |
| BG (1) | BG65502B1 (el) |
| BR (1) | BRPI9913945B8 (el) |
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| IL (1) | IL142135A0 (el) |
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| NO (1) | NO332226B1 (el) |
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| FR2758459B1 (fr) * | 1997-01-17 | 1999-05-07 | Pharma Pass | Composition pharmaceutique de fenofibrate presentant une biodisponibilite elevee et son procede de preparation |
| US5968547A (en) * | 1997-02-24 | 1999-10-19 | Euro-Celtique, S.A. | Method of providing sustained analgesia with buprenorphine |
| DE19749724A1 (de) * | 1997-11-11 | 1999-06-10 | Gruenenthal Gmbh | Verwendung einer Kombination aus Opioid und alpha-adrenergem Agonisten in Schmerzmitteln |
| KR100289471B1 (ko) * | 1998-01-19 | 2001-09-17 | 김충섭 | 휀타닐계마취제의이식형서방성제제 |
| US6974590B2 (en) * | 1998-03-27 | 2005-12-13 | Cima Labs Inc. | Sublingual buccal effervescent |
| US6264974B1 (en) * | 1998-07-07 | 2001-07-24 | Salvagnini Italia Spa | Buccal and sublingual administration of physostigmine |
| SE9803239D0 (sv) * | 1998-09-24 | 1998-09-24 | Diabact Ab | Composition for the treatment of acute pain |
| SE9803240D0 (sv) | 1998-09-24 | 1998-09-24 | Diabact Ab | A pharmaceutical composition having a rapid action |
| EP1005863A1 (en) | 1998-12-04 | 2000-06-07 | Synthelabo | Controlled-release dosage forms comprising a short acting hypnotic or a salt thereof |
| WO2001030391A2 (en) | 1999-10-27 | 2001-05-03 | Farmarc Nederland Bv | Pharmaceutical composition containing midazolam |
| EP1272181A2 (en) * | 2000-04-13 | 2003-01-08 | Synthon B.V. | Modified release formulations containing a hypnotic agent |
| CN1290525A (zh) | 2000-10-10 | 2001-04-11 | 北京万全阳光医药科技有限公司 | 冷冻干燥的扎来普隆速溶口服组合物 |
| US20030035839A1 (en) | 2001-05-15 | 2003-02-20 | Peirce Management, Llc | Pharmaceutical composition for both intraoral and oral administration |
| ATE389402T1 (de) | 2002-01-10 | 2008-04-15 | Biovail Lab Int Srl | Sedierende nicht-benzodiazepin-formulierungen |
| CN1418631A (zh) | 2002-12-19 | 2003-05-21 | 王登之 | 治疗失眠的佐匹克隆口腔崩解片及其制备方法 |
| US20040265375A1 (en) | 2003-04-16 | 2004-12-30 | Platteeuw Johannes J. | Orally disintegrating tablets |
-
1998
- 1998-09-24 SE SE9803240A patent/SE9803240D0/xx unknown
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1999
- 1999-09-24 EP EP99952867A patent/EP1115383B1/en not_active Expired - Lifetime
- 1999-09-24 US US09/787,888 patent/US6761910B1/en not_active Expired - Lifetime
- 1999-09-24 CN CNB998135453A patent/CN1173694C/zh not_active Expired - Lifetime
- 1999-09-24 EP EP10001408.3A patent/EP2236133B1/en not_active Expired - Lifetime
- 1999-09-24 HU HU0103856A patent/HU230342B1/hu unknown
- 1999-09-24 EP EP10001406.7A patent/EP2236132B1/en not_active Expired - Lifetime
- 1999-09-24 KR KR1020017003715A patent/KR100760536B1/ko not_active Expired - Lifetime
- 1999-09-24 AT AT99952867T patent/ATE365540T1/de active
- 1999-09-24 TR TR2001/00855T patent/TR200100855T2/xx unknown
- 1999-09-24 CA CA2820588A patent/CA2820588C/en not_active Expired - Lifetime
- 1999-09-24 NZ NZ510284A patent/NZ510284A/en not_active IP Right Cessation
- 1999-09-24 BR BRPI9913945A patent/BRPI9913945B8/pt not_active IP Right Cessation
- 1999-09-24 EP EP05077875.2A patent/EP1652518B1/en not_active Expired - Lifetime
- 1999-09-24 DK DK14175085.1T patent/DK2805716T3/en active
- 1999-09-24 IL IL14213599A patent/IL142135A0/xx not_active IP Right Cessation
- 1999-09-24 MX MXPA01003068A patent/MXPA01003068A/es active IP Right Grant
- 1999-09-24 SK SK402-2001A patent/SK283302B6/sk not_active IP Right Cessation
- 1999-09-24 PT PT100014083T patent/PT2236133E/pt unknown
- 1999-09-24 ES ES10001408.3T patent/ES2498095T3/es not_active Expired - Lifetime
- 1999-09-24 CZ CZ20011029A patent/CZ302975B6/cs not_active IP Right Cessation
- 1999-09-24 PT PT141750851T patent/PT2805716T/pt unknown
- 1999-09-24 EE EEP200800028A patent/EE05555B1/xx unknown
- 1999-09-24 EP EP14175085.1A patent/EP2805716B1/en not_active Revoked
- 1999-09-24 RU RU2001111025/14A patent/RU2193879C1/ru active
- 1999-09-24 DK DK10001406.7T patent/DK2236132T3/da active
- 1999-09-24 CA CA002345121A patent/CA2345121C/en not_active Expired - Lifetime
- 1999-09-24 PL PL383971A patent/PL204264B1/pl unknown
- 1999-09-24 ES ES14175085.1T patent/ES2644770T3/es not_active Expired - Lifetime
- 1999-09-24 ES ES10001406.7T patent/ES2507579T3/es not_active Expired - Lifetime
- 1999-09-24 ES ES05077875T patent/ES2433930T3/es not_active Expired - Lifetime
- 1999-09-24 PT PT99952867T patent/PT1115383E/pt unknown
- 1999-09-24 PL PL347126A patent/PL201644B1/pl unknown
- 1999-09-24 DE DE69936393T patent/DE69936393T2/de not_active Expired - Lifetime
- 1999-09-24 EE EEP200700030A patent/EE05023B1/xx unknown
- 1999-09-24 HU HU0800435A patent/HU230468B1/hu unknown
- 1999-09-24 CZ CZ2008-315A patent/CZ2008315A3/cs not_active IP Right Cessation
- 1999-09-24 WO PCT/SE1999/001687 patent/WO2000016750A1/en not_active Ceased
- 1999-09-24 DK DK10001408.3T patent/DK2236133T3/da active
- 1999-09-24 EE EEP200100182A patent/EE04927B1/xx unknown
- 1999-09-24 PT PT100014067T patent/PT2236132E/pt unknown
- 1999-09-24 PT PT50778752T patent/PT1652518E/pt unknown
- 1999-09-24 DK DK99952867T patent/DK1115383T3/da active
- 1999-09-24 DK DK05077875.2T patent/DK1652518T3/da active
- 1999-09-24 ES ES99952867T patent/ES2289829T3/es not_active Expired - Lifetime
- 1999-09-24 CA CA2629988A patent/CA2629988C/en not_active Expired - Lifetime
- 1999-09-24 JP JP2000573711A patent/JP3381220B2/ja not_active Expired - Lifetime
- 1999-09-24 AU AU64927/99A patent/AU764346B2/en not_active Expired
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2001
- 2001-03-22 NO NO20011473A patent/NO332226B1/no not_active IP Right Cessation
- 2001-03-23 BG BG105379A patent/BG65502B1/bg unknown
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2004
- 2004-05-24 US US10/851,215 patent/US20040213855A1/en not_active Abandoned
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2006
- 2006-10-10 US US11/544,660 patent/US7910132B2/en not_active Expired - Fee Related
-
2007
- 2007-08-07 CY CY20071101054T patent/CY1107711T1/el unknown
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2008
- 2008-07-01 US US12/216,197 patent/US20080286368A1/en not_active Abandoned
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2011
- 2011-11-22 US US13/302,720 patent/US8512747B2/en not_active Expired - Fee Related
- 2011-11-22 US US13/302,694 patent/US8454996B2/en not_active Expired - Fee Related
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2013
- 2013-03-13 US US13/799,640 patent/US20130195976A1/en not_active Abandoned
- 2013-07-30 US US13/954,141 patent/US20140030336A1/en not_active Abandoned
- 2013-11-04 CY CY20131100974T patent/CY1114620T1/el unknown
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2014
- 2014-08-04 CY CY20141100588T patent/CY1115685T1/el unknown
- 2014-09-10 CY CY20141100730T patent/CY1115688T1/el unknown
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2015
- 2015-01-20 LU LU92636C patent/LU92636I2/xx unknown
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2017
- 2017-11-30 CY CY20171101261T patent/CY1119644T1/el unknown
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