NO20053396L - Acykliske pyrazolforbindelser for inhibering av mitogenaktivert proteinkinase aktivert protein kinase 2. - Google Patents
Acykliske pyrazolforbindelser for inhibering av mitogenaktivert proteinkinase aktivert protein kinase 2.Info
- Publication number
- NO20053396L NO20053396L NO20053396A NO20053396A NO20053396L NO 20053396 L NO20053396 L NO 20053396L NO 20053396 A NO20053396 A NO 20053396A NO 20053396 A NO20053396 A NO 20053396A NO 20053396 L NO20053396 L NO 20053396L
- Authority
- NO
- Norway
- Prior art keywords
- protein kinase
- activated protein
- mitogen
- inhibition
- compounds
- Prior art date
Links
- 102100034069 MAP kinase-activated protein kinase 2 Human genes 0.000 title abstract 5
- 101710141394 MAP kinase-activated protein kinase 2 Proteins 0.000 title abstract 5
- -1 Acyclic pyrazole compounds Chemical class 0.000 title 1
- 230000005764 inhibitory process Effects 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 4
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 230000002401 inhibitory effect Effects 0.000 abstract 2
- 108060008682 Tumor Necrosis Factor Proteins 0.000 abstract 1
- 102000000852 Tumor Necrosis Factor-alpha Human genes 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000035475 disorder Diseases 0.000 abstract 1
- 230000001404 mediated effect Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US43496202P | 2002-12-20 | 2002-12-20 | |
| PCT/US2003/040932 WO2004058176A2 (fr) | 2002-12-20 | 2003-12-19 | Composes de pyrazole acyclique pour l'inhibition d'une proteine kinase activee par mitogene / d'une proteine kinase 2 activee |
Publications (2)
| Publication Number | Publication Date |
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| NO20053396D0 NO20053396D0 (no) | 2005-07-13 |
| NO20053396L true NO20053396L (no) | 2005-09-12 |
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| NO20053396A NO20053396L (no) | 2002-12-20 | 2005-07-13 | Acykliske pyrazolforbindelser for inhibering av mitogenaktivert proteinkinase aktivert protein kinase 2. |
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| Country | Link |
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| US (3) | US20040209897A1 (fr) |
| EP (2) | EP1572682A4 (fr) |
| JP (2) | JP2006514043A (fr) |
| KR (1) | KR20050104339A (fr) |
| CN (1) | CN1747949A (fr) |
| AU (2) | AU2003301226A1 (fr) |
| BR (2) | BR0317525A (fr) |
| CA (2) | CA2510298A1 (fr) |
| IL (1) | IL169177A0 (fr) |
| MX (2) | MXPA05006569A (fr) |
| NO (1) | NO20053396L (fr) |
| PL (1) | PL377461A1 (fr) |
| RU (1) | RU2005119173A (fr) |
| WO (2) | WO2004058176A2 (fr) |
| ZA (1) | ZA200504898B (fr) |
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-
2003
- 2003-12-19 WO PCT/US2003/040932 patent/WO2004058176A2/fr not_active Ceased
- 2003-12-19 EP EP03814309A patent/EP1572682A4/fr not_active Withdrawn
- 2003-12-19 JP JP2004563888A patent/JP2006514043A/ja not_active Withdrawn
- 2003-12-19 AU AU2003301226A patent/AU2003301226A1/en not_active Withdrawn
- 2003-12-19 BR BR0317525-1A patent/BR0317525A/pt not_active IP Right Cessation
- 2003-12-19 BR BR0317430-1A patent/BR0317430A/pt not_active Application Discontinuation
- 2003-12-19 CN CNA2003801096266A patent/CN1747949A/zh active Pending
- 2003-12-19 US US10/742,072 patent/US20040209897A1/en not_active Abandoned
- 2003-12-19 RU RU2005119173/04A patent/RU2005119173A/ru not_active Application Discontinuation
- 2003-12-19 EP EP03814268A patent/EP1572693A1/fr not_active Withdrawn
- 2003-12-19 US US10/742,494 patent/US20040152739A1/en not_active Abandoned
- 2003-12-19 MX MXPA05006569A patent/MXPA05006569A/es unknown
- 2003-12-19 AU AU2003297431A patent/AU2003297431A1/en not_active Abandoned
- 2003-12-19 ZA ZA200504898A patent/ZA200504898B/en unknown
- 2003-12-19 KR KR1020057011474A patent/KR20050104339A/ko not_active Withdrawn
- 2003-12-19 MX MXPA05006568A patent/MXPA05006568A/es not_active Application Discontinuation
- 2003-12-19 JP JP2004563946A patent/JP2006511583A/ja not_active Withdrawn
- 2003-12-19 CA CA002510298A patent/CA2510298A1/fr not_active Abandoned
- 2003-12-19 CA CA002509565A patent/CA2509565A1/fr not_active Abandoned
- 2003-12-19 WO PCT/US2003/040811 patent/WO2004058762A1/fr not_active Ceased
- 2003-12-19 PL PL377461A patent/PL377461A1/pl unknown
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2005
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- 2005-07-13 NO NO20053396A patent/NO20053396L/no not_active Application Discontinuation
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2007
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| Publication number | Publication date |
|---|---|
| JP2006511583A (ja) | 2006-04-06 |
| PL377461A1 (pl) | 2006-02-06 |
| MXPA05006569A (es) | 2005-09-22 |
| EP1572693A1 (fr) | 2005-09-14 |
| EP1572682A2 (fr) | 2005-09-14 |
| AU2003297431A1 (en) | 2004-07-22 |
| WO2004058176A2 (fr) | 2004-07-15 |
| NO20053396D0 (no) | 2005-07-13 |
| MXPA05006568A (es) | 2005-09-22 |
| AU2003301226A1 (en) | 2004-07-22 |
| US20080113971A1 (en) | 2008-05-15 |
| ZA200504898B (en) | 2006-11-29 |
| US20040152739A1 (en) | 2004-08-05 |
| RU2005119173A (ru) | 2006-02-27 |
| WO2004058176A3 (fr) | 2004-09-16 |
| BR0317430A (pt) | 2005-10-25 |
| BR0317525A (pt) | 2005-11-16 |
| IL169177A0 (en) | 2007-07-04 |
| KR20050104339A (ko) | 2005-11-02 |
| JP2006514043A (ja) | 2006-04-27 |
| EP1572682A4 (fr) | 2008-01-23 |
| CA2509565A1 (fr) | 2004-07-15 |
| CN1747949A (zh) | 2006-03-15 |
| WO2004058762A1 (fr) | 2004-07-15 |
| CA2510298A1 (fr) | 2004-07-15 |
| US20040209897A1 (en) | 2004-10-21 |
| AU2003301226A2 (en) | 2004-07-22 |
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