AU2002210687A1 - Use of compound in the manufacture of a pharmaceutical for inhibiting steroid sulphatase and steroid dehydrogenase activity - Google Patents
Use of compound in the manufacture of a pharmaceutical for inhibiting steroid sulphatase and steroid dehydrogenase activityInfo
- Publication number
- AU2002210687A1 AU2002210687A1 AU2002210687A AU1068702A AU2002210687A1 AU 2002210687 A1 AU2002210687 A1 AU 2002210687A1 AU 2002210687 A AU2002210687 A AU 2002210687A AU 1068702 A AU1068702 A AU 1068702A AU 2002210687 A1 AU2002210687 A1 AU 2002210687A1
- Authority
- AU
- Australia
- Prior art keywords
- steroid
- pharmaceutical
- manufacture
- compound
- dehydrogenase activity
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- 101710088194 Dehydrogenase Proteins 0.000 title 1
- 102000009134 Steryl-Sulfatase Human genes 0.000 title 1
- 108010087999 Steryl-Sulfatase Proteins 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
- 230000000694 effects Effects 0.000 title 1
- 230000002401 inhibitory effect Effects 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
- 150000003431 steroids Chemical class 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0025788.1A GB0025788D0 (en) | 2000-10-20 | 2000-10-20 | Use |
| GB0025788.1 | 2000-10-20 | ||
| PCT/GB2001/004645 WO2002032409A2 (fr) | 2000-10-20 | 2001-10-18 | Utilisation |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2002210687A1 true AU2002210687A1 (en) | 2002-04-29 |
Family
ID=9901713
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2002210687A Abandoned AU2002210687A1 (en) | 2000-10-20 | 2001-10-18 | Use of compound in the manufacture of a pharmaceutical for inhibiting steroid sulphatase and steroid dehydrogenase activity |
Country Status (3)
| Country | Link |
|---|---|
| AU (1) | AU2002210687A1 (fr) |
| GB (1) | GB0025788D0 (fr) |
| WO (1) | WO2002032409A2 (fr) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1657247B1 (fr) * | 2001-10-18 | 2008-09-17 | Sterix Limited | Composes steroides pour inhiber la sulfatase de steroides |
| PT1448592E (pt) * | 2001-10-18 | 2006-07-31 | Sterix Ltd | Compostos esteroides para inibicao da esteroide sulfatase |
| GB0127923D0 (en) | 2001-11-21 | 2002-01-16 | Sterix Ltd | Compound |
| MXPA04004802A (es) * | 2001-11-21 | 2004-08-11 | Sterix Ltd | Derivados del 1,2,4-triazol que contienen un grupo sulfamato como inhibidores de aromatasa. |
| DE10307103A1 (de) * | 2003-02-19 | 2004-09-09 | Schering Ag | Antitumor wirksame 2-substituierte D-Homostra-1,3,5(10)-trien-3-yl sulfamate |
| GB0306718D0 (en) | 2003-03-24 | 2003-04-30 | Sterix Ltd | Compound |
| US20070275935A1 (en) * | 2003-05-13 | 2007-11-29 | Stewart Alastair G | Estratriene Derivatives |
| US7419972B2 (en) | 2004-07-02 | 2008-09-02 | Schering Ag | 2-substituted estra-1,3,5(10)-trien-17-ones as inhibitors of 17β-hydroxy steroid dehydrogenase type 1 |
| DE102004032674A1 (de) * | 2004-07-02 | 2006-01-26 | Schering Ag | Neue 2-substituierte Estra-1,3,5(10)-trien-17-one als Inhibitoren der 17β-Hydroxysteroiddehydrogenase Typ 1 |
| US8030298B2 (en) | 2005-05-26 | 2011-10-04 | Abbott Products Gmbh | 17β-HSD1 and STS inhibitors |
| GB0604142D0 (en) * | 2006-03-01 | 2006-04-12 | Sterix Ltd | Compound |
| US8288367B2 (en) | 2006-11-30 | 2012-10-16 | Solvay Pharmaceuticals Gmbh | Substituted estratriene derivatives as 17BETA HSD inhibitors |
| CA2671075A1 (fr) * | 2006-11-30 | 2008-06-05 | Solvay Pharmaceuticals Gmbh | Derives oestatrienes substitues en tant qu'inhibiteurs de la 17beta hsd |
| WO2009037539A2 (fr) | 2007-09-17 | 2009-03-26 | Preglem S.A. | Traitement d'états pathologiques œstrogénodépendants chez des femmes pré-ménopausées |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9625334D0 (en) * | 1996-12-05 | 1997-01-22 | Imperial College | Compound |
| DE4447714C2 (de) * | 1994-08-09 | 1998-02-05 | Jenapharm Gmbh | Verwendung von Estra-1,3,5(10)-trien-Derivaten zur Hormonsubstitutions-Therapie |
| GB9422777D0 (en) * | 1994-11-11 | 1995-01-04 | Imperial College | Assay |
| US5880115A (en) * | 1997-07-18 | 1999-03-09 | Duquesne University Of The Holy Ghost | Steroid sulfatase inhibitors and methods for making and using the same |
| GB2331987B (en) * | 1997-12-04 | 2002-11-27 | Imperial College | Polycyclic sulphamate inhibitors of oestrone sulphatase |
| US6046186A (en) * | 1997-12-24 | 2000-04-04 | Sri International | Estrone sulfamate inhibitors of estrone sulfatase, and associated pharmaceutical compositions and methods of use |
| DE60121293T2 (de) * | 2000-01-14 | 2007-06-28 | Sterix Ltd., Slough | Pharmazeutische zusammensetzungen, welche steroidische strukturen enthalten, und deren verwendungen |
-
2000
- 2000-10-20 GB GBGB0025788.1A patent/GB0025788D0/en not_active Ceased
-
2001
- 2001-10-18 WO PCT/GB2001/004645 patent/WO2002032409A2/fr not_active Ceased
- 2001-10-18 AU AU2002210687A patent/AU2002210687A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO2002032409A3 (fr) | 2002-08-08 |
| GB0025788D0 (en) | 2000-12-06 |
| WO2002032409A2 (fr) | 2002-04-25 |
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