AR106423A1 - Un proceso para la preparación de triptaminas y sus derivados - Google Patents
Un proceso para la preparación de triptaminas y sus derivadosInfo
- Publication number
- AR106423A1 AR106423A1 ARP160103209A ARP160103209A AR106423A1 AR 106423 A1 AR106423 A1 AR 106423A1 AR P160103209 A ARP160103209 A AR P160103209A AR P160103209 A ARP160103209 A AR P160103209A AR 106423 A1 AR106423 A1 AR 106423A1
- Authority
- AR
- Argentina
- Prior art keywords
- alkyl
- aryl
- alkoxy
- substituted
- compound
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/32—Oxygen atoms
- C07D209/34—Oxygen atoms in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
- C07D209/16—Tryptamines
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Abstract
Reivindicación 1: Un proceso para la preparación del compuesto de la fórmula (1) o una sal de este, en donde el anillo aromático opcionalmente puede sustituirse con uno o más sustituyentes seleccionados a partir de alquilo, alquilo sustituido con alcoxi o hidroxilo, cicloalquilo, arilo, arilo sustituido con hidroxilo, alquilo, alcoxi, halógeno, carboxi, alcoxicarbonilo, amido, N-alquilamido, sulfonilamido, ciano, haloalquilo, haloalcoxi, nitro, heteroarilo, heterociclilo, alquenilo, alquinilo, halógeno, hidroxilo, alcoxi, ariloxi, alcoxicarbonilo, ariloxicarbonilo, tiol, tioéter de alquilo, tioéter de arilo, tioéster de alquilo, tioéster de arilo, grupo aldehído, arilcarbonilo, alquilocarbonilo, carboxilo, carboxilo esterificado con alquilo o arilo, amida, amina, nitrilo, alquilsulfonilo, arilsulfonilo y amidosulfonilo, que comprenden la conversión del compuesto de la fórmula (2), en donde el anillo aromático opcionalmente puede sustituirse con uno o más sustituyentes como se definió anteriormente, en el compuesto de la fórmula (1) en presencia de un agente reductor.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP2015002105 | 2015-10-23 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR106423A1 true AR106423A1 (es) | 2018-01-10 |
Family
ID=57209421
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP160103209A AR106423A1 (es) | 2015-10-23 | 2016-10-21 | Un proceso para la preparación de triptaminas y sus derivados |
Country Status (3)
| Country | Link |
|---|---|
| CN (1) | CN108271369A (es) |
| AR (1) | AR106423A1 (es) |
| WO (1) | WO2017067670A1 (es) |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5403851A (en) | 1994-04-05 | 1995-04-04 | Interneuron Pharmaceuticals, Inc. | Substituted tryptamines, phenalkylamines and related compounds |
| EE9800353A (et) | 1996-04-23 | 1999-04-15 | Merck & Co., Inc. | Pürasinoonidest trombiini inhibiitorid |
| EP1268477B1 (en) | 2000-03-15 | 2010-04-21 | Sanofi-Aventis Deutschland GmbH | Substituted beta-carbolines with ikb-kinase inhibiting activity |
| KR100894189B1 (ko) | 2001-03-29 | 2009-04-22 | 일라이 릴리 앤드 캄파니 | 5-ｈｔ6 수용체의 길항제로서의 ｎ-(2-아릴에틸)벤질아민 |
| GB0119243D0 (en) | 2001-08-07 | 2001-10-03 | Pharma Mar Sa | Antitumoral analogs of ET-743 |
| US7595311B2 (en) | 2002-05-24 | 2009-09-29 | Exelixis, Inc. | Azepinoindole derivatives as pharmaceutical agents |
| DE10252667A1 (de) | 2002-11-11 | 2004-05-27 | Grünenthal GmbH | Spirocyclische Cyclohexan-Derivate |
| US7645886B2 (en) * | 2002-12-20 | 2010-01-12 | Ciba Specialty Corporation | Synthesis of amines and intermediates for the synthesis thereof |
| JP2006522824A (ja) | 2003-04-09 | 2006-10-05 | ミレニアム・ファーマシューティカルズ・インコーポレイテッド | 炎症性疾患を処置するために有用なβ−カルボリン |
| JP2007532582A (ja) | 2004-04-09 | 2007-11-15 | ミレニアム・ファーマシューティカルズ・インコーポレイテッド | 炎症性疾患の処置に有用なβ−カルボリン |
| CA2657227A1 (en) | 2006-07-14 | 2008-01-17 | Novartis Ag | Pyrimidine derivatives as alk-5 inhibitors |
| DE102006033109A1 (de) * | 2006-07-18 | 2008-01-31 | Grünenthal GmbH | Substituierte Heteroaryl-Derivate |
| WO2009073118A1 (en) | 2007-12-04 | 2009-06-11 | Merck & Co., Inc. | Tryptamine sulfonamides as 5-ht6 antagonists |
| KR20110071004A (ko) | 2008-10-14 | 2011-06-27 | 액테리온 파마슈티칼 리미티드 | 페네틸아미드 유도체 및 이의 헤테로시클릭 유사체 |
| WO2010080864A1 (en) | 2009-01-12 | 2010-07-15 | Array Biopharma Inc. | Piperidine-containing compounds and use thereof |
| CN102177686A (zh) | 2009-06-12 | 2011-09-07 | 华为技术有限公司 | 一种传送视频报文的方法、路由器设备及系统 |
| TW201139370A (en) * | 2009-12-23 | 2011-11-16 | Lundbeck & Co As H | Processes for the manufacture of a pharmaceutically active agent |
| CN102659662A (zh) * | 2012-03-28 | 2012-09-12 | 华东师范大学 | 3-r-3-羟基-2-氧化吲哚类化合物的合成方法 |
-
2016
- 2016-10-19 WO PCT/EP2016/025121 patent/WO2017067670A1/en not_active Ceased
- 2016-10-19 CN CN201680061481.4A patent/CN108271369A/zh active Pending
- 2016-10-21 AR ARP160103209A patent/AR106423A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2017067670A1 (en) | 2017-04-27 |
| CN108271369A (zh) | 2018-07-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure | ||
| FB | Suspension of granting procedure | ||
| FB | Suspension of granting procedure |