NO20051187L - Depotformuleringer bestaende av aktive arylheterocykliske forbindelser i form av en suspensjon - Google Patents
Depotformuleringer bestaende av aktive arylheterocykliske forbindelser i form av en suspensjonInfo
- Publication number
- NO20051187L NO20051187L NO20051187A NO20051187A NO20051187L NO 20051187 L NO20051187 L NO 20051187L NO 20051187 A NO20051187 A NO 20051187A NO 20051187 A NO20051187 A NO 20051187A NO 20051187 L NO20051187 L NO 20051187L
- Authority
- NO
- Norway
- Prior art keywords
- depositional
- suspension
- active
- formulations consisting
- arylheterocyclic
- Prior art date
Links
- 238000009472 formulation Methods 0.000 title abstract 3
- 239000000203 mixture Substances 0.000 title abstract 3
- 150000001875 compounds Chemical class 0.000 title abstract 2
- 239000000725 suspension Substances 0.000 title 1
- 238000000034 method Methods 0.000 abstract 1
- MVWVFYHBGMAFLY-UHFFFAOYSA-N ziprasidone Chemical compound C1=CC=C2C(N3CCN(CC3)CCC3=CC=4CC(=O)NC=4C=C3Cl)=NSC2=C1 MVWVFYHBGMAFLY-UHFFFAOYSA-N 0.000 abstract 1
- 229960000607 ziprasidone Drugs 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/40—Cyclodextrins; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Inorganic Chemistry (AREA)
- Dermatology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurosurgery (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Dispersion Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
Farmasøytisk sett for fremstilling av en injiserbar depotformulering av en aryl-heterocyklisk farmasøytiske forbindelse, så som ziprasidon og en metode for fremstilling av nevnte depotformulering er beskrevet.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US42129502P | 2002-10-25 | 2002-10-25 | |
| PCT/IB2003/004535 WO2004037224A1 (en) | 2002-10-25 | 2003-10-13 | Depot formulations of arylheterocyclic active agents in the form of a suspension |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NO20051187L true NO20051187L (no) | 2005-04-11 |
Family
ID=32176696
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20051187A NO20051187L (no) | 2002-10-25 | 2005-03-04 | Depotformuleringer bestaende av aktive arylheterocykliske forbindelser i form av en suspensjon |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US20040146562A1 (no) |
| EP (1) | EP1562546A1 (no) |
| JP (2) | JP2006505579A (no) |
| KR (1) | KR20050071611A (no) |
| CN (1) | CN1703198A (no) |
| AR (1) | AR041826A1 (no) |
| AU (1) | AU2003267763A1 (no) |
| BR (1) | BR0315663A (no) |
| CA (1) | CA2498276A1 (no) |
| GT (1) | GT200300227A (no) |
| MX (1) | MXPA05004299A (no) |
| NL (1) | NL1024616C (no) |
| NO (1) | NO20051187L (no) |
| PA (1) | PA8586301A1 (no) |
| PE (1) | PE20040471A1 (no) |
| PL (1) | PL375603A1 (no) |
| RU (1) | RU2292207C2 (no) |
| TW (1) | TW200418477A (no) |
| UY (1) | UY28035A1 (no) |
| WO (1) | WO2004037224A1 (no) |
| ZA (1) | ZA200501979B (no) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20080113025A1 (en) * | 1998-11-02 | 2008-05-15 | Elan Pharma International Limited | Compositions comprising nanoparticulate naproxen and controlled release hydrocodone |
| US20040001889A1 (en) | 2002-06-25 | 2004-01-01 | Guohua Chen | Short duration depot formulations |
| DE60327225D1 (de) * | 2002-08-20 | 2009-05-28 | Bristol Myers Squibb Co | Aripiprazol-komplex-formulierung und verfahren |
| CA2507522C (en) | 2002-12-13 | 2015-02-24 | Durect Corporation | Oral drug delivery system |
| JP2007522095A (ja) * | 2003-05-16 | 2007-08-09 | ファイザー・プロダクツ・インク | ジプラシドンを用いた不安の治療 |
| WO2006000913A1 (en) * | 2004-06-23 | 2006-01-05 | Pfizer Products Inc. | Method for sterile filtration of viscous pharmaceutical compositions |
| EP2767292B1 (en) * | 2004-09-17 | 2016-08-24 | Durect Corporation | Sustained Local Anesthetic Composition Containing SAIB |
| JP2008531721A (ja) * | 2005-03-03 | 2008-08-14 | エラン・ファルマ・インターナショナル・リミテッド | 複素環式アミド誘導体のナノ粒子状組成物 |
| US20070027105A1 (en) | 2005-07-26 | 2007-02-01 | Alza Corporation | Peroxide removal from drug delivery vehicle |
| CN100391458C (zh) * | 2006-02-07 | 2008-06-04 | 上海医药工业研究院 | 齐拉西酮或其盐包合物制备方法 |
| JP2009536195A (ja) * | 2006-05-09 | 2009-10-08 | アストラゼネカ・アクチエボラーグ | 最終容器中で電離放射線により滅菌されるプロトンポンプ阻害剤を含む非経口製剤 |
| AU2007325918B2 (en) | 2006-11-03 | 2013-10-17 | Durect Corporation | Transdermal delivery systems comprising bupivacaine |
| EP2219622A1 (en) * | 2007-12-06 | 2010-08-25 | Durect Corporation | Methods useful for the treatment of pain, arthritic conditions, or inflammation associated with a chronic condition |
| US20100260844A1 (en) | 2008-11-03 | 2010-10-14 | Scicinski Jan J | Oral pharmaceutical dosage forms |
| US9555113B2 (en) | 2013-03-15 | 2017-01-31 | Durect Corporation | Compositions with a rheological modifier to reduce dissolution variability |
| SG11201811760VA (en) | 2016-07-06 | 2019-01-30 | Durect Corp | Oral dosage form with drug composition, barrier layer and drug layer |
| WO2018153315A1 (zh) | 2017-02-23 | 2018-08-30 | 上海华汇拓医药科技有限公司 | 一种多奈哌齐半帕莫酸盐的粉针剂、包含其的组合物及它们的制备方法 |
| KR20220140711A (ko) | 2020-01-13 | 2022-10-18 | 듀렉트 코퍼레이션 | 불순물이 감소된 지속 방출 약물 전달 시스템 및 관련 방법 |
| EP4277702A1 (en) | 2021-01-12 | 2023-11-22 | Durect Corporation | Sustained release drug delivery systems and related methods |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0331755B2 (en) * | 1987-09-07 | 2003-02-05 | Teijin Limited | Medicine-containing fat emulsion of the type prepared immediately before use and process for preparing medicine-containing fat emulsion |
| GB9200247D0 (en) * | 1992-01-07 | 1992-02-26 | Erba Carlo Spa | Pharmaceutical compositions containing polymer derivative-bound anthracycline glycosides and a method for their preparation |
| JP3954115B2 (ja) * | 1992-07-28 | 2007-08-08 | アストラゼネカ・アクチエボラーグ | 注射剤および注射剤キット |
| US5594141A (en) * | 1994-11-23 | 1997-01-14 | Neurogen Corporation | Certain aminomethyl biphenyl, aminomethyl phenyl pyridine and aminomethyl phenyl pyrimidine derivatives; novel dopamine receptor subtype selective ligands |
| US6040295A (en) * | 1995-01-13 | 2000-03-21 | Genemedicine, Inc. | Formulated nucleic acid compositions and methods of administering the same for gene therapy |
| UA57734C2 (uk) * | 1996-05-07 | 2003-07-15 | Пфайзер Інк. | Комплекси включення арилгетероциклічних солей |
| ATE277641T1 (de) * | 1996-05-07 | 2004-10-15 | Pfizer | Verfahren zur selektion eines salzes zur herstellung eines inklusionskomplexes |
| US6130200A (en) * | 1996-12-20 | 2000-10-10 | Alza Corporation | Gel composition and methods |
| EA199901013A1 (ru) * | 1997-05-16 | 2000-06-26 | Амген Инк. | Гели пролонгированного действия |
| UA72189C2 (uk) * | 1997-11-17 | 2005-02-15 | Янссен Фармацевтика Н.В. | Фармацевтична композиція, що містить водну суспензію субмікронних ефірів 9-гідроксирисперидон жирних кислот |
| SI1181018T1 (en) * | 1999-05-27 | 2003-06-30 | Pfizer Products Inc. | Ziprasidone suspension |
| MY137726A (en) * | 2000-11-22 | 2009-03-31 | Nycomed Gmbh | Freeze-dried pantoprazole preparation and pantoprazole injection |
| AU2002254309B2 (en) * | 2001-03-20 | 2006-02-02 | Cydex, Inc. | Formulations containing propofol and a sulfoalkyl ether cyclodextrin |
| EP1269994A3 (en) * | 2001-06-22 | 2003-02-12 | Pfizer Products Inc. | Pharmaceutical compositions comprising drug and concentration-enhancing polymers |
| CA2458968A1 (en) * | 2001-08-31 | 2003-03-13 | The Rockefeller University | Method for classification of anti-psychotic drugs |
-
2003
- 2003-10-13 PL PL03375603A patent/PL375603A1/xx not_active Application Discontinuation
- 2003-10-13 BR BR0315663-0A patent/BR0315663A/pt not_active IP Right Cessation
- 2003-10-13 KR KR1020057006963A patent/KR20050071611A/ko not_active Ceased
- 2003-10-13 CA CA002498276A patent/CA2498276A1/en not_active Abandoned
- 2003-10-13 RU RU2005112202/15A patent/RU2292207C2/ru not_active IP Right Cessation
- 2003-10-13 AU AU2003267763A patent/AU2003267763A1/en not_active Abandoned
- 2003-10-13 MX MXPA05004299A patent/MXPA05004299A/es unknown
- 2003-10-13 CN CNA2003801011573A patent/CN1703198A/zh active Pending
- 2003-10-13 EP EP03748458A patent/EP1562546A1/en not_active Withdrawn
- 2003-10-13 WO PCT/IB2003/004535 patent/WO2004037224A1/en not_active Ceased
- 2003-10-13 JP JP2004546259A patent/JP2006505579A/ja active Pending
- 2003-10-14 PA PA20038586301A patent/PA8586301A1/es unknown
- 2003-10-21 US US10/689,778 patent/US20040146562A1/en not_active Abandoned
- 2003-10-21 GT GT200300227A patent/GT200300227A/es unknown
- 2003-10-21 PE PE2003001065A patent/PE20040471A1/es not_active Application Discontinuation
- 2003-10-22 UY UY28035A patent/UY28035A1/es not_active Application Discontinuation
- 2003-10-23 AR ARP030103869A patent/AR041826A1/es unknown
- 2003-10-24 NL NL1024616A patent/NL1024616C/nl not_active IP Right Cessation
- 2003-10-24 TW TW092129567A patent/TW200418477A/zh unknown
-
2005
- 2005-03-04 NO NO20051187A patent/NO20051187L/no not_active Application Discontinuation
- 2005-04-08 ZA ZA200501979A patent/ZA200501979B/en unknown
-
2006
- 2006-05-23 JP JP2006142886A patent/JP2006219501A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| GT200300227A (es) | 2004-06-23 |
| NL1024616C (nl) | 2010-04-19 |
| AR041826A1 (es) | 2005-06-01 |
| PA8586301A1 (es) | 2004-05-07 |
| RU2005112202A (ru) | 2005-11-20 |
| PE20040471A1 (es) | 2004-08-14 |
| CA2498276A1 (en) | 2004-05-06 |
| NL1024616A1 (nl) | 2004-04-27 |
| AU2003267763A1 (en) | 2004-05-13 |
| PL375603A1 (en) | 2005-12-12 |
| US20040146562A1 (en) | 2004-07-29 |
| TW200418477A (en) | 2004-10-01 |
| JP2006505579A (ja) | 2006-02-16 |
| WO2004037224A1 (en) | 2004-05-06 |
| JP2006219501A (ja) | 2006-08-24 |
| CN1703198A (zh) | 2005-11-30 |
| EP1562546A1 (en) | 2005-08-17 |
| UY28035A1 (es) | 2004-05-31 |
| MXPA05004299A (es) | 2005-08-03 |
| BR0315663A (pt) | 2005-08-30 |
| KR20050071611A (ko) | 2005-07-07 |
| ZA200501979B (en) | 2006-04-26 |
| RU2292207C2 (ru) | 2007-01-27 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |