BR9909487A - Herbicidas de n-piridonila - Google Patents
Herbicidas de n-piridonilaInfo
- Publication number
- BR9909487A BR9909487A BR9909487-8A BR9909487A BR9909487A BR 9909487 A BR9909487 A BR 9909487A BR 9909487 A BR9909487 A BR 9909487A BR 9909487 A BR9909487 A BR 9909487A
- Authority
- BR
- Brazil
- Prior art keywords
- alkyl
- haloalkyl
- alkoxy
- phenyl
- halogen
- Prior art date
Links
- 239000004009 herbicide Substances 0.000 title abstract 3
- 125000000217 alkyl group Chemical group 0.000 abstract 31
- 125000001188 haloalkyl group Chemical group 0.000 abstract 16
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 11
- 229910052736 halogen Inorganic materials 0.000 abstract 9
- 150000002367 halogens Chemical class 0.000 abstract 9
- 125000003342 alkenyl group Chemical group 0.000 abstract 6
- 125000000304 alkynyl group Chemical group 0.000 abstract 6
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 6
- 229910052739 hydrogen Inorganic materials 0.000 abstract 6
- 239000001257 hydrogen Substances 0.000 abstract 6
- 150000002431 hydrogen Chemical class 0.000 abstract 6
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 5
- 125000000262 haloalkenyl group Chemical group 0.000 abstract 5
- 125000003545 alkoxy group Chemical group 0.000 abstract 4
- 125000004448 alkyl carbonyl group Chemical group 0.000 abstract 4
- -1 nitro, amino Chemical group 0.000 abstract 4
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 3
- 125000001584 benzyloxycarbonyl group Chemical group C(=O)(OCC1=CC=CC=C1)* 0.000 abstract 3
- 125000004692 haloalkylcarbonyl group Chemical group 0.000 abstract 3
- 125000002768 hydroxyalkyl group Chemical group 0.000 abstract 3
- UYWQUFXKFGHYNT-UHFFFAOYSA-N phenylmethyl ester of formic acid Natural products O=COCC1=CC=CC=C1 UYWQUFXKFGHYNT-UHFFFAOYSA-N 0.000 abstract 3
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 2
- 125000005092 alkenyloxycarbonyl group Chemical group 0.000 abstract 2
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 2
- 229910052760 oxygen Inorganic materials 0.000 abstract 2
- 239000001301 oxygen Substances 0.000 abstract 2
- 229910052717 sulfur Inorganic materials 0.000 abstract 2
- 239000011593 sulfur Substances 0.000 abstract 2
- WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical compound [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 abstract 1
- ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical compound [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 abstract 1
- PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical compound FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 abstract 1
- 125000005090 alkenylcarbonyl group Chemical group 0.000 abstract 1
- 125000003302 alkenyloxy group Chemical group 0.000 abstract 1
- 125000005108 alkenylthio group Chemical group 0.000 abstract 1
- 125000005196 alkyl carbonyloxy group Chemical group 0.000 abstract 1
- 125000004414 alkyl thio group Chemical group 0.000 abstract 1
- 125000005133 alkynyloxy group Chemical group 0.000 abstract 1
