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NO20076357L - Azabicykliske heterocykler som cannabinoid reseptor modulatorer - Google Patents

Azabicykliske heterocykler som cannabinoid reseptor modulatorer

Info

Publication number
NO20076357L
NO20076357L NO20076357A NO20076357A NO20076357L NO 20076357 L NO20076357 L NO 20076357L NO 20076357 A NO20076357 A NO 20076357A NO 20076357 A NO20076357 A NO 20076357A NO 20076357 L NO20076357 L NO 20076357L
Authority
NO
Norway
Prior art keywords
formula
receptor modulators
cannabinoid receptor
compounds
azabicyclic
Prior art date
Application number
NO20076357A
Other languages
English (en)
Inventor
William R Ewing
Bruce A Ellsworth
Yeheng Zhu
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of NO20076357L publication Critical patent/NO20076357L/no

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P17/06—Antipsoriatics
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P9/12—Antihypertensives

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Life Sciences & Earth Sciences (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
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  • Hematology (AREA)
  • Obesity (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
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  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Anesthesiology (AREA)
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  • Hospice & Palliative Care (AREA)
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Abstract

Foreliggende søknad beskriver forbindelser med formel I, farmasøytiske preparater omfattende minst én forbindelse med formel I og eventuelt én eller flere ytterligere terapeutiske midler og metoder for behandling ved anvendelse av forbindelsene i henhold til Formel I både alene og i kombinasjon med én eller flere ytterligere terapeutiske midler. Forbindelsene har den generelle Formel I og Formel II: omfattende alle prodroger, farmasøytisk akseptable salter og stereoisomerer, R1, R2, R3 og R4 er beskrevet her.
NO20076357A 2005-06-17 2007-12-12 Azabicykliske heterocykler som cannabinoid reseptor modulatorer NO20076357L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US69203405P 2005-06-17 2005-06-17
US11/454,324 US7629342B2 (en) 2005-06-17 2006-06-16 Azabicyclic heterocycles as cannabinoid receptor modulators
PCT/US2006/023683 WO2006138682A1 (en) 2005-06-17 2006-06-19 Azabicyclic heterocycles as cannabinoid receptor modulators

Publications (1)

Publication Number Publication Date
NO20076357L true NO20076357L (no) 2008-03-14

Family

ID=37012092

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20076357A NO20076357L (no) 2005-06-17 2007-12-12 Azabicykliske heterocykler som cannabinoid reseptor modulatorer

Country Status (5)

Country Link
US (1) US7629342B2 (no)
EP (1) EP1891074B1 (no)
JP (1) JP2008543875A (no)
NO (1) NO20076357L (no)
WO (1) WO2006138682A1 (no)

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