AR074607A1 - Oximeteres e hidrazonas de tiazolilo como agentes fitoprotectores. - Google Patents
Oximeteres e hidrazonas de tiazolilo como agentes fitoprotectores.Info
- Publication number
- AR074607A1 AR074607A1 ARP090104825A ARP090104825A AR074607A1 AR 074607 A1 AR074607 A1 AR 074607A1 AR P090104825 A ARP090104825 A AR P090104825A AR P090104825 A ARP090104825 A AR P090104825A AR 074607 A1 AR074607 A1 AR 074607A1
- Authority
- AR
- Argentina
- Prior art keywords
- alkyl
- haloalkyl
- substituents
- cycloalkyl
- phenyl
- Prior art date
Links
- 150000007857 hydrazones Chemical class 0.000 title 1
- 239000003223 protective agent Substances 0.000 title 1
- 125000001424 substituent group Chemical group 0.000 abstract 21
- 125000000217 alkyl group Chemical group 0.000 abstract 16
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 16
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 14
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 abstract 13
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 13
- 125000006583 (C1-C3) haloalkyl group Chemical group 0.000 abstract 12
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 abstract 12
- 229910052736 halogen Inorganic materials 0.000 abstract 12
- 150000002367 halogens Chemical class 0.000 abstract 12
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 11
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 10
- 125000000232 haloalkynyl group Chemical group 0.000 abstract 10
- 125000004448 alkyl carbonyl group Chemical group 0.000 abstract 9
- 125000000262 haloalkenyl group Chemical group 0.000 abstract 9
- 125000005347 halocycloalkyl group Chemical group 0.000 abstract 9
- 125000001181 organosilyl group Chemical group [SiH3]* 0.000 abstract 9
- -1 1-methoxycyclopropyl Chemical group 0.000 abstract 8
- 125000005119 alkyl cycloalkyl group Chemical group 0.000 abstract 8
- 125000001188 haloalkyl group Chemical group 0.000 abstract 8
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 6
- 125000000229 (C1-C4)alkoxy group Chemical group 0.000 abstract 6
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 abstract 6
- 125000004414 alkyl thio group Chemical group 0.000 abstract 6
- 125000001316 cycloalkyl alkyl group Chemical group 0.000 abstract 6
- 125000004995 haloalkylthio group Chemical group 0.000 abstract 6
- 125000005196 alkyl carbonyloxy group Chemical group 0.000 abstract 5
- 125000005120 alkyl cycloalkyl alkyl group Chemical group 0.000 abstract 5
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 5
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 5
- 229910052739 hydrogen Inorganic materials 0.000 abstract 5
- 239000001257 hydrogen Substances 0.000 abstract 5
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 5
- 125000004768 (C1-C4) alkylsulfinyl group Chemical group 0.000 abstract 4
- 125000004769 (C1-C4) alkylsulfonyl group Chemical group 0.000 abstract 4
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 abstract 4
- 125000004771 (C1-C4) haloalkylsulfinyl group Chemical group 0.000 abstract 4
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 4
- 125000003320 C2-C6 alkenyloxy group Chemical group 0.000 abstract 4
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical compound [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 abstract 4
- 125000004183 alkoxy alkyl group Chemical group 0.000 abstract 4
- 125000005133 alkynyloxy group Chemical group 0.000 abstract 4
- 229910052799 carbon Inorganic materials 0.000 abstract 4
- 150000002431 hydrogen Chemical class 0.000 abstract 4
- 229910052757 nitrogen Inorganic materials 0.000 abstract 4
- 125000006700 (C1-C6) alkylthio group Chemical group 0.000 abstract 3
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 abstract 3
