AU2001229320A1 - Inhibitors of prenyl-protein transferase - Google Patents
Inhibitors of prenyl-protein transferaseInfo
- Publication number
- AU2001229320A1 AU2001229320A1 AU2001229320A AU2932001A AU2001229320A1 AU 2001229320 A1 AU2001229320 A1 AU 2001229320A1 AU 2001229320 A AU2001229320 A AU 2001229320A AU 2932001 A AU2932001 A AU 2932001A AU 2001229320 A1 AU2001229320 A1 AU 2001229320A1
- Authority
- AU
- Australia
- Prior art keywords
- prenyl
- inhibitors
- protein transferase
- transferase
- protein
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D419/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen, oxygen, and sulfur atoms as the only ring hetero atoms
- C07D419/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen, oxygen, and sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D419/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen, oxygen, and sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US17578400P | 2000-01-12 | 2000-01-12 | |
| US60175784 | 2000-01-12 | ||
| PCT/US2001/000633 WO2001051126A1 (en) | 2000-01-12 | 2001-01-09 | Inhibitors of prenyl-protein transferase |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2001229320A1 true AU2001229320A1 (en) | 2001-07-24 |
Family
ID=22641611
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2001229320A Abandoned AU2001229320A1 (en) | 2000-01-12 | 2001-01-09 | Inhibitors of prenyl-protein transferase |
Country Status (3)
| Country | Link |
|---|---|
| US (1) | US6525074B2 (en) |
| AU (1) | AU2001229320A1 (en) |
| WO (1) | WO2001051126A1 (en) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP4673833B2 (en) * | 2003-01-07 | 2011-04-20 | メルク・シャープ・エンド・ドーム・コーポレイション | Macrocyclic β-secretase inhibitor for the treatment of Alzheimer's disease |
| CA2528375C (en) | 2003-06-18 | 2013-11-19 | Tranzyme Pharma, Inc. | Macrocyclic antagonists of the motilin receptor |
| US20050154451A1 (en) * | 2003-12-18 | 2005-07-14 | Medtronic Vascular, Inc. | Medical devices to treat or inhibit restenosis |
| JP4917021B2 (en) * | 2004-05-03 | 2012-04-18 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | Diastereoselective addition of lithiated N-methylimidazole to sulfimines |
| CA2563806C (en) * | 2004-05-03 | 2012-11-20 | Janssen Pharmaceutica N.V. | Diastereoselective synthesis process with 6-bromo-4-(3-chlorophenyl)-2-methoxy-quinoline |
| WO2006055434A2 (en) * | 2004-11-17 | 2006-05-26 | Merck & Co., Inc. | Macrocyclic tertiary amine beta-secretase inhibitors for the treatment of alzheimer's disease |
| JP2008520727A (en) * | 2004-11-23 | 2008-06-19 | メルク エンド カムパニー インコーポレーテッド | Macrocyclic aminopyridyl beta-secretase inhibitors for the treatment of Alzheimer's disease |
| US7888376B2 (en) * | 2005-11-23 | 2011-02-15 | Bristol-Myers Squibb Company | Heterocyclic CETP inhibitors |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5719148A (en) | 1993-10-15 | 1998-02-17 | Schering Corporation | Tricyclic amide and urea compounds useful for inhibition of g-protein function and for treatment of proliferative diseases |
| US5721236A (en) | 1993-10-15 | 1998-02-24 | Schering Corporation | Tricyclic carbamate compounds useful for inhibition of G-protein function and for treatment of proliferative diseases |
| US5891872A (en) | 1995-04-07 | 1999-04-06 | Schering Corporation | Tricyclic compounds |
| US5801175A (en) | 1995-04-07 | 1998-09-01 | Schering Corporation | Tricyclic compounds useful for inhibition of G-protein function and for treatment of proliferative diseases |
| US5712280A (en) | 1995-04-07 | 1998-01-27 | Schering Corporation | Tricyclic compounds useful for inhibition of G-protein function and for treatment of proliferative diseases |
| US5756528A (en) | 1995-06-06 | 1998-05-26 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
| US5968965A (en) | 1996-01-30 | 1999-10-19 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
| JP2000504017A (en) | 1996-01-30 | 2000-04-04 | メルク エンド カンパニー インコーポレーテッド | Farnesyl-protein transferase inhibitor |
| US5981562A (en) | 1996-01-30 | 1999-11-09 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
| US6028201A (en) | 1996-01-30 | 2000-02-22 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
| US5922883A (en) | 1996-04-03 | 1999-07-13 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
| US5780488A (en) | 1996-04-03 | 1998-07-14 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
| JP2001500515A (en) | 1996-09-13 | 2001-01-16 | シェーリング コーポレイション | Compounds useful for inhibiting farnesyl protein transferase |
| JP2002519428A (en) | 1998-07-02 | 2002-07-02 | メルク エンド カムパニー インコーポレーテッド | Inhibitors of prenyl-protein transferase |
| AU760028B2 (en) | 1998-07-02 | 2003-05-08 | Merck & Co., Inc. | Inhibitors of prenyl-protein transferase |
| EP1091736A4 (en) | 1998-07-02 | 2001-10-24 | Merck & Co Inc | Inhibitors of prenyl-protein transferase |
-
2001
- 2001-01-09 AU AU2001229320A patent/AU2001229320A1/en not_active Abandoned
- 2001-01-09 US US09/757,251 patent/US6525074B2/en not_active Expired - Fee Related
- 2001-01-09 WO PCT/US2001/000633 patent/WO2001051126A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| US20020049217A1 (en) | 2002-04-25 |
| US6525074B2 (en) | 2003-02-25 |
| WO2001051126A1 (en) | 2001-07-19 |
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