NO20031952L - 3-aroylinderivater og deres anvendelse som CB2 reseptoragonister - Google Patents

3-aroylinderivater og deres anvendelse som CB2 reseptoragonister

Info

Publication number: NO20031952L
Authority: NO; Norway
Prior art keywords: aroylin; derivatives; receptor agonists; agonists; receptor
Prior art date: 2000-11-22

Application number

NO20031952A

Other languages

English (en)

Other versions

NO20031952D0 (no

Inventor

Francis Barth

Christian Congy

Carole Guillaumont

Murielle Rinaldi

Fabienne Vasse

Claude Vernhet

Original Assignee

Sanofi Synthelabo

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-11-22

Filing date

2003-04-29

Publication date

2003-07-22

2003-04-29 Application filed by Sanofi Synthelabo filed Critical Sanofi Synthelabo

2003-04-29 Publication of NO20031952D0 publication Critical patent/NO20031952D0/no

2003-07-22 Publication of NO20031952L publication Critical patent/NO20031952L/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/12—Radicals substituted by oxygen atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
- A—HUMAN NECESSITIES
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Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Physical Education & Sports Medicine (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Pulmonology (AREA)
Orthopedic Medicine & Surgery (AREA)
Immunology (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Cardiology (AREA)
Psychiatry (AREA)
Heart & Thoracic Surgery (AREA)
Virology (AREA)
Diabetes (AREA)
Hematology (AREA)
Psychology (AREA)
Hospice & Palliative Care (AREA)
Tropical Medicine & Parasitology (AREA)
Urology & Nephrology (AREA)
Dermatology (AREA)
AIDS & HIV (AREA)
Molecular Biology (AREA)
Ophthalmology & Optometry (AREA)

NO20031952A 2000-11-22 2003-04-29 3-aroylinderivater og deres anvendelse som CB2 reseptoragonister NO20031952L (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR0015158A FR2816938B1 (fr)	2000-11-22	2000-11-22	Derives de 3-aroylindole, leur procede de preparation et les compositions pharmaceutiques en contenant
PCT/FR2001/003665 WO2002042269A1 (fr)	2000-11-22	2001-11-21	Derives de 3-aroylindole et leur utilisation en tant qu'agonistes des recepteurs cb2

Publications (2)

Publication Number	Publication Date
NO20031952D0 NO20031952D0 (no)	2003-04-29
NO20031952L true NO20031952L (no)	2003-07-22

Family

ID=8856819

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20031952A NO20031952L (no)	2000-11-22	2003-04-29	3-aroylinderivater og deres anvendelse som CB2 reseptoragonister

Country Status (32)

