NO20091970L - Krystallmodifikasjoner av 3-(1,H-indol-3-yl)-4-[2-(4-metyl-piperazin-1-yl)-quinazolin-4-yl]-pyrrol-2,5-dion - Google Patents
Krystallmodifikasjoner av 3-(1,H-indol-3-yl)-4-[2-(4-metyl-piperazin-1-yl)-quinazolin-4-yl]-pyrrol-2,5-dionInfo
- Publication number
- NO20091970L NO20091970L NO20091970A NO20091970A NO20091970L NO 20091970 L NO20091970 L NO 20091970L NO 20091970 A NO20091970 A NO 20091970A NO 20091970 A NO20091970 A NO 20091970A NO 20091970 L NO20091970 L NO 20091970L
- Authority
- NO
- Norway
- Prior art keywords
- quinazolin
- pyrrol
- piperazin
- indol
- dione
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Immunology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Epidemiology (AREA)
- Transplantation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US85338406P | 2006-10-20 | 2006-10-20 | |
| PCT/US2007/022241 WO2008051440A1 (fr) | 2006-10-20 | 2007-10-18 | Modifications cristallines |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NO20091970L true NO20091970L (no) | 2009-05-20 |
Family
ID=38921707
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20091970A NO20091970L (no) | 2006-10-20 | 2009-05-20 | Krystallmodifikasjoner av 3-(1,H-indol-3-yl)-4-[2-(4-metyl-piperazin-1-yl)-quinazolin-4-yl]-pyrrol-2,5-dion |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US8865897B2 (fr) |
| EP (1) | EP2102195A1 (fr) |
| JP (1) | JP5302199B2 (fr) |
| KR (1) | KR20090073231A (fr) |
| CN (2) | CN103265533A (fr) |
| AR (1) | AR063491A1 (fr) |
| AU (1) | AU2007309558B2 (fr) |
| BR (1) | BRPI0717461A2 (fr) |
| CA (1) | CA2666965A1 (fr) |
| CL (1) | CL2007003006A1 (fr) |
| EC (1) | ECSP099344A (fr) |
| IL (1) | IL197962A (fr) |
| MA (1) | MA30886B1 (fr) |
| MX (1) | MX2009004048A (fr) |
| MY (1) | MY158026A (fr) |
| NO (1) | NO20091970L (fr) |
| NZ (1) | NZ576241A (fr) |
| PE (1) | PE20081133A1 (fr) |
| RU (1) | RU2481341C2 (fr) |
| TN (1) | TN2009000147A1 (fr) |
| TW (1) | TWI399374B (fr) |
| WO (1) | WO2008051440A1 (fr) |
| ZA (1) | ZA200902048B (fr) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2010520879A (ja) * | 2007-03-09 | 2010-06-17 | ノバルティス アーゲー | 3−(1h−インドール−3−イル)−4−[2−(4−メチル−ピペラジン−1−イル)−キナゾリン−4−イル]−ピロール−2,5−ジオンの塩 |
| US9017528B2 (en) | 2011-04-14 | 2015-04-28 | Tel Nexx, Inc. | Electro chemical deposition and replenishment apparatus |
| US9005409B2 (en) | 2011-04-14 | 2015-04-14 | Tel Nexx, Inc. | Electro chemical deposition and replenishment apparatus |
| US9303329B2 (en) | 2013-11-11 | 2016-04-05 | Tel Nexx, Inc. | Electrochemical deposition apparatus with remote catholyte fluid management |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PE20020544A1 (es) * | 2000-11-07 | 2002-07-30 | Novartis Ag | Derivados de indolilmaleimida |
| GB0504203D0 (en) * | 2005-03-01 | 2005-04-06 | Novartis Ag | Organic compounds |
| MX2009013431A (es) | 2007-06-18 | 2010-01-15 | Sanofi Aventis | Derivados de pirrol como antagonistas de p2y12. |