- 125000005225 alkynyloxycarbonyl group Chemical group 0.000 abstract 1
- 125000005109 alkynylthio group Chemical group 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- 125000000051 benzyloxy group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])O* 0.000 abstract 1
- GDTBXPJZTBHREO-UHFFFAOYSA-N bromine Substances BrBr GDTBXPJZTBHREO-UHFFFAOYSA-N 0.000 abstract 1
- 229910052794 bromium Inorganic materials 0.000 abstract 1
- 229910052801 chlorine Inorganic materials 0.000 abstract 1
- 239000000460 chlorine Substances 0.000 abstract 1
- 229910052731 fluorine Inorganic materials 0.000 abstract 1
- 239000011737 fluorine Substances 0.000 abstract 1
- 125000005291 haloalkenyloxy group Chemical group 0.000 abstract 1
- 125000004438 haloalkoxy group Chemical group 0.000 abstract 1
- 125000004993 haloalkoxycarbonyl group Chemical group 0.000 abstract 1
- 125000005347 halocycloalkyl group Chemical group 0.000 abstract 1
- 125000001072 heteroaryl group Chemical group 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
- 125000003373 pyrazinyl group Chemical group 0.000 abstract 1
- 125000002098 pyridazinyl group Chemical group 0.000 abstract 1
- 125000004076 pyridyl group Chemical group 0.000 abstract 1
- 125000000714 pyrimidinyl group Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000005389 trialkylsiloxy group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
- A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/58—1,2-Diazines; Hydrogenated 1,2-diazines
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
- A01N43/647—Triazoles; Hydrogenated triazoles
- A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
Patente de Invenção: <B>"HERBICIDAS DE N-PIRIDONILA"<D>. Os compostos de fórmula I na qual R~ 1~ é hidrogênio, flúor, cloro, bromo ou metila; R~ 2~ é C~ 1~-C~ 4~alquila, C~ 1~-C~ 4~haloalquila, halogênio, nitro, amino, ciano ou R~ 43~O-; R~ 43~ é hidrogênio, C~ 1~-C~ 8~alquila, C~ 3~-C~ 8~alquenila, C~ 3~-C~ 8~alquinila, C~ 3~-C~ 6~cicloalquila, C~ 1~-C~ 8~haloalquila, ciano-C~ 1~-C~ 8~alquila, C~ 3~-C~ 8~haloalquenila, hidróxi-C~ 1~-C~ 4~alquila, C~ 1~-C~ 4~alcóxi-C~ 1~-C~ 4~alquila, C~ 3~-C~ 6~alquenilóxi-C~ 1~-C~ 4~-alquila, C~ 3~-C~ 6~alquinilóxi-C~ 1~-C~ 4~alquila, C~ 1~-C~ 4~alcóxi-C~ 1~-C~ 4~alcóxi-C~ 1~-C~ 4~alquila, C~ 1~-C~ 4~-alquiltio-C~ 1~-C~ 4~alquila, C~ 1~-C~ 8~alquilcarbonila, C~ 1~-C~ 8~alcoxicarbonila, C~ 3~-C~ 8~alqueniloxicarbonila, benzilóxi-C~ 1~- ou -C~ 2~-alquila, benzilcarbonila, benziloxicarbonila, fenila, fenil-C~ 2~-C~ 8~alquila, benzila, piridila, pirimidinila, pirazinila ou piridazinila, aqueles anéis aromáticos e heteroaromáticos sendo insubstituídos ou mono- a tri-substituídos por halogênio, C~ 1~-C~ 4~alquila ou por C~ 1~-C~ 4~haloalquila; ou R~ 43~ é R~ 44~X~ 16~C(O)-C~ 1~-C~ 8~alquil- ou X~ 16~ é oxigênio, enxofre ou R~ 44~ é hidrogênio, C~ 1~-C~ 8~alquila, C~ 3~-C~ 8~alquenila, C~ 3~-C~ 8~alquinila, C~ 3~-C~ 6~cicloalquila, C~ 1~-C~ 8~haloalquila, C~ 3~-C~ 8~haloalquenila, C~ 1~-C~ 4~alcoxi-C~ 1~-C~ 4~alquila, C~ 3~-C~ 6~alqueniloxi-C~ 1~-C~ 4~alquila, C~ 1~-C~ 4~alquiltio-C~ 