Country	Link
US (1)	US6995184B2 (no)
EP (1)	EP1339679B1 (no)
JP (1)	JP4264258B2 (no)
KR (1)	KR20030048161A (no)
CN (1)	CN1234688C (no)
AR (1)	AR033594A1 (no)
AT (1)	ATE301638T1 (no)
AU (1)	AU2002222001A1 (no)
BG (1)	BG107827A (no)
BR (1)	BR0115580A (no)
CA (1)	CA2427444A1 (no)
CZ (1)	CZ20031392A3 (no)
DE (1)	DE60112607T2 (no)
DK (1)	DK1339679T3 (no)
DZ (1)	DZ3443A1 (no)
EA (1)	EA005854B1 (no)
EE (1)	EE200300244A (no)
ES (1)	ES2247201T3 (no)
FR (1)	FR2816938B1 (no)
HR (1)	HRP20030417A2 (no)
HU (1)	HUP0400561A2 (no)
IL (1)	IL155634A0 (no)
IS (1)	IS6802A (no)
MA (1)	MA26959A1 (no)
MX (1)	MXPA03004549A (no)
NO (1)	NO20031952L (no)
NZ (1)	NZ525609A (no)
PL (1)	PL362276A1 (no)
SK (1)	SK6042003A3 (no)
TW (1)	TWI224592B (no)
WO (1)	WO2002042269A1 (no)
ZA (1)	ZA200303728B (no)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
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TW200407110A (en) *	2001-11-23	2004-05-16	Astrazeneca Ab	New use for the treatment of gastroesophageal reflux disease
EP1487436A4 (en)	2002-03-08	2009-06-03	Signal Pharm Inc	POLYTHERAPY FOR TREATING, PREVENTING OR MANAGING PROLIFERATIVE DISORDERS AND CANCERS
JP2006517194A (ja)	2002-06-06	2006-07-20	イッサムリサーチディベロップメントカンパニーオブザヘブリューユニバーシティオブエルサレム	骨成長を調節するための方法、組成物および製造物
AU2003257145B2 (en)	2002-08-02	2008-11-13	Merck Sharp & Dohme Corp.	Substituted furo (2,3-b) pyridine derivatives
FR2843964B1 (fr) *	2002-08-29	2004-10-01	Sanofi Synthelabo	Derives de dioxane-2-alkylcarbamates, leur preparation et leur application en therapeutique
FR2847899B1 (fr) *	2002-11-29	2006-04-28	Sanofi Synthelabo	Derives d'indole-3-carboxamide, leur preparation et leur application en therapeutique
FR2854633B1 (fr) *	2003-05-07	2005-06-24	Sanofi Synthelabo	Derives de piperidinyl-et piperazinyl-alkylcarbamates, leur preparation et leur application en therapeutique
FR2856684B1 (fr) *	2003-06-26	2008-04-11	Sanofi Synthelabo	Derives de diphenylpyridine, leur preparation et leur application en therapeutique
FR2865205B1 (fr) *	2004-01-16	2006-02-24	Sanofi Synthelabo	Derives de type aryloxyalkylcarbamates, leur preparation et leur application en therapeutique
EP1758566A2 (en) *	2004-06-22	2007-03-07	Pharmos Limited	Use of cb2 receptors agonists for the treatment of huntington"s disease
CN101014605A (zh)	2004-07-12	2007-08-08	卡地拉健康护理有限公司	用作大麻素受体调节物的三环吡唑衍生物
US20060025448A1 (en)	2004-07-22	2006-02-02	Cadila Healthcare Limited	Hair growth stimulators
CA2587210A1 (en) *	2004-11-22	2006-06-01	Threshold Pharmaceuticals, Inc.	Tubulin binding anti cancer agents and prodrugs thereof
US7560481B2 (en)	2004-12-21	2009-07-14	Abbott Laboratories	Indoles are cannabinoid receptor ligands
FR2893615B1 (fr) *	2005-11-18	2008-03-07	Sanofi Aventis Sa	Derives de 3-acylindole, leur preparation et leur application en therapeutique
RU2306906C1 (ru) *	2006-04-21	2007-09-27	Федеральное государственное учреждение "Межотраслевой научно-технический комплекс "Микрохирургия глаза" имени академика С.Н. Федорова Федерального агентства по здравоохранению и социальному развитию"	Способ повышения зрительных функций при сублюксации хрусталика в случаях нарушения обмена в системе соединительной ткани
WO2007140439A2 (en)	2006-05-31	2007-12-06	Abbott Laboratories	Compounds as cannabinoid receptor ligands and uses thereof
US8841334B2 (en)	2006-05-31	2014-09-23	Abbvie Inc.	Compounds as cannabinoid receptor ligands and uses thereof
GB0702862D0 (en) *	2007-02-14	2007-03-28	Univ Aberdeen	Therapeutic compounds
EP2142522A1 (en)	2007-03-28	2010-01-13	Abbott Laboratories	1, 3-thiazol-2 (3h) -ylidene compounds as cannabinoid receptor ligands
US7872033B2 (en)	2007-04-17	2011-01-18	Abbott Laboratories	Compounds as cannabinoid receptor ligands
FR2915199B1 (fr) *	2007-04-18	2010-01-22	Sanofi Aventis	Derives de triazolopyridine-carboxamides et triazolopyrimidine-carboxamides, leur preparation et leur application en therapeutique.
MX2009012374A (es) *	2007-05-18	2009-12-01	Abbott Lab	Compuestos novedosos como ligandos del receptor de canabinoides.
US9193713B2 (en)	2007-10-12	2015-11-24	Abbvie Inc.	Compounds as cannabinoid receptor ligands
FR2933697B1 (fr) *	2008-07-11	2010-08-13	Sanofi Aventis	Derives de 1-benzyl-cinnolin-4-(1h)-one substitues, leur preparation et leur application en therapeutique
US8846730B2 (en)	2008-09-08	2014-09-30	Abbvie Inc.	Compounds as cannabinoid receptor ligands
US8859596B2 (en)	2008-09-16	2014-10-14	Abbvie Inc.	Compounds as cannabinoid receptor ligands
PA8854001A1 (es)	2008-12-16	2010-07-27	Abbott Lab	Compuestos novedosos como ligandos de receptores de canabinoides
FR2941696B1 (fr)	2009-02-05	2011-04-15	Sanofi Aventis	Derives d'azaspiranyl-alkylcarbamates d'heterocycles a 5 chainons, leur preparation et leur application en therapeutique
FR2945533B1 (fr)	2009-05-12	2011-05-27	Sanofi Aventis	Derives de cyclopenta°c!pyrrolyl-alkylcarbamates d'heterocycles a 5 chainons, leur preparation et leur application en therapeutique
EP2456428A1 (en)	2009-07-23	2012-05-30	INSERM - Institut National de la Santé et de la Recherche Médicale	Selective cb2 receptor agonists for use in the prevention or treatment of alcoholic liver disease
FR2950055A1 (fr)	2009-09-17	2011-03-18	Sanofi Aventis	Derives de 3-amino-cinnolin-4(1h)-one substitues, leur preparation et leur application en therapeutique
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2000
- 2000-11-22 FR FR0015158A patent/FR2816938B1/fr not_active Expired - Fee Related
2001
- 2001-11-21 AU AU2002222001A patent/AU2002222001A1/en not_active Abandoned
- 2001-11-21 EA EA200300453A patent/EA005854B1/ru not_active IP Right Cessation
- 2001-11-21 EE EEP200300244A patent/EE200300244A/xx unknown
- 2001-11-21 AT AT01997476T patent/ATE301638T1/de not_active IP Right Cessation
- 2001-11-21 CZ CZ20031392A patent/CZ20031392A3/cs unknown
- 2001-11-21 CN CNB018211755A patent/CN1234688C/zh not_active Expired - Fee Related
- 2001-11-21 US US10/416,617 patent/US6995184B2/en not_active Expired - Fee Related
- 2001-11-21 JP JP2002544405A patent/JP4264258B2/ja not_active Expired - Fee Related
- 2001-11-21 HR HR20030417A patent/HRP20030417A2/hr not_active Application Discontinuation
- 2001-11-21 DK DK01997476T patent/DK1339679T3/da active
- 2001-11-21 DE DE60112607T patent/DE60112607T2/de not_active Expired - Lifetime
- 2001-11-21 MX MXPA03004549A patent/MXPA03004549A/es active IP Right Grant
- 2001-11-21 DZ DZ013443A patent/DZ3443A1/fr active
- 2001-11-21 NZ NZ525609A patent/NZ525609A/en unknown
- 2001-11-21 PL PL01362276A patent/PL362276A1/xx not_active Application Discontinuation
- 2001-11-21 KR KR10-2003-7006862A patent/KR20030048161A/ko not_active Withdrawn
- 2001-11-21 BR BR0115580-6A patent/BR0115580A/pt not_active IP Right Cessation
- 2001-11-21 IL IL15563401A patent/IL155634A0/xx unknown
- 2001-11-21 HU HU0400561A patent/HUP0400561A2/hu unknown
- 2001-11-21 CA CA002427444A patent/CA2427444A1/fr not_active Abandoned
- 2001-11-21 ES ES01997476T patent/ES2247201T3/es not_active Expired - Lifetime
- 2001-11-21 AR ARP010105425A patent/AR033594A1/es not_active Application Discontinuation
- 2001-11-21 WO PCT/FR2001/003665 patent/WO2002042269A1/fr not_active Ceased
- 2001-11-21 EP EP01997476A patent/EP1339679B1/fr not_active Expired - Lifetime
- 2001-11-21 SK SK604-2003A patent/SK6042003A3/sk unknown
- 2001-11-22 TW TW090128947A patent/TWI224592B/zh active
2003
- 2003-04-29 NO NO20031952A patent/NO20031952L/no unknown
- 2003-04-30 IS IS6802A patent/IS6802A/is unknown
- 2003-05-13 MA MA27157A patent/MA26959A1/fr unknown
- 2003-05-14 ZA ZA200303728A patent/ZA200303728B/en unknown
- 2003-05-19 BG BG107827A patent/BG107827A/bg unknown

