ATE354365T1 - N-thiazol-2-yl-benzamid-derivate - Google Patents
N-thiazol-2-yl-benzamid-derivateInfo
- Publication number
- ATE354365T1 ATE354365T1 AT04762951T AT04762951T ATE354365T1 AT E354365 T1 ATE354365 T1 AT E354365T1 AT 04762951 T AT04762951 T AT 04762951T AT 04762951 T AT04762951 T AT 04762951T AT E354365 T1 ATE354365 T1 AT E354365T1
- Authority
- AT
- Austria
- Prior art keywords
- thiazole
- benzamide derivatives
- benzamide
- derivatives
- Prior art date
Links
- SCQBDADQAVXTMZ-UHFFFAOYSA-N n-(1,3-thiazol-2-yl)benzamide Chemical class C=1C=CC=CC=1C(=O)NC1=NC=CS1 SCQBDADQAVXTMZ-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/44—Acylated amino or imino radicals
- C07D277/46—Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Biomedical Technology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Epidemiology (AREA)
- Psychiatry (AREA)
- Psychology (AREA)
- Pain & Pain Management (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Vascular Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DKPA200301579 | 2003-10-27 | ||
| DKPA200400229 | 2004-02-13 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE354365T1 true ATE354365T1 (de) | 2007-03-15 |
Family
ID=34524309
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT04762951T ATE354365T1 (de) | 2003-10-27 | 2004-10-25 | N-thiazol-2-yl-benzamid-derivate |
Country Status (28)
| Country | Link |
|---|---|
| US (2) | US20060154974A1 (de) |
| EP (2) | EP1803455A1 (de) |
| JP (1) | JP2007509083A (de) |
| KR (1) | KR20060093726A (de) |
| AR (1) | AR047621A1 (de) |
| AT (1) | ATE354365T1 (de) |
| AU (1) | AU2004283019A1 (de) |
| BR (1) | BRPI0415661A (de) |
| CA (1) | CA2542816A1 (de) |
| CO (1) | CO5690582A2 (de) |
| CY (1) | CY1106526T1 (de) |
| DE (1) | DE602004004925T2 (de) |
| DK (1) | DK1682129T3 (de) |
| EA (2) | EA200801734A1 (de) |
| ES (1) | ES2279414T3 (de) |
| HR (1) | HRP20070194T3 (de) |
| IL (1) | IL175189A0 (de) |
| IS (1) | IS8364A (de) |
| ME (1) | MEP6708A (de) |
| MX (1) | MXPA06004436A (de) |
| NO (1) | NO20062417L (de) |
| PL (1) | PL1682129T3 (de) |
| PT (1) | PT1682129E (de) |
| RS (1) | RS20060289A (de) |
| SG (1) | SG147472A1 (de) |
| SI (1) | SI1682129T1 (de) |
| TW (1) | TW200524887A (de) |
| WO (1) | WO2005039572A1 (de) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20060106040A1 (en) | 2002-12-19 | 2006-05-18 | Michael Grzelak | Adenosine A2a receptor antagonists for the treatment of extra-pyramidal syndrome and other movement disorders |
| TW200524887A (en) * | 2003-10-27 | 2005-08-01 | Lundbeck & Co As H | N-thiazol-2-yl-benzamide derivatives |
| EP1794157B1 (de) | 2004-09-22 | 2014-02-26 | H. Lundbeck A/S | 2-acylaminothiazol derivate |
| US7674912B2 (en) | 2005-04-25 | 2010-03-09 | H. Lundbeck A/S | Pro-drugs of N-thiazol-2-yl-benzamide derivatives |
| TW200720264A (en) * | 2005-04-25 | 2007-06-01 | Lundbeck & Co As H | Pro-drugs of n-thiazol-2-yl-benzamide derivatives |
| EP1894930A4 (de) * | 2005-06-23 | 2010-06-23 | Kyowa Hakko Kirin Co Ltd | Thiazolderivat |
| SI1921077T1 (sl) * | 2005-08-02 | 2017-11-30 | Kyowa Hakko Kirin Co., Ltd. | Sredstvo za zdravljenje in/ali preprečevanje motnje spanja |
