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NO20080740L - Heterocyklylamid-substituerte tiazoler, pyrroler og tiofener - Google Patents

Heterocyklylamid-substituerte tiazoler, pyrroler og tiofener

Info

Publication number
NO20080740L
NO20080740L NO20080740A NO20080740A NO20080740L NO 20080740 L NO20080740 L NO 20080740L NO 20080740 A NO20080740 A NO 20080740A NO 20080740 A NO20080740 A NO 20080740A NO 20080740 L NO20080740 L NO 20080740L
Authority
NO
Norway
Prior art keywords
heterocyclylamide
thiophenes
pyrroles
substituted thiazoles
prophylaxis
Prior art date
Application number
NO20080740A
Other languages
English (en)
Other versions
NO340507B1 (no
Inventor
Kerstin Henninger
Martin Radtke
Martin Hendrix
Holger Zimmermann
David Brueckner
Original Assignee
Aicuris Gmbh & Co Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aicuris Gmbh & Co Kg filed Critical Aicuris Gmbh & Co Kg
Publication of NO20080740L publication Critical patent/NO20080740L/no
Publication of NO340507B1 publication Critical patent/NO340507B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/20—Antivirals for DNA viruses
    • A61P31/22—Antivirals for DNA viruses for herpes viruses
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)

Abstract

Det beskrives heterocyklylamidsubstituerte tiazoler, pyrroler og tiofener og fremgangsmåter for fremstilling av disse. Videre beskrives anvendelsen for terapi og/eller profylakse av sykdommer samt deres anvendelse for fremstilling av legemidler for terapi og/eller profylakse av sykdommer, og særlig for anvendelse som antivirale midler, særlig mot cytomegalovira.
NO20080740A 2005-07-15 2008-02-11 Heterocyklylamidsubstituerte tiazoler, pyrroler og tiofener NO340507B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102005033103A DE102005033103A1 (de) 2005-07-15 2005-07-15 Heterocyclylamid-substituierte Thiazole, Pyrrole und Thiophene
PCT/EP2006/006434 WO2007009578A1 (de) 2005-07-15 2006-07-01 Heterocyclylamid-substituierte thiazole, pyrrole und thiophene

Publications (2)

Publication Number Publication Date
NO20080740L true NO20080740L (no) 2008-02-11
NO340507B1 NO340507B1 (no) 2017-05-02

Family

ID=37056618

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20080740A NO340507B1 (no) 2005-07-15 2008-02-11 Heterocyklylamidsubstituerte tiazoler, pyrroler og tiofener

Country Status (17)

Country Link
US (1) US8410090B2 (no)
EP (1) EP1910330B1 (no)
JP (1) JP5140582B2 (no)
KR (1) KR101352646B1 (no)
CN (1) CN101277946B (no)
AU (1) AU2006272059B2 (no)
BR (1) BRPI0615550A2 (no)
CA (1) CA2615049C (no)
DE (1) DE102005033103A1 (no)
ES (1) ES2518966T3 (no)
IL (1) IL188785A (no)
MX (1) MX2008000685A (no)
NO (1) NO340507B1 (no)
NZ (1) NZ564562A (no)
RU (1) RU2425829C2 (no)
WO (1) WO2007009578A1 (no)
ZA (1) ZA200801149B (no)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102011113749A1 (de) * 2011-09-14 2013-03-14 Aicuris Gmbh & Co. Kg Sulfonsäuresalze Heterocyclylamid-substituiertr Imidazole
IL252190B2 (en) * 2014-11-10 2024-04-01 Evrys Bio Llc Anti- human cytomegalovirus compounds and compositions

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2109934C (en) * 1991-07-03 2002-12-10 Donna Lee Romero Substituted indoles as anti-aids pharmaceuticals
US6080763A (en) 1997-11-03 2000-06-27 Boehringer Ingelheim Pharmaceuticals, Inc. Aromatic heterocyclic compounds and their use as anti-inflammatory agents
UA73492C2 (en) * 1999-01-19 2005-08-15 Aromatic heterocyclic compounds as antiinflammatory agents
WO2000053591A1 (de) 1999-03-08 2000-09-14 Bayer Aktiengesellschaft Thiazolylharnstoff-derivate und ihre verwendung als antivirale mittel
DE10131133A1 (de) 2001-06-28 2003-01-16 Bayer Ag Pyridazinone
WO2004002481A1 (en) * 2002-06-27 2004-01-08 Novo Nordisk A/S Aryl carbonyl derivatives as therapeutic agents
DE10257358A1 (de) 2002-12-09 2004-07-08 Bayer Healthcare Ag Substituierte Pyrrole
KR100574547B1 (ko) 2003-03-21 2006-04-27 율촌화학 주식회사 내수성이 개선된 생분해성 조성물 및 그 제조방법
AU2005287692B2 (en) * 2004-09-20 2012-07-12 4Sc Ag Novel heterocyclic NF-kappaB inhibitors
EP1637529A1 (en) * 2004-09-20 2006-03-22 4Sc Ag Novel piperidin-4-yl-thiazole-carboxamide analogues as inhibitors of T-cell proliferation and uses thereof

Also Published As

Publication number Publication date
DE102005033103A1 (de) 2007-01-25
RU2425829C2 (ru) 2011-08-10
AU2006272059B2 (en) 2012-05-17
CN101277946A (zh) 2008-10-01
US20100144752A1 (en) 2010-06-10
US8410090B2 (en) 2013-04-02
EP1910330A1 (de) 2008-04-16
CN101277946B (zh) 2013-01-02
IL188785A0 (en) 2008-11-03
KR20080091074A (ko) 2008-10-09
IL188785A (en) 2012-08-30
CA2615049A1 (en) 2007-01-25
EP1910330B1 (de) 2014-07-23
ZA200801149B (en) 2009-07-29
KR101352646B1 (ko) 2014-01-16
BRPI0615550A2 (pt) 2011-05-24
AU2006272059A1 (en) 2007-01-25
CA2615049C (en) 2013-12-03
RU2008105353A (ru) 2009-08-20
JP5140582B2 (ja) 2013-02-06
JP2009501170A (ja) 2009-01-15
HK1115385A1 (en) 2008-11-28
NZ564562A (en) 2010-12-24
MX2008000685A (es) 2008-03-18
WO2007009578A1 (de) 2007-01-25
ES2518966T3 (es) 2014-11-06
NO340507B1 (no) 2017-05-02

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