Also Published As

Publication number	Publication date
ES2247201T3 (es)	2006-03-01
PL362276A1 (en)	2004-10-18
DK1339679T3 (da)	2005-12-12
NZ525609A (en)	2004-11-26
EP1339679A1 (fr)	2003-09-03
MA26959A1 (fr)	2004-12-20
BG107827A (bg)	2004-01-30
EA200300453A1 (ru)	2003-10-30
US6995184B2 (en)	2006-02-07
FR2816938A1 (fr)	2002-05-24
ZA200303728B (en)	2004-05-14
EA005854B1 (ru)	2005-06-30
FR2816938B1 (fr)	2003-01-03
DZ3443A1 (fr)	2002-05-30
EP1339679B1 (fr)	2005-08-10
NO20031952D0 (no)	2003-04-29
US20040034090A1 (en)	2004-02-19
AU2002222001A1 (en)	2002-06-03
CN1483023A (zh)	2004-03-17
AR033594A1 (es)	2003-12-26
KR20030048161A (ko)	2003-06-18
CZ20031392A3 (cs)	2003-09-17
CN1234688C (zh)	2006-01-04
EE200300244A (et)	2003-10-15
MXPA03004549A (es)	2004-03-26
JP2004514668A (ja)	2004-05-20
JP4264258B2 (ja)	2009-05-13
DE60112607D1 (de)	2005-09-15
HRP20030417A2 (en)	2003-08-31
DE60112607T2 (de)	2006-06-14
SK6042003A3 (en)	2003-12-02
TWI224592B (en)	2004-12-01
ATE301638T1 (de)	2005-08-15
BR0115580A (pt)	2003-09-09
CA2427444A1 (fr)	2002-05-30
WO2002042269A1 (fr)	2002-05-30
IL155634A0 (en)	2003-11-23
IS6802A (is)	2003-04-30
HUP0400561A2 (hu)	2004-07-28

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