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NO20061701L - Tiazolderivater som cannabionoide reseptor modulatorer - Google Patents

Tiazolderivater som cannabionoide reseptor modulatorer

Info

Publication number
NO20061701L
NO20061701L NO20061701A NO20061701A NO20061701L NO 20061701 L NO20061701 L NO 20061701L NO 20061701 A NO20061701 A NO 20061701A NO 20061701 A NO20061701 A NO 20061701A NO 20061701 L NO20061701 L NO 20061701L
Authority
NO
Norway
Prior art keywords
thiazole derivatives
receptor
compounds
cannabionoid
receptor modulators
Prior art date
Application number
NO20061701A
Other languages
English (en)
Inventor
Herman Heinrich Va Stuivenberg
Cornelis Gerrit Kruse
Josephus H M Lange
Leonardus A J M Sliedregt
Original Assignee
Solvay Pharm Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Solvay Pharm Bv filed Critical Solvay Pharm Bv
Publication of NO20061701L publication Critical patent/NO20061701L/no

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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

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Abstract

Gruppe av tiazolderivater, fremgangsmåter for fremstilling av disse forbindelsene, farmasøytiske preparater som inneholder minst en av disse forbindelsene som aktiv bestanddel, samt anvendelsen av disse preparatene for behandling av psykiatriske og neurologiske forstyrrelser og andre sykdommer som involverer cannabinoid CB neurotransmisjon. Tiazolderivatene ifølge oppfinnelsen er enten cannabinoid (CB) reseptor antagonister, CB reseptor agonister, CB reseptor inverse agonister eller CB reseptor partial agonister.Forbindelsene har den generelle formel (I). hvor R, Ri og X har de betydninger som er angitt heri.
NO20061701A 2003-09-19 2006-04-18 Tiazolderivater som cannabionoide reseptor modulatorer NO20061701L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP03078309 2003-09-19
PCT/EP2004/052239 WO2005028456A1 (en) 2003-09-19 2004-09-20 Thiazole derivatives as cannabinoid receptor modulators

Publications (1)

Publication Number Publication Date
NO20061701L true NO20061701L (no) 2006-06-16

Family

ID=34923999

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20061701A NO20061701L (no) 2003-09-19 2006-04-18 Tiazolderivater som cannabionoide reseptor modulatorer

Country Status (17)

Country Link
US (1) US20050065189A1 (no)
EP (1) EP1664005B1 (no)
JP (1) JP2007533621A (no)
CN (1) CN100475796C (no)
AR (1) AR045651A1 (no)
AT (1) ATE497953T1 (no)
AU (1) AU2004274184B2 (no)
BR (1) BRPI0414514A (no)
CA (1) CA2534798A1 (no)
MX (1) MXPA06002061A (no)
NO (1) NO20061701L (no)
RU (1) RU2348620C2 (no)
SA (1) SA04250288B1 (no)
TW (1) TWI336697B (no)
UA (1) UA83862C2 (no)
WO (1) WO2005028456A1 (no)
ZA (1) ZA200603087B (no)

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