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 abstract 3
- 125000002485 formyl group Chemical group [H]C(*)=O 0.000 abstract 3
- 125000004441 haloalkylsulfonyl group Chemical group 0.000 abstract 3
- 125000001183 hydrocarbyl group Chemical group 0.000 abstract 3
- 229910052760 oxygen Inorganic materials 0.000 abstract 3
- 229920006395 saturated elastomer Chemical group 0.000 abstract 3
- 229910052717 sulfur Inorganic materials 0.000 abstract 3
- 241000233866 Fungi Species 0.000 abstract 2
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 2
- 125000003545 alkoxy group Chemical group 0.000 abstract 2
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 2
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 125000000000 cycloalkoxy group Chemical group 0.000 abstract 2
- 125000004438 haloalkoxy group Chemical group 0.000 abstract 2
- 125000004692 haloalkylcarbonyl group Chemical group 0.000 abstract 2
- 125000001072 heteroaryl group Chemical group 0.000 abstract 2
- 125000005842 heteroatom Chemical group 0.000 abstract 2
- 125000000623 heterocyclic group Chemical group 0.000 abstract 2
- 238000000034 method Methods 0.000 abstract 2
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 2
- QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 abstract 2
- 125000004043 oxo group Chemical group O=* 0.000 abstract 2
- 239000001301 oxygen Substances 0.000 abstract 2
- 230000003032 phytopathogenic effect Effects 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 239000011593 sulfur Substances 0.000 abstract 2
- 125000004454 (C1-C6) alkoxycarbonyl group Chemical group 0.000 abstract 1
- 125000004738 (C1-C6) alkyl sulfinyl group Chemical group 0.000 abstract 1
- 125000004916 (C1-C6) alkylcarbonyl group Chemical group 0.000 abstract 1
- 125000004739 (C1-C6) alkylsulfonyl group Chemical group 0.000 abstract 1
- 125000004749 (C1-C6) haloalkylsulfinyl group Chemical group 0.000 abstract 1
- 125000004741 (C1-C6) haloalkylsulfonyl group Chemical group 0.000 abstract 1
- 125000006376 (C3-C10) cycloalkyl group Chemical group 0.000 abstract 1
- 125000006570 (C5-C6) heteroaryl group Chemical group 0.000 abstract 1
- YBYIRNPNPLQARY-UHFFFAOYSA-N 1H-indene Natural products C1=CC=C2CC=CC2=C1 YBYIRNPNPLQARY-UHFFFAOYSA-N 0.000 abstract 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 125000005083 alkoxyalkoxy group Chemical group 0.000 abstract 1
- 125000005130 alkyl carbonyl thio group Chemical group 0.000 abstract 1
- 125000000392 cycloalkenyl group Chemical group 0.000 abstract 1
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 1
- 125000005366 cycloalkylthio group Chemical group 0.000 abstract 1
- 125000004994 halo alkoxy alkyl group Chemical group 0.000 abstract 1
- 125000006769 halocycloalkoxy group Chemical group 0.000 abstract 1
- 125000003454 indenyl group Chemical group C1(C=CC2=CC=CC=C12)* 0.000 abstract 1
- 125000001624 naphthyl group Chemical group 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- 125000004430 oxygen atom Chemical group O* 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
- A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
- A01N43/78—1,3-Thiazoles; Hydrogenated 1,3-thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Environmental Sciences (AREA)
- Zoology (AREA)
- Wood Science & Technology (AREA)
- Dentistry (AREA)
- Plant Pathology (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Diabetes (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Hematology (AREA)
- Animal Behavior & Ethology (AREA)
- Obesity (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
Así corno sus sales agroquímicamente activas y su uso para combatir hongos perjudiciales fitopatógenos, así como procedimientos para combatir hongos perjudiciales fitopatógenos y procedimientos para preparar los compuestos de la fórmula (1). Reivindicación 1: Compuestos de la fórmula (1) en la que los símbolos tienen los significados siguientes: A representa metilo o A representa fenilo sustituido o no sustituido, seleccionándose los sustituyentes, independientemente unos de otros de la lista siguiente: ciano, nitro, halógeno, alquilo C1-6, haloalquilo C1-3, cicloalquilo C3-6, halocicloalquilo C3-6, cicloalquilalquilo C4-10, alquilcicloalquilo C4-10, alquilcicloalquilalquilo C5-10, alquenilo C2-6, haloalquenilo C2-6, alquinilo C2-6, haloalquinilo C2-6, tri(alquil C1-2)sililo, bencilo, fenilo, hidroxilo, alcoxi C1-4, haloalcoxi C1-4, OCH2OCH3, SH, alquiltio C1-4, haloalquiltio C1-6, CHO, COOH, alcoxi C1-4-carbonilo, CONR4R5, CR4=NOR5, alquil C1-4-carbonilo, haloalquil C1-4-carbonilo, alquil C1-4-carboniloxi, alquil C1-4-carboniltio, alquilsulfinilo C1-4, haloalquilsulfinilo C1-4, alquilsulfonilo C1-4, haloalquilsulfonilo C1-4, NR4R5, NR4COR5, SF5, SO2NR4R5, alcoxialquilo C2-4 o 1-metoxiciclopropilo o A es un heteroarilo de 5 o 6 miembros, dado el caso benzocondensado, sustituido o no sustituido, seleccionándose los sustituyentes independientemente unos de otros, de la lista siguiente: Sustituyentes en el carbono: ciano, nitro, halógeno, alquilo C1-6, haloalquilo C1-3, cicloalquilo C3-6, halocicloalquilo C3-6, cicloalquilalquilo C4-10, alquilcicloalquilo C4-10, alquilcicloalquilalquilo C5-10, alquenilo C2-6, haloalquenilo C2-6, alquinilo C2-6, haloalquinilo C2-6, tri(alquil C1-2)sililo, bencilo, fenilo, hidroxilo, alcoxi C1-4, haloalcoxi C1-4, OCH2OCH3, SH, alquiltio C1-4, haloalquiltio C1-6, CHO, COOH, alcoxi C1-4-carbonilo, CONR4R5, CR4=NOR5, alquil C1-4-carbonilo, haloalquil C1-4-carbonilo, alquil C1-4-carboniloxi, alquil C1-4-carboniltio, alquilsulfinilo C1-4, haloalquilsulfinilo C1-4, alquilsulfonilo C1-4, haloalquilsulfonilo C1-4, NR4R5, NR4COR5, SF5, SO2NR4R5, alcoxialquilo C2-4 o 1-metoxiciclopropilo, Sustituyentes en el nitrógeno: hidroxilo, NR4R5, alquilo C1-6, haloalquilo C1-3, cicloalquilo C3-6, halocicloalquilo C3-6, alquilcicloalquilo C4-10, alquenilo C2-6, haloalquenilo C2-6, alquinilo C2-6 o haloalquinilo C2-6; L1 es (C(R1)2)n, con n = 0 a 3; R1 es igual o diferente, independientemente uno de otro, hidrógeno, halógeno, alquilo C1-2, haloalquilo C1-2 o ciano, con la condición de que L1 puede contener como máximo cuatro R1 que sean distintos de hidrógeno; Y representa azufre u oxígeno; W es una cadena de hidrocarburo C1 a C3 no sustituida o monosustituida, seleccionándose el sustituyente de entre oxo, hidroxilo, ciano o alquilo C1-4; X es una cadena de hidrocarburo C1 a C2 no sustituida o monosustituida seleccionándose el sustituyente de entre oxo, hidroxilo, ciano o alquilo C1-4; R2 representa hidrógeno, alquilo C1-2, haloalquilo C1-2 o halógeno; L2 representa -CH=N-O-, -C(R6)=N-O-, -CH=N-N(R7)- o -C(R6)=N-N(R7)-; L3 representa un enlace directo, o L3 representa una cadena de hidrocarburo C1 a C4, que puede contener hasta cuatro sustituyentes, seleccionándose los sustituyentes, independientemente unos de otros de la lista siguiente: halógeno, alquilo C1-2, alcoxi C1-2, haloalquilo C1-2 o cicloalquilo C3-6; R3 representa metilo, haloalquilo C1-2, -CH=CH2, -C:::CH o cicloalquilo C3-10 no sustituido o monosustituido, seleccionándose el sustituyente de la lista siguiente: ciano, halógeno, alquilo C1-6, haloalquilo C1-3, cicloalquilo C3-6, alquenilo C2-6, haloalquenilo C2-6, alquinilo C2-6, haloalquinilo C2-6, tri(alquil C1-2)sililo, fenilo, hidroxilo, alcoxi C1-6, haloalcoxi C1-6, alqueniloxi C2-6, alquiniloxi C2-6, alquiltio C1-6, haloalquiltio C1-6, o R3 representa fenilo sustituido o no sustituido, seleccionándose los sustituyentes, independientemente unos de otros, de la lista