| ES2273599B1 (es) | 2005-10-14 | 2008-06-01 | Universidad De Barcelona | Compuestos para el tratamiento de la fibrilacion auricular. |
| EP2210891A1 (de) * | 2009-01-26 | 2010-07-28 | Domain Therapeutics | Neue Adenosin-Rezeptorliganden und Verwendungen davon |
| GB201106817D0 (en) | 2011-04-21 | 2011-06-01 | Astex Therapeutics Ltd | New compound |
| RU2483722C1 (ru) * | 2012-05-22 | 2013-06-10 | Автономная Некоммерческая Организация "Научно-Исследовательский Центр Биотехнологии Антибиотиков И Других Биологически Активных Веществ "Биоан" | Аминотиазольные производные усниновой кислоты как новые противотуберкулезные агенты |
| US9980973B2 (en) | 2012-10-19 | 2018-05-29 | Astex Therapeutics Limited | Bicyclic heterocycle compounds and their uses in therapy |
| GB201218864D0 (en) | 2012-10-19 | 2012-12-05 | Astex Therapeutics Ltd | Bicyclic heterocycle compounds and their uses in therapy |
| GB201218862D0 (en) | 2012-10-19 | 2012-12-05 | Astex Therapeutics Ltd | Bicyclic heterocycle compounds and their uses in therapy |
| GB201218850D0 (en) | 2012-10-19 | 2012-12-05 | Astex Therapeutics Ltd | Bicyclic heterocycle compounds and their uses in therapy |
| CN105829310B (zh) | 2013-12-20 | 2019-04-12 | 阿斯特克斯治疗有限公司 | 双环杂环化合物及其治疗用途 |
| ES2578363B1 (es) * | 2015-01-22 | 2017-01-31 | Palobiofarma, S.L. | Moduladores de los receptores A3 de adenosina |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE855120C (de) * | 1950-10-08 | 1953-01-05 | Schering Ag | Verfahren zur Herstellung von Aminosalicylsaeureamiden |
| JP2903339B2 (ja) * | 1990-10-12 | 1999-06-07 | 大日精化工業株式会社 | 電子写真感光体 |
| CN1072652C (zh) * | 1996-10-24 | 2001-10-10 | 泽里新药工业株式会社 | 取代的苯甲酰氨基噻唑衍生物以及含有它们的药物 |
| GB9823871D0 (en) * | 1998-10-30 | 1998-12-23 | Pharmacia & Upjohn Spa | 2-Amino-thiazole derivatives, process for their preparation, and their use as antitumour agents |
| GB0028383D0 (en) * | 2000-11-21 | 2001-01-03 | Novartis Ag | Organic compounds |
| CN1516696A (zh) * | 2001-01-26 | 2004-07-28 | 盐野义制药株式会社 | 对血小板生成素受体具有激动作用的卤素化合物 |
| US7429593B2 (en) * | 2001-09-14 | 2008-09-30 | Shionogi & Co., Ltd. | Utilities of amide compounds |
| US6624163B2 (en) * | 2001-11-29 | 2003-09-23 | Hoffman-La Roche Inc. | Benzothiazole derivatives |
| US6713499B2 (en) * | 2001-12-12 | 2004-03-30 | Hoffman-La Roche Inc. | 7-Amino-benzothiazole derivatives |
| TW200524887A (en) * | 2003-10-27 | 2005-08-01 | Lundbeck & Co As H | N-thiazol-2-yl-benzamide derivatives |
| CA2551611C (en) * | 2003-12-26 | 2013-06-25 | Kyowa Hakko Kogyo Co., Ltd. | Thiazole derivatives for treating or preventing parkinson's disease |
| US7674912B2 (en) * | 2005-04-25 | 2010-03-09 | H. Lundbeck A/S | Pro-drugs of N-thiazol-2-yl-benzamide derivatives |
-
2004
- 2004-10-08 TW TW093130498A patent/TW200524887A/zh unknown
- 2004-10-21 AR ARP040103822A patent/AR047621A1/es not_active Application Discontinuation
- 2004-10-25 KR KR1020067008181A patent/KR20060093726A/ko not_active Ceased
- 2004-10-25 ES ES04762951T patent/ES2279414T3/es not_active Expired - Lifetime
- 2004-10-25 RS YUP-2006/0289A patent/RS20060289A/sr unknown
- 2004-10-25 EA EA200801734A patent/EA200801734A1/ru unknown
- 2004-10-25 AU AU2004283019A patent/AU2004283019A1/en not_active Abandoned
- 2004-10-25 JP JP2006535952A patent/JP2007509083A/ja not_active Withdrawn
- 2004-10-25 EA EA200600860A patent/EA010790B1/ru not_active IP Right Cessation
- 2004-10-25 DK DK04762951T patent/DK1682129T3/da active
- 2004-10-25 WO PCT/DK2004/000733 patent/WO2005039572A1/en not_active Ceased
- 2004-10-25 ME MEP-67/08A patent/MEP6708A/xx unknown
- 2004-10-25 SI SI200430225T patent/SI1682129T1/sl unknown
- 2004-10-25 DE DE602004004925T patent/DE602004004925T2/de not_active Expired - Fee Related
- 2004-10-25 EP EP07102639A patent/EP1803455A1/de not_active Withdrawn
- 2004-10-25 CA CA002542816A patent/CA2542816A1/en not_active Abandoned
- 2004-10-25 EP EP04762951A patent/EP1682129B1/de not_active Expired - Lifetime
- 2004-10-25 AT AT04762951T patent/ATE354365T1/de not_active IP Right Cessation
- 2004-10-25 HR HR20070194T patent/HRP20070194T3/xx unknown
- 2004-10-25 SG SG200807988-1A patent/SG147472A1/en unknown
- 2004-10-25 PL PL04762951T patent/PL1682129T3/pl unknown
- 2004-10-25 BR BRPI0415661-7A patent/BRPI0415661A/pt not_active IP Right Cessation
- 2004-10-25 MX MXPA06004436A patent/MXPA06004436A/es active IP Right Grant
- 2004-10-25 PT PT04762951T patent/PT1682129E/pt unknown
-
2005
- 2005-12-20 US US11/312,661 patent/US20060154974A1/en not_active Abandoned
-
2006
- 2006-03-20 IS IS8364A patent/IS8364A/is unknown
- 2006-04-25 IL IL175189A patent/IL175189A0/en unknown
- 2006-04-25 CO CO06039105A patent/CO5690582A2/es not_active Application Discontinuation
- 2006-05-26 NO NO20062417A patent/NO20062417L/no not_active Application Discontinuation
-
2007
- 2007-04-19 CY CY20071100529T patent/CY1106526T1/el unknown
-
2008
- 2008-12-19 US US12/339,438 patent/US20090247593A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| KR20060093726A (ko) | 2006-08-25 |
| IL175189A0 (en) | 2006-09-05 |
| EA010790B1 (ru) | 2008-10-30 |
| NO20062417L (no) | 2006-05-26 |
| EA200801734A1 (ru) | 2008-12-30 |
| TW200524887A (en) | 2005-08-01 |
| MEP6708A (xx) | 2010-02-10 |
| HRP20070194T3 (hr) | 2007-06-30 |
| EP1803455A1 (de) | 2007-07-04 |
| DE602004004925T2 (de) | 2007-10-31 |
| PT1682129E (pt) | 2007-04-30 |
| CY1106526T1 (el) | 2012-01-25 |
| RS20060289A (sr) | 2008-06-05 |
| EA200600860A1 (ru) | 2006-08-25 |
| JP2007509083A (ja) | 2007-04-12 |
| EP1682129A1 (de) | 2006-07-26 |
| US20090247593A1 (en) | 2009-10-01 |
| SI1682129T1 (sl) | 2007-06-30 |
| MXPA06004436A (es) | 2006-06-20 |
| CA2542816A1 (en) | 2005-05-06 |
| DK1682129T3 (da) | 2007-06-11 |
| ES2279414T3 (es) | 2007-08-16 |
| WO2005039572A1 (en) | 2005-05-06 |
| SG147472A1 (en) | 2008-11-28 |
| BRPI0415661A (pt) | 2006-12-19 |
| US20060154974A1 (en) | 2006-07-13 |
| EP1682129B1 (de) | 2007-02-21 |
| AU2004283019A1 (en) | 2005-05-06 |
| IS8364A (is) | 2006-03-20 |
| AR047621A1 (es) | 2006-02-01 |
| PL1682129T3 (pl) | 2007-07-31 |
| CO5690582A2 (es) | 2006-10-31 |
| DE602004004925D1 (de) | 2007-04-05 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification |
Ref document number: 1682129 Country of ref document: EP |
|
| REN | Ceased due to non-payment of the annual fee |