1~-C~ 4~alquila, fenila, fenila mono- a tri-substituída por halogênio, C~ 1~-C~ 4~alquila ou por C~ 1~-C~ 4~haloalquila, benzila ou benzila mono- a tri-substituída no anel de fenila por halogênio, C~ 1~-C~ 4~alquila ou por C~ 1~-C~ 4~haloalquila; R~ 45~ é hidrogênio, C~ 1~-C~ 8~alquila, C~ 3~-C~ 8~alquenila, C~ 3~-C~ 8~alquinila, C~ 3~-C~ 6~cicloalquila, C~ 1~-C~ 8~haloalquila ou benzila; R~ 3~ é hidróxi, C~ 1~-C~ 6~alcóxi, C~ 3~-C~ 6~alquenilóxi, C~ 3~-C~ 6~alquinilóxi, C~ 1~-C~ 6~haloalcóxi, C~ 3~-C~ 6~haloalquenilóxi, C~ 1~-C~ 6~alcóxi-C~ 1~-C~ 6~alquila, C~ 3~-C~ 6~alquenilóxi-C~ 1~-C~ 6~alquila, C~ 3~-C~ 6~alquiniloxi-C~ 1~-C~ 6~alquila, C~ 1~-C~ 6~alcoxi-C~ 1~-C~ 6~alcoxi-C~ 1~-C~ 6~alquila, B~ 1~-C~ 1~-C~ 6~alcóxi, R~ 4~(R~ 5~)N-, C~ 1~-C~ 6~alquila, C~ 3~-C~ 6~alquenila, C~ 3~-C~ 6~alquinila, C~ 2~-C~ 6~haloalquila, C~ 3~-C~ 6~háloalquenila, C~ 3~-C~ 6~cicloalquila, C~ 3~-C~ 6~halocicloalquila, B~ 1~-C~ 1~-C~ 6~alquila, OHC-, C~ 1~-C~ 6~alquilcarbonila, C~ 1~-C~ 6~alquilcarbonilóxi, C~ 1~-C~ 6~haloalquilcarbonila, C~ 2~-C~ 6~alquenilcarbonila, C~ 1~-C~ 6~alcoxicarbonila, C~ 1~-C~ 6~alquil-S(O)~ 2~-, C~ 1~-C~ 6~haloalquil-S(O)~ 2~-, C~ 3~-C~ 8~trialquilsililóxi, (C~ 1~-C~ 6~alquil)~ 2~N-N=CH-, B~ 1~CH=N-, (CH~ 3~)~ 2~N-CH=N-, (C~ 1~-C~ 5~hidroxialquil)-CH~ 2~-, (B~ 1~-C~ 1~-C~ 5~hidroxialquil)-CH~ 2~-, (B-C~ 1~-C~ 5~haloalquil)-CH~ 2~-, (Hidróxi-C~ 1~-C~ 5~alquil)-O- ou (B~ 1~-C~ 1~-C~ 5~hidroxialquil)-O-; B~ 1~ é ciano, OHC-, HOC(O)-, C~ 1~-C~ 6~alquilcarbonila, C~ 1~-C~ 6~haloalquilcarbonila, C~ 1~-C~ 6~alcoxicarbonila, C~ 3~-C~ 6~alqueniloxicarbonila, C~ 3~-C~ 6~alquiniloxicarbonila, benzilóxi, benziloxicarbonila, benziloxicarbonila mono- a tri-substituída no anel de fenila por halogênio, C~ 1~-C~ 4~alquila ou por C~ 1~-C~ 4~haloalquila, benziltio, benziltiocarbonila, benziltiocarbonila mono- a tri-substituída no anel de fenila por halogênio, C~ 1~-C~ 4~alquila ou por C~ 1~-C~ 4~haloalquila, C~ 1~-C~ 6~haloalcoxicarbonila, C~ 1~-C~ 6~alquiltio-C(O)-, R~ 6~(R~ 7~)NC(O)-, fenila, fenila mono- a tri-substituída por halogênio, C~ 1~-C~ 4~alquila ou por C~ 1~-C~ 4~haloalquila, C~ 1~-C~ 6~alquil-S(O)~ 2~-, C~ 1~-C~ 6~alquil-S(O)-, C~ 1~-C~ 6~alquiltio-, C~ 3~-C~ 6~cicloalquila, C~ 1~-C~ 6~alcóxi, C~ 3~-C~ 6~alqueniltio ou C~ 3~C~ 6~alquiniltio; R~ 4~ e R~ 5~ são, cada um independentemente do outro, hidrogênio, C~ 1~-C~ 6~alquila, C~ 3~-C~ 6~alquenila, C~ 3~-C~ 6~alquinila, C~ 1~-C~ 6~haloalquila, C~ 3~-C~ 6~haloalquenila, C~ 3~-C~ 6~-cicloalquila, C~ 1~-C~ 6~alcóxi-C~ 1~-C~ 6~alquila, OHC-, C~ 1~-C~ 6~alquilcarbonila, C~ 1~-C~ 6~haloalquilcarbonila, C~ 1~-C~ 6~alquil-S(O)~ 2~- ou C~ 1~-C~ 6~haloalquil-S(O)~ 2~-; R~ 6~ e R~ 7~ são, cada um independentemente do outro, hidrogênio, C~ 1~-C~ 6~alquila, C~ 3~-C~ 6~alquenila, C~ 3~-C~ 6~alquinila, C~ 1~-C~ 6~haloalquila, C~ 3~-C~ 6~haloalquenila, fenila, fenila mono- a tri-substituída por halogênio, C~ 1~-C~ 4~-alquila ou por C~ 1~-C~ 4~haloalquila, benzila ou benzila mono- a tri-substituída no anel de fenila por halogênio, C~ 1~-C~ 4~alquila ou por C~ 1~-C~ 4~haloalquila; X~ 1~ é oxigênio ou enxofre; W é um grupo e R~ 8~ a R~ 32~ e X~ 2~ a X~ 15~ são como definidos na reivindicação 1, e os sais e os estereoisómeros agroquimicamente aceitáveis de tais compostos de fórmula I, são adequados para uso como herbicidas.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH84098 | 1998-04-08 | ||
| PCT/EP1999/002313 WO1999052893A1 (en) | 1998-04-08 | 1999-04-06 | N-pyridonyl herbicides |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR9909487A true BR9909487A (pt) | 2000-12-12 |
Family
ID=4196437
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR9909487-8A BR9909487A (pt) | 1998-04-08 | 1999-04-06 | Herbicidas de n-piridonila |
Country Status (8)
| Country | Link |
|---|---|
| EP (1) | EP1076655A1 (pt) |
| JP (1) | JP2002511461A (pt) |
| KR (1) | KR20010042521A (pt) |
| CN (1) | CN1295570A (pt) |
| AU (1) | AU738222B2 (pt) |
| BR (1) | BR9909487A (pt) |
| ID (1) | ID27165A (pt) |
| WO (1) | WO1999052893A1 (pt) |
Families Citing this family (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2002351412B2 (en) | 2001-12-21 | 2010-05-20 | Exelixis Patent Company Llc | Modulators of LXR |
| US7482366B2 (en) | 2001-12-21 | 2009-01-27 | X-Ceptor Therapeutics, Inc. | Modulators of LXR |
| PT1490064E (pt) | 2002-02-14 | 2009-12-28 | Pharmacia Corp | Piridinonas substituídas como moduladores de p38 map-quinase |
| KR100574350B1 (ko) * | 2004-08-31 | 2006-04-27 | 한국화학연구원 | 2-아미노피리딘 유도체의 제조방법 |
| EP1942898B2 (en) | 2005-09-14 | 2014-05-14 | Takeda Pharmaceutical Company Limited | Dipeptidyl peptidase inhibitors for treating diabetes |
| AR059898A1 (es) | 2006-03-15 | 2008-05-07 | Janssen Pharmaceutica Nv | Derivados de 3-ciano-piridona 1,4-disustituida y su uso como moduladores alostericos de los receptores mglur2 |
| TW200900065A (en) | 2007-03-07 | 2009-01-01 | Janssen Pharmaceutica Nv | 3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives |
| TW200845978A (en) | 2007-03-07 | 2008-12-01 | Janssen Pharmaceutica Nv | 3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives |
| HRP20110278T1 (hr) | 2007-09-14 | 2011-05-31 | Ortho-Mcneil-Janssen Pharmaceuticals | 1',3'-disupstituirani-4-fenil,3,4,5,6-tetrahidro-2h,1'h[1,4']bipiridinil-2'-oni |
| JP5547194B2 (ja) | 2008-09-02 | 2014-07-09 | ジャンセン ファーマシューティカルズ, インコーポレイテッド. | 代謝型グルタミン酸受容体の調節因子としての3−アザビシクロ[3.1.0]ヘキシル誘導体 |
| CN102232074B (zh) | 2008-11-28 | 2014-12-03 | 奥梅-杨森制药有限公司 | 作为代谢性谷氨酸盐受体调节剂的吲哚和苯并噁嗪衍生物 |
| CN102439008B (zh) | 2009-05-12 | 2015-04-29 | 杨森制药有限公司 | 1,2,4-三唑并[4,3-a]吡啶衍生物及其用于治疗或预防神经和精神病症的用途 |
| MY153913A (en) | 2009-05-12 | 2015-04-15 | Janssen Pharmaceuticals Inc | 7-aryl-1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors |
| CA2760259C (en) | 2009-05-12 | 2018-05-01 | Janssen Pharmaceuticals, Inc. | 1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors |
| CA2815002C (en) | 2010-11-08 | 2019-10-22 | Janssen Pharmaceuticals, Inc. | 1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors |
| CA2814996C (en) | 2010-11-08 | 2019-10-01 | Janssen Pharmaceuticals, Inc. | 1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors |
| CN103261195B (zh) | 2010-11-08 | 2015-09-02 | 杨森制药公司 | 1,2,4-三唑并[4,3-a]吡啶衍生物及其作为MGLUR2受体的正变构调节剂的用途 |
| IN2014DN11218A (pt) * | 2012-06-30 | 2015-10-02 | Dow Agrosciences Llc | |
| JO3368B1 (ar) | 2013-06-04 | 2019-03-13 | Janssen Pharmaceutica Nv | مركبات 6، 7- ثاني هيدرو بيرازولو [5،1-a] بيرازين- 4 (5 يد)- اون واستخدامها بصفة منظمات تفارغية سلبية لمستقبلات ميجلور 2 |
| JO3367B1 (ar) | 2013-09-06 | 2019-03-13 | Janssen Pharmaceutica Nv | مركبات 2،1، 4- ثلاثي زولو [3،4-a] بيريدين واستخدامها بصفة منظمات تفارغية موجبة لمستقبلات ميجلور 2 |
| KR20200036063A (ko) | 2014-01-21 | 2020-04-06 | 얀센 파마슈티카 엔.브이. | 대사 조절형 글루탐산 작동성 수용체 제2아형의 양성 알로스테릭 조절제 또는 오르토스테릭 작동제를 포함하는 조합 및 그 용도 |
| EP3096790B1 (en) | 2014-01-21 | 2019-07-10 | Janssen Pharmaceutica, N.V. | Combinations comprising positive allosteric modulators or orthosteric agonists of metabotropic glutamatergic receptor subtype 2 and their use |
| MX2023009059A (es) | 2021-02-02 | 2023-09-15 | Liminal Biosciences Ltd | Antagonistas de gpr84 y usos de estos. |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS58213776A (ja) * | 1982-06-07 | 1983-12-12 | Ishihara Sangyo Kaisha Ltd | ピリダジノン系化合物及びそれらを含有する殺菌剤 |
| JPS62258731A (ja) * | 1986-05-06 | 1987-11-11 | Kao Corp | 水中油型乳化組成物 |
| DE3917469A1 (de) * | 1989-05-30 | 1990-12-06 | Bayer Ag | Heterocyclylpyridine |
| NO179282C (no) * | 1991-01-18 | 1996-09-11 | Rhone Poulenc Agrochimie | Nye 1-(2-pyridyl)pyrazolforbindelser til kontroll av skadeinsekter |
| US5726124A (en) * | 1992-07-17 | 1998-03-10 | Rohm And Haas Company | 2-arylpyrimidines and herbicidal use thereof |
| JPH06172306A (ja) * | 1992-10-05 | 1994-06-21 | Nissan Chem Ind Ltd | 環状アミド化合物および除草剤 |
| DE19518054A1 (de) * | 1995-03-08 | 1996-09-12 | Hoechst Schering Agrevo Gmbh | N-Arylpyrazolketone und deren Derivate, Verfahren zu ihrer Herstellung, sie enthaltende Mittel und ihre Verwendung als Schädlingsbekämpfungsmittel |
| DE19530606A1 (de) * | 1995-08-21 | 1997-02-27 | Basf Ag | 1-(Pyridyl)-pyrazole |
| GB9711753D0 (en) * | 1997-06-06 | 1997-08-06 | Merck Sharp & Dohme | Therapeutic agents |
-
1999
- 1999-04-06 BR BR9909487-8A patent/BR9909487A/pt not_active IP Right Cessation
- 1999-04-06 EP EP99919194A patent/EP1076655A1/en not_active Withdrawn
- 1999-04-06 AU AU37056/99A patent/AU738222B2/en not_active Ceased
- 1999-04-06 CN CN99804531A patent/CN1295570A/zh active Pending
- 1999-04-06 ID IDW20002021A patent/ID27165A/id unknown
- 1999-04-06 WO PCT/EP1999/002313 patent/WO1999052893A1/en not_active Ceased
- 1999-04-06 JP JP2000543452A patent/JP2002511461A/ja active Pending
- 1999-04-06 KR KR1020007011155A patent/KR20010042521A/ko not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| ID27165A (id) | 2001-03-08 |
| EP1076655A1 (en) | 2001-02-21 |
| CN1295570A (zh) | 2001-05-16 |
| JP2002511461A (ja) | 2002-04-16 |
| AU738222B2 (en) | 2001-09-13 |
| AU3705699A (en) | 1999-11-01 |
| WO1999052893A1 (en) | 1999-10-21 |
| KR20010042521A (ko) | 2001-05-25 |
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