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NO20071230L - Oksazolidinoner inneholdende oksindoler som antibakterielle midler - Google Patents

Oksazolidinoner inneholdende oksindoler som antibakterielle midler

Info

Publication number
NO20071230L
NO20071230L NO20071230A NO20071230A NO20071230L NO 20071230 L NO20071230 L NO 20071230L NO 20071230 A NO20071230 A NO 20071230A NO 20071230 A NO20071230 A NO 20071230A NO 20071230 L NO20071230 L NO 20071230L
Authority
NO
Norway
Prior art keywords
oxindoles
antibacterial agents
oxazolidinones containing
oxazolidinones
cycloalkyl
Prior art date
Application number
NO20071230A
Other languages
English (en)
Inventor
Mikhail Fedorovich Gordeev
Gary Wayne Luehr
Rama Jain
Adam Robert Renslo
Vara Prasad Venkata Na Josyula
Original Assignee
Pharmacia & Upjohn Co Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35079333&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20071230(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacia & Upjohn Co Llc filed Critical Pharmacia & Upjohn Co Llc
Publication of NO20071230L publication Critical patent/NO20071230L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Foreliggende oppfinnelsen angår nye oksazolidinonderivater av oksindoler med formel I, eller et farmasøytisk akseptabelt salt derav, hvori Y1 er -CH- eller -CF-; R1 er -C1-4 alkyl, eventuelt substituert med et fluoroatom, eller R1 er -C3-5 cykloalkyl; og R2 er -H eller -CH3. Disse forbindelsene er anvendelige som antibakterielle midler.
NO20071230A 2004-08-06 2007-03-06 Oksazolidinoner inneholdende oksindoler som antibakterielle midler NO20071230L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US59982204P 2004-08-06 2004-08-06
PCT/IB2005/002197 WO2006016221A1 (en) 2004-08-06 2005-07-19 Oxazolidinones containing oxindoles as antibacterial agents

Publications (1)

Publication Number Publication Date
NO20071230L true NO20071230L (no) 2007-05-04

Family

ID=35079333

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20071230A NO20071230L (no) 2004-08-06 2007-03-06 Oksazolidinoner inneholdende oksindoler som antibakterielle midler

Country Status (24)

Country Link
US (2) US20080262056A1 (no)
EP (2) EP1781642A1 (no)
JP (2) JP2008509125A (no)
CN (1) CN101001853A (no)
AP (1) AP2007003904A0 (no)
AR (1) AR050101A1 (no)
AU (1) AU2005270951A1 (no)
BR (2) BRPI0513083A (no)
CA (2) CA2575702A1 (no)
EA (1) EA200700322A1 (no)
GT (1) GT200500204A (no)
IL (1) IL180957A0 (no)
MA (1) MA28793B1 (no)
MX (2) MX2007001568A (no)
NL (1) NL1029686C2 (no)
NO (1) NO20071230L (no)
PA (1) PA8640901A1 (no)
PE (1) PE20060351A1 (no)
SV (1) SV2006002180A (no)
TN (1) TNSN07043A1 (no)
TW (1) TWI289448B (no)
UY (1) UY29048A1 (no)
WO (2) WO2006016221A1 (no)
ZA (1) ZA200700476B (no)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2603943A1 (en) * 2005-04-06 2006-10-12 Pharmacia & Upjohn Company Llc An oxindole oxazolidinone as antibacterial agent
AU2006231919A1 (en) 2005-04-06 2006-10-12 Pharmacia & Upjohn Company Llc 7-fluoro-1,3-dihydro-indol-2-one oxazolidinones as antibacterial agents
CN103483329B (zh) * 2013-09-07 2015-08-05 吉首大学 呋喃酮-芳基-噁唑烷酮型化合物及其制法和用途
CN103420995B (zh) * 2013-09-07 2015-07-01 吉首大学 噁唑烷酮-烷胺基-呋喃酮型化合物及其制法和用途
CN107698567B (zh) * 2017-10-25 2020-09-15 西南大学 靛红唑醇类化合物及其制备方法和医药应用

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5164510A (en) * 1988-09-15 1992-11-17 The Upjohn Company 5'Indolinyl-5β-amidomethyloxazolidin-2-ones
EP0609905B1 (en) * 1988-09-15 2001-06-06 PHARMACIA & UPJOHN COMPANY 3-(Nitrogen substituted)phenyl-5beta-amidomethyloxazolidin-2-ones
DE4425612A1 (de) * 1994-07-20 1996-04-04 Bayer Ag 6-gliedrige stickstoffhaltige Heteroaryl-oxazolidinone
ATE233766T1 (de) * 1994-11-15 2003-03-15 Upjohn Co Antibakterielle bizyklische oxazin und thiazin- oxazolidinone
HRP960159A2 (en) * 1995-04-21 1997-08-31 Bayer Ag Benzocyclopentane oxazolidinones containing heteroatoms
CA2228647A1 (en) * 1995-09-01 1997-03-13 Pharmacia & Upjohn Company Phenyloxazolidinones having a c-c bond to 4-8 membered heterocyclic rings
DE19601265A1 (de) * 1996-01-16 1997-07-17 Bayer Ag 2-Oxo- und 2-Thio-1,2-dihydrochinolinyl-oxazolidinone
DE19601627A1 (de) * 1996-01-18 1997-07-24 Bayer Ag Heteroatomhaltige Cyclopentanopyridyl-Oxazolidinone
GB9601666D0 (en) * 1996-01-27 1996-03-27 Zeneca Ltd Chemical compounds
GB9702213D0 (en) * 1996-02-24 1997-03-26 Zeneca Ltd Chemical compounds
GB9609919D0 (en) * 1996-05-11 1996-07-17 Zeneca Ltd Chemical compounds
ES2186916T3 (es) * 1996-08-21 2003-05-16 Upjohn Co Derivados de isoxazolina como agentes antimicrobianos.
GB9717804D0 (en) * 1997-08-22 1997-10-29 Zeneca Ltd Chemical compounds
EP1049682A1 (en) * 1998-01-23 2000-11-08 Versicor, Inc. Oxazolidinone combinatorial libraries, compositions and methods of preparation
GB9812019D0 (en) * 1998-06-05 1998-07-29 Zeneca Ltd Chemical compounds
AU767579B2 (en) * 1999-02-01 2003-11-20 Pharmacia & Upjohn Company Process to prepare cyclic-sulfur fluorine containing oxazolidinones
BR0010982A (pt) * 1999-05-27 2002-03-05 Upjohn Co Novas oxazolidinonas bicìclicas como agentes antibacterianos
AR038536A1 (es) * 2002-02-25 2005-01-19 Upjohn Co N-aril-2-oxazolidinona-5- carboxamidas y sus derivados
US7012088B2 (en) * 2003-02-24 2006-03-14 Pharmacia & Upjohn Company Indolone oxazolidinones and derivatives thereof
AU2006231919A1 (en) * 2005-04-06 2006-10-12 Pharmacia & Upjohn Company Llc 7-fluoro-1,3-dihydro-indol-2-one oxazolidinones as antibacterial agents

Also Published As

Publication number Publication date
WO2006016221A1 (en) 2006-02-16
EP1781643A1 (en) 2007-05-09
EA200700322A1 (ru) 2007-08-31
BRPI0513083A (pt) 2008-04-22
AP2007003904A0 (en) 2007-02-28
AU2005270951A1 (en) 2006-02-16
CA2576041A1 (en) 2006-02-16
JP2008509126A (ja) 2008-03-27
US20060030609A1 (en) 2006-02-09
CN101001853A (zh) 2007-07-18
PA8640901A1 (es) 2007-01-17
CA2575702A1 (en) 2006-02-16
NL1029686C2 (nl) 2006-07-18
EP1781642A1 (en) 2007-05-09
US20080262056A1 (en) 2008-10-23
TWI289448B (en) 2007-11-11
JP2008509125A (ja) 2008-03-27
MX2007001568A (es) 2007-04-16
MA28793B1 (fr) 2007-08-01
TW200612924A (en) 2006-05-01
SV2006002180A (es) 2006-06-26
NL1029686A1 (nl) 2006-02-07
GT200500204A (es) 2006-03-02
PE20060351A1 (es) 2006-05-03
UY29048A1 (es) 2006-03-31
IL180957A0 (en) 2007-07-04
TNSN07043A1 (fr) 2008-06-02
MX2007001526A (es) 2007-03-27
BRPI0514020A (pt) 2008-05-27
WO2006016220A1 (en) 2006-02-16
AR050101A1 (es) 2006-09-27
ZA200700476B (en) 2008-10-29

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