siguiente: ciano, nitro, halógeno, alquilo C1-6, haloalquilo C1-3, cicloalquilo C3-6, halocicloalquilo C3-6, cicloalquilalquilo C4-10, halocicloalquilalquilo C4-10, alquilcicloalquilo C4-10, alquilcicloalquilalquilo C5-10, cicloalcoxialquilo C4-10, alquenilo C2-6, haloalquenilo C2-6, cicloalquenilo C3-8, halocicloalquenilo C3-8, alquinilo C2-6, haloalquinilo C2-6, alcoxialquilo C2-6, haloalcoxialquilo C2-6, alcoxialcoxialquilo C3-8, tri(alquil C1-2)sililo, bencilo, fenilo, hidroxilo, alcoxi C1-6, alcoxialcoxi C2-6, haloalcoxi C1-6, alqueniloxi C2-6, haloalqueniloxi C2-6, alquiniloxi C2-6, haloalquiniloxi C2-6, cicloalcoxi C3-6, cicloalquiloxi C3-6, halocicloalcoxi C3-6, cicloalquilalquiloxi C4-10, NR4R5, SH, SF5, alquiltio C1-6, haloalquiltio C1-6, alquilalquiltio C2-6, cicloalquiltio C3-6, CHO, COOH, alcoxi C1-6-carbonilo, CONR4R5, CR4=NOR5, alquilo C1-6-carbonilo, haloalquilo C1-6-carbonilo, alquilo C1-6-carboniloxi, haloalquilo C1-6-carboniloxi, alquil C1-6-carboniltio, alquilsulfinilo C1-6, haloalquilsulfinilo C1-6, alquilsulfonilo C1-6, haloalquilsulfonilo C1-6, NR4COR5, o SO2NR4R5, o R3 representa indenilo o naftilo, saturado o parcial o totalmente insaturado, que puede contener hasta dos sustituyentes, seleccionándose los sustituyentes, independientemente uno de otro, de la lista siguiente: ciano, halógeno, alquilo C1-6, haloalquilo C1-3, cicloalquilo C3-6, alquenilo C2-6, haloalquenilo C2-6, alquinilo C2-6, haloalquinilo C2-6, tri(alquil C1-2)sililo, fenilo, hidroxilo, alcoxi C1-6, haloalcoxi C1-6, alqueniloxi C2-6, alquiniloxi C2-6, alquiltio C1-6 o haloalquiltio C1-6, o R3 representa un resto heteroarilo de 5 o 6 miembros, sustituido o no sustituido, seleccionándose los sustituyentes, independientemente unos de otros de la lista siguiente: Sustituyentes en el carbono: ciano, nitro, halógeno, alquilo C1-6, haloalquilo C1-3, cicloalquilo C3-6, halocicloalquilo C3-6, cicloalquilalquilo C4-10, alquilcicloalquilo C4-10, alquilcicloalquilalquilo C5-10, alquenilo C2-6, haloalquenilo C2-6, alquinilo C2-6, haloalquinilo C2-6, tri(alquil C1-2)sililo, bencilo, fenilo, hidroxilo, alcoxi C1-4, haloalcoxi C1-4, OCH2OCH3, SH, alquiltio C1-4, haloalquiltio C1-6, COOH, alcoxi C1-4-carbonilo, CONR4R5, alquil C1-4-carbonilo, haloalquil C1-4-carbonilo, alquil C1-4-carboniloxi, alquil C1-4-carboniltio, alquilsulfinilo C1-4, haloalquilsulfinilo C1-4, alquilsulfonilo C1-4, haloalquilsulfonilo C1-4, NR4R5, NR4COR5, SF5, SO2NR4R5, alcoxialquilo C2-4 o 1-metoxiciclopropilo, Sustituyentes en el nitrógeno: hidroxilo, alquilo C1-6, haloalquilo C1-3, cicloalquilo C3-6, halocicloalquilo C3-6, alquilcicloalquilo C4-10, alquenilo C2-6, haloalquenilo C2-6, alquinilo C2-6 o haloalquinilo C2-6 o fenilo o R3 representa heteroarilo de 5 o 6 miembros benzocondensado, sustituido o no sustituido, que puede contener hasta dos sustituyentes, seleccionándose los sustituyentes independientemente uno de otro de la lista siguiente: Sustituyentes en el carbono: ciano, nitro, halógeno, alquilo C1-6, haloalquilo C1-3, cicloalquilo C3-6, halocicloalquilo C3-6, cicloalquilalquilo C4-10, alquilcicloalquilo C4-10, alquilcicloalquilalquilo C5-10, alquenilo C2-6, haloalquenilo C2-6, alquinilo C2-6, haloalquinilo C2-6, tri(alquil C1-2)sililo, bencilo, fenilo, hidroxilo, alcoxi C1-4, haloalcoxi C1-4, OCH2OCH3, SH, alquiltio C1-4, haloalquiltio C1-6, COOH, alcoxi C1-4-carbonilo, CONR4R5, alquil C1-4-carbonilo, haloalquil C1-4-carbonilo, alquil C1-4-carboniloxi, alquil C1-4-carboniltio, alquilsulfinilo C1-4, haloalquilsulfinilo C1-4, alquilsulfonilo C1-4, haloalquilsulfonilo C1-4, NR4R5, NR4COR5, SF5, SO2NR4R5, alcoxialquilo C2-4 o 1-metoxiciclopropilo, Sustituyentes en el nitrógeno: alquilo C1-6, haloalquilo C1-3, cicloalquilo C3-6, halocicloalquilo C3-6, alquilcicloalquilo C4-10, alquenilo C2-6, haloalquenilo C2-6, alquinilo C2-6, haloalquinilo C2-6 o fenilo o R3 es un resto heterociclilo de 5 a 15 miembros unido a través de un átomo de carbono, no sustituido o monosustituido, que puede contener hasta dos heteroátomos adicionales, seleccionados de entre nitrógeno, oxígeno y azufre, seleccionándose el sustituyente de la lista siguiente: Sustituyentes en el carbono: ciano, halógeno, alquilo C1-6, haloalquilo C1-3, cicloalquilo C3-6, alquenilo C2-6, haloalquenilo C2-6, alquinilo C2-6, haloalquinilo C2-6, tri(alquil C1-2)sililo, fenilo, hidroxilo, alcoxi C1-6, haloalcoxi C1-6, alqueniloxi C2-6, alquiniloxi C2-6, alquiltio C1-6 o haloalquiltio C1-6, Sustituyentes en el nitrógeno: alquilo C1-6, haloalquilo C1-3, cicloalquilo C3-6, alquenilo C2-6, haloalquenilo C2-6, alquinilo C2-6, haloalquinilo C2-6, tri(alquil C1-2)sililo, o fenilo, R4, R5 representar, independientemente uno de otro, hidrógeno, alquilo C1-4, haloalquilo C1-3, cicloalquilo C3-6 o fenilo, R6 representa alquilo C1-4, haloalquilo C1-2, cicloalquilo C3-6 o fenilo; R7 representa hidrógeno, alquilo C1-4, haloalquilo C1-2, cicloalquilo C3-6 o fenilo, o en el caso de que L2 represente un grupo -CH=N-N(R7)- o -C(R6)=N-N(R7)-, los restos R7 y R3 forman conjuntamente con el átomo de nitrógeno a través del cual están unidos a través de L3 un heterociclo de 5 a 8 miembros, sustituido o no sustituido, saturado o parcialmente saturado o insaturado, que puede contener hasta dos heteroátomos adicionales seleccionados de entre N, O y S, no siendo adyacentes dos átomos de oxígeno, seleccionándose los posibles sustituyentes, independientemente uno de otro, de entre alquilo C1-4, alcoxi C1-4, hidroxilo o halógeno, y sus sales agroquímicamente activas.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP08171392 | 2008-12-11 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR074607A1 true AR074607A1 (es) | 2011-01-26 |
Family
ID=41664742
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP090104825A AR074607A1 (es) | 2008-12-11 | 2009-12-11 | Oximeteres e hidrazonas de tiazolilo como agentes fitoprotectores. |
Country Status (8)
| Country | Link |
|---|---|
| US (2) | US8697878B2 (es) |
| EP (1) | EP2376487B1 (es) |
| JP (1) | JP2012511525A (es) |
| CN (1) | CN102292334A (es) |
| AR (1) | AR074607A1 (es) |
| BR (1) | BRPI0923366A2 (es) |
| MX (1) | MX2011006042A (es) |
| WO (1) | WO2010066353A1 (es) |
Families Citing this family (27)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102292334A (zh) | 2008-12-11 | 2011-12-21 | 拜尔农作物科学股份公司 | 噻唑基肟醚和腙植物保护剂 |
| MX2012007200A (es) | 2009-12-21 | 2012-07-10 | Bayer Cropscience Ag | Bis(difluorometil)pirazoles como fungicidas. |
| WO2011134969A1 (de) | 2010-04-28 | 2011-11-03 | Bayer Cropscience Ag | Ketoheteroarylpiperidin und -piperazin derivate als fungizide |
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- 2009-11-28 EP EP09759910.4A patent/EP2376487B1/de not_active Not-in-force
- 2009-11-28 BR BRPI0923366A patent/BRPI0923366A2/pt not_active IP Right Cessation
- 2009-11-28 WO PCT/EP2009/008492 patent/WO2010066353A1/de not_active Ceased
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- 2009-11-28 MX MX2011006042A patent/MX2011006042A/es not_active Application Discontinuation
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| US8697878B2 (en) | 2014-04-15 |
| CN102292334A (zh) | 2011-12-21 |
| EP2376487B1 (de) | 2016-01-06 |
| US9215875B2 (en) | 2015-12-22 |
| US20100190828A1 (en) | 2010-07-29 |
| EP2376487A1 (de) | 2011-10-19 |
| JP2012511525A (ja) | 2012-05-24 |
| WO2010066353A1 (de) | 2010-06-17 |
| BRPI0923366A2 (pt) | 2019-09-24 |
| MX2011006042A (es) | 2011-07-04 |
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