-
2007
- 2007-10-18 PE PE2007001411A patent/PE20081133A1/es not_active Application Discontinuation
- 2007-10-18 BR BRPI0717461-6A2A patent/BRPI0717461A2/pt not_active IP Right Cessation
- 2007-10-18 CA CA002666965A patent/CA2666965A1/fr not_active Abandoned
- 2007-10-18 AU AU2007309558A patent/AU2007309558B2/en not_active Ceased
- 2007-10-18 MY MYPI20091403A patent/MY158026A/en unknown
- 2007-10-18 WO PCT/US2007/022241 patent/WO2008051440A1/fr not_active Ceased
- 2007-10-18 NZ NZ576241A patent/NZ576241A/en not_active IP Right Cessation
- 2007-10-18 CN CN2013101739586A patent/CN103265533A/zh active Pending
- 2007-10-18 EP EP07839661A patent/EP2102195A1/fr not_active Withdrawn
- 2007-10-18 CN CN2007800383914A patent/CN101522664B/zh not_active Expired - Fee Related
- 2007-10-18 KR KR1020097010201A patent/KR20090073231A/ko not_active Ceased
- 2007-10-18 JP JP2009533377A patent/JP5302199B2/ja not_active Expired - Fee Related
- 2007-10-18 AR ARP070104622A patent/AR063491A1/es unknown
- 2007-10-18 MX MX2009004048A patent/MX2009004048A/es active IP Right Grant
- 2007-10-18 US US12/445,371 patent/US8865897B2/en not_active Expired - Fee Related
- 2007-10-18 RU RU2009118816/04A patent/RU2481341C2/ru not_active IP Right Cessation
- 2007-10-19 CL CL200703006A patent/CL2007003006A1/es unknown
- 2007-10-19 TW TW096139386A patent/TWI399374B/zh not_active IP Right Cessation
-
2009
- 2009-03-24 ZA ZA200902048A patent/ZA200902048B/xx unknown
- 2009-04-05 IL IL197962A patent/IL197962A/en not_active IP Right Cessation
- 2009-04-17 TN TNP2009000147A patent/TN2009000147A1/fr unknown
- 2009-05-13 MA MA31867A patent/MA30886B1/fr unknown
- 2009-05-19 EC EC2009009344A patent/ECSP099344A/es unknown
- 2009-05-20 NO NO20091970A patent/NO20091970L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| CN101522664B (zh) | 2013-06-12 |
| CN101522664A (zh) | 2009-09-02 |
| CL2007003006A1 (es) | 2008-05-23 |
| US8865897B2 (en) | 2014-10-21 |
| AU2007309558B2 (en) | 2012-05-24 |
| JP2010506927A (ja) | 2010-03-04 |
| RU2009118816A (ru) | 2010-11-27 |
| BRPI0717461A2 (pt) | 2013-10-08 |
| CA2666965A1 (fr) | 2008-05-02 |
| TW200829572A (en) | 2008-07-16 |
| CN103265533A (zh) | 2013-08-28 |
| WO2008051440A1 (fr) | 2008-05-02 |
| AU2007309558A1 (en) | 2008-05-02 |
| KR20090073231A (ko) | 2009-07-02 |
| TN2009000147A1 (en) | 2010-10-18 |
| AR063491A1 (es) | 2009-01-28 |
| MY158026A (en) | 2016-08-30 |
| RU2481341C2 (ru) | 2013-05-10 |
| ECSP099344A (es) | 2009-06-30 |
| EP2102195A1 (fr) | 2009-09-23 |
| TWI399374B (zh) | 2013-06-21 |
| NZ576241A (en) | 2012-05-25 |
| PE20081133A1 (es) | 2008-09-16 |
| IL197962A (en) | 2013-08-29 |
| US20100041884A1 (en) | 2010-02-18 |
| IL197962A0 (en) | 2009-12-24 |
| ZA200902048B (en) | 2010-01-27 |
| MA30886B1 (fr) | 2009-11-02 |
| JP5302199B2 (ja) | 2013-10-02 |
| MX2009004048A (es) | 2009-04-27 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |