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CU24087B1 - Compuestos de carbazol - Google Patents

Compuestos de carbazol

Info

Publication number
CU24087B1
CU24087B1 CU2011000078A CU20110078A CU24087B1 CU 24087 B1 CU24087 B1 CU 24087B1 CU 2011000078 A CU2011000078 A CU 2011000078A CU 20110078 A CU20110078 A CU 20110078A CU 24087 B1 CU24087 B1 CU 24087B1
Authority
CU
Cuba
Prior art keywords
compounds
diseases
carbazol
conditions
carbazol compounds
Prior art date
Application number
CU2011000078A
Other languages
English (en)
Other versions
CU20110078A7 (es
Inventor
John Tucker
Sergey Sviridov
Leonid Brodsky
Catherine Burkhart
Andrei Purmal
Katerina Gurova
Andrei Gudkov
Original Assignee
Incuron
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Incuron filed Critical Incuron
Publication of CU20110078A7 publication Critical patent/CU20110078A7/es
Publication of CU24087B1 publication Critical patent/CU24087B1/es

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    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
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    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
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    • C07D209/82Carbazoles; Hydrogenated carbazoles
    • C07D209/86Carbazoles; Hydrogenated carbazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the ring system
    • CCHEMISTRY; METALLURGY
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    • C07D209/82Carbazoles; Hydrogenated carbazoles
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
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    • C07ORGANIC CHEMISTRY
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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
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  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Pharmacology & Pharmacy (AREA)
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  • General Engineering & Computer Science (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Oncology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Mechanical Engineering (AREA)
  • Nursing (AREA)
  • Wood Science & Technology (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Immunology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Se exponen compuestos de la fórmula estructural general (I) y (II) ESPACIO PARA LAS FÓRMULAS como agentes terapéuticos. Las enfermedades y condiciones tratables incluyen cánceres, enfermedades y condiciones inflamatorias y enfermedades de inmunodeficiencia.
CU2011000078A 2008-10-06 2009-10-05 Compuestos de carbazol CU24087B1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10291308P 2008-10-06 2008-10-06
PCT/US2009/059558 WO2010042445A1 (en) 2008-10-06 2009-10-05 Carbazole compounds and therapeutic uses of the compounds

Publications (2)

Publication Number Publication Date
CU20110078A7 CU20110078A7 (es) 2012-01-31
CU24087B1 true CU24087B1 (es) 2015-03-30

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CU2011000078A CU24087B1 (es) 2008-10-06 2009-10-05 Compuestos de carbazol

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US (5) US8765738B2 (es)
EP (1) EP2356093B1 (es)
JP (1) JP5694172B2 (es)
KR (1) KR101586112B1 (es)
CN (1) CN102203063B (es)
AP (1) AP2860A (es)
AU (1) AU2009302546B2 (es)
BR (1) BRPI0920876A2 (es)
CA (1) CA2736097C (es)
CU (1) CU24087B1 (es)
CY (1) CY1113924T1 (es)
DK (1) DK2356093T3 (es)
ES (1) ES2402395T3 (es)
GE (1) GEP20146131B (es)
HR (1) HRP20130313T1 (es)
IL (1) IL211430A0 (es)
MX (1) MX2011003416A (es)
NZ (1) NZ591516A (es)
PL (1) PL2356093T3 (es)
PT (1) PT2356093E (es)
RS (1) RS52702B (es)
RU (1) RU2497807C2 (es)
SI (1) SI2356093T1 (es)
SM (1) SMT201300042B (es)
UA (1) UA107652C2 (es)
WO (1) WO2010042445A1 (es)
ZA (1) ZA201101513B (es)

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Publication number Priority date Publication date Assignee Title
UA107652C2 (en) * 2008-10-06 2015-02-10 Incuron Llc Carbazole compounds and therapeutic uses of the compounds
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