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NO20043370L - N-pyrazinylfenylsulfonamider og deres anvendelse ved behandling av kemokinmedierte sykdommer - Google Patents

N-pyrazinylfenylsulfonamider og deres anvendelse ved behandling av kemokinmedierte sykdommer

Info

Publication number
NO20043370L
NO20043370L NO20043370A NO20043370A NO20043370L NO 20043370 L NO20043370 L NO 20043370L NO 20043370 A NO20043370 A NO 20043370A NO 20043370 A NO20043370 A NO 20043370A NO 20043370 L NO20043370 L NO 20043370L
Authority
NO
Norway
Prior art keywords
pyrazinylphenylsulfonamides
chemokine
treatment
mediated diseases
mediated
Prior art date
Application number
NO20043370A
Other languages
English (en)
Inventor
Michael Stocks
Nicholas Kindon
Bryan Roberts
Andrew Baxter
Timothy Johnson
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from SE0200119A external-priority patent/SE0200119D0/xx
Priority claimed from SE0201857A external-priority patent/SE0201857D0/xx
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of NO20043370L publication Critical patent/NO20043370L/no

Links

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
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    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
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    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
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    • C07D241/10Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/14Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07F7/081Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring

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  • Health & Medical Sciences (AREA)
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  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
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  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Diabetes (AREA)
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  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hematology (AREA)
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  • Molecular Biology (AREA)
  • Obesity (AREA)
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  • Hospice & Palliative Care (AREA)
NO20043370A 2002-01-16 2004-08-13 N-pyrazinylfenylsulfonamider og deres anvendelse ved behandling av kemokinmedierte sykdommer NO20043370L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
SE0200119A SE0200119D0 (sv) 2002-01-16 2002-01-16 Novel compounds
SE0201857A SE0201857D0 (sv) 2002-06-17 2002-06-17 Novel compounds
PCT/SE2003/000041 WO2003059893A1 (en) 2002-01-16 2003-01-14 N-pyrazinyl-phenylsulphonamides and their use in the treatment of chemokine mediated diseases

Publications (1)

Publication Number Publication Date
NO20043370L true NO20043370L (no) 2004-09-28

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Family Applications (1)

Application Number Title Priority Date Filing Date
NO20043370A NO20043370L (no) 2002-01-16 2004-08-13 N-pyrazinylfenylsulfonamider og deres anvendelse ved behandling av kemokinmedierte sykdommer

Country Status (21)

Country Link
US (2) US7662825B2 (no)
EP (1) EP1467976B1 (no)
JP (1) JP4504021B2 (no)
KR (1) KR20040073566A (no)
CN (1) CN100357275C (no)
AR (1) AR038179A1 (no)
AT (1) ATE534635T1 (no)
AU (1) AU2003201802A1 (no)
BR (1) BR0306922A (no)
CA (1) CA2472204A1 (no)
CO (1) CO5640137A2 (no)
ES (1) ES2375107T3 (no)
IL (1) IL162678A0 (no)
IS (1) IS7348A (no)
MX (1) MXPA04006806A (no)
NO (1) NO20043370L (no)
NZ (1) NZ533750A (no)
PL (1) PL371432A1 (no)
RU (1) RU2312105C9 (no)
TW (1) TWI328007B (no)
WO (1) WO2003059893A1 (no)

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WO2004007472A1 (ja) * 2002-07-10 2004-01-22 Ono Pharmaceutical Co., Ltd. Ccr4アンタゴニストおよびその医薬用途
GB0217431D0 (en) 2002-07-27 2002-09-04 Astrazeneca Ab Novel compounds
US7482355B2 (en) 2002-08-24 2009-01-27 Astrazeneca Ab Pyrimidine derivatives as modulators of chemokine receptor activity
SE0301653D0 (sv) * 2003-06-05 2003-06-05 Astrazeneca Ab Novel compounds
SE0302304D0 (sv) * 2003-08-27 2003-08-27 Astrazeneca Ab Novel compounds
JPWO2005023771A1 (ja) * 2003-09-05 2006-11-02 小野薬品工業株式会社 ケモカインレセプターアンタゴニストおよびその医薬用途
GB0401269D0 (en) * 2004-01-21 2004-02-25 Astrazeneca Ab Compounds
EP1786782B1 (en) 2004-08-12 2010-03-31 Amgen Inc. Bisaryl-sulfonamides
ME01620B (me) 2004-08-28 2014-09-20 Astrazeneca Ab Pirimidin sulfonamidni derivati kao modulatori hemokinskih receptora
TW200800921A (en) * 2005-09-19 2008-01-01 Astrazeneca Ab Novel compounds
EP1956009A1 (en) * 2005-12-02 2008-08-13 Mitsubishi Tanabe Pharma Corporation Aromatic compound
US20090182140A1 (en) * 2005-12-02 2009-07-16 Mitsubishi Tanabe Pharma Corporation Alicyclic Heterocyclic Compound
TW200730512A (en) 2005-12-12 2007-08-16 Astrazeneca Ab Novel compounds
GB0526255D0 (en) 2005-12-22 2006-02-01 Novartis Ag Organic compounds
DK2170848T3 (en) 2007-06-27 2015-01-05 Astrazeneca Ab Pyrazinonderivater and their use to treat lung diseases
EP2276731A1 (en) * 2008-04-09 2011-01-26 Boehringer Ingelheim International GmbH 2-sulfonylamino-4-heteroaryl butyramide antagonists of ccr10
JP5687903B2 (ja) 2008-11-10 2015-03-25 協和発酵キリン株式会社 キヌレニン産生抑制剤
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