NO20025154L - Imidazopyrimidinderivater og triazolpyrimidinderivater - Google Patents

Imidazopyrimidinderivater og triazolpyrimidinderivater

Info

Publication number: NO20025154L
Authority: NO; Norway
Prior art keywords: derivatives; imidazopyrimidine; triazole pyrimidine; triazole; pyrimidine derivatives
Prior art date: 2000-04-28

Application number

NO20025154A

Other languages

English (en)

Norwegian (no)

Other versions

NO20025154D0 (no

Inventor

Takeshi Yura

Arnel B Concepcion

Gyoonhee Han

Makiko Marumo

Hiroko Katsumata

Norihiro Kawamura

Toshio Kokubo

Hiroshi Komura

Yingfu Li

Timothy Bruno Lowinger

Muneto Mogi

Noriyuki Yamamoto

Nagahiro Yoshida

Scott C Miller

Margaret A Popp

Niko M Redmann

Martha E Rodriguez

William J Scott

Ming Wang

Original Assignee

Bayer Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-04-28

Filing date

2002-10-25

Publication date

2002-10-25

2002-10-25 Application filed by Bayer Ag filed Critical Bayer Ag

2002-10-25 Publication of NO20025154L publication Critical patent/NO20025154L/no

2002-10-25 Publication of NO20025154D0 publication Critical patent/NO20025154D0/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/04—Antipruritics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/04—Drugs for disorders of the muscular or neuromuscular system for myasthenia gravis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/14—Decongestants or antiallergics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/06—Antianaemics

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Immunology (AREA)
Pulmonology (AREA)
Diabetes (AREA)
Hematology (AREA)
Dermatology (AREA)
Neurology (AREA)
Ophthalmology & Optometry (AREA)
Physical Education & Sports Medicine (AREA)
Biomedical Technology (AREA)
Orthopedic Medicine & Surgery (AREA)
Neurosurgery (AREA)
Rheumatology (AREA)
Pain & Pain Management (AREA)
Transplantation (AREA)
Psychiatry (AREA)
Hospice & Palliative Care (AREA)
Obesity (AREA)
Child & Adolescent Psychology (AREA)
Otolaryngology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Plural Heterocyclic Compounds (AREA)

NO20025154A 2000-04-28 2002-10-25 Imidazopyrimidinderivater og triazolpyrimidinderivater NO20025154D0 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP2000128870A JP2001302667A (ja)	2000-04-28	2000-04-28	イミダゾピリミジン誘導体およびトリアゾロピリミジン誘導体
PCT/EP2001/004357 WO2001083485A1 (en)	2000-04-28	2001-04-17	Imidazopyrimidine derivatives and triazolopyrimidine derivatives

Publications (2)

Publication Number	Publication Date
NO20025154L true NO20025154L (no)	2002-10-25
NO20025154D0 NO20025154D0 (no)	2002-10-25

Family

ID=18638240

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20025154A NO20025154D0 (no)	2000-04-28	2002-10-25	Imidazopyrimidinderivater og triazolpyrimidinderivater

Country Status (37)

Country	Link
US (1)	US6911443B2 (es)
EP (1)	EP1278750B1 (es)
JP (2)	JP2001302667A (es)
KR (1)	KR20030009456A (es)
CN (1)	CN1263756C (es)
AR (1)	AR033367A1 (es)
AT (1)	ATE272639T1 (es)
AU (1)	AU783043B2 (es)
BG (1)	BG107166A (es)
BR (1)	BR0110404A (es)
CA (1)	CA2407531A1 (es)
CZ (1)	CZ20023551A3 (es)
DE (1)	DE60104671T2 (es)
DK (1)	DK1278750T3 (es)
DO (1)	DOP2001000151A (es)
EE (1)	EE200200606A (es)
ES (1)	ES2225546T3 (es)
HR (1)	HRP20020943A2 (es)
HU (1)	HUP0300846A2 (es)
IL (1)	IL151919A0 (es)
MA (1)	MA25746A1 (es)
MX (1)	MXPA02010579A (es)
MY (1)	MY141578A (es)
NO (1)	NO20025154D0 (es)
NZ (2)	NZ526221A (es)
PE (1)	PE20011287A1 (es)
PL (1)	PL358106A1 (es)
PT (1)	PT1278750E (es)
RU (1)	RU2306313C2 (es)
SI (1)	SI1278750T1 (es)
SK (1)	SK15332002A3 (es)
SV (1)	SV2001000416A (es)
TR (1)	TR200402300T4 (es)
TW (1)	TWI222974B (es)
UA (1)	UA72615C2 (es)
WO (1)	WO2001083485A1 (es)
ZA (1)	ZA200207676B (es)

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Publication number	Publication date
EP1278750B1 (en)	2004-08-04
ZA200207676B (en)	2003-09-25
IL151919A0 (en)	2003-04-10
NZ522241A (en)	2004-04-30
CN1439009A (zh)	2003-08-27
KR20030009456A (ko)	2003-01-29
PT1278750E (pt)	2004-11-30
AU6220401A (en)	2001-11-12
NO20025154D0 (no)	2002-10-25
ES2225546T3 (es)	2005-03-16
CA2407531A1 (en)	2001-10-25
AR033367A1 (es)	2003-12-17
US20040054179A1 (en)	2004-03-18
HUP0300846A2 (hu)	2003-08-28
BR0110404A (pt)	2003-02-11
DK1278750T3 (da)	2004-11-22
US6911443B2 (en)	2005-06-28
PE20011287A1 (es)	2002-02-27
UA72615C2 (en)	2005-03-15
TR200402300T4 (tr)	2004-12-21
CN1263756C (zh)	2006-07-12
CZ20023551A3 (cs)	2003-01-15
ATE272639T1 (de)	2004-08-15
MA25746A1 (fr)	2003-04-01
AU783043B2 (en)	2005-09-22
NZ526221A (en)	2005-01-28
EP1278750A1 (en)	2003-01-29
JP2001302667A (ja)	2001-10-31
SV2001000416A (es)	2001-07-03
RU2306313C2 (ru)	2007-09-20
JP2003535067A (ja)	2003-11-25
TWI222974B (en)	2004-11-01
MY141578A (en)	2010-05-14
PL358106A1 (en)	2004-08-09
HRP20020943A2 (en)	2005-02-28
DOP2001000151A (es)	2002-05-15
WO2001083485A1 (en)	2001-11-08
EE200200606A (et)	2004-04-15
HK1058362A1 (en)	2004-05-14
MXPA02010579A (es)	2003-05-14
DE60104671D1 (de)	2004-09-09
SI1278750T1 (en)	2005-02-28
DE60104671T2 (de)	2005-12-29
SK15332002A3 (sk)	2003-06-03
BG107166A (bg)	2003-06-30

Publication	Publication Date	Title
NO20025154L (no)	2002-10-25	Imidazopyrimidinderivater og triazolpyrimidinderivater
DK1122244T3 (da)	2004-10-25	Uracilforbindelser og anvendelse deraf
DE60130463D1 (de)	2007-10-25	Pyrimidin-derivate
NO20024355L (no)	2002-11-12	Nukleosidforbindelser og anvendelser derav
NO20025517L (no)	2002-11-18	Triazolderivater
NO20042676L (no)	2004-08-24	3-beta-d-ribofuranolsyltiazolo[4,5-d]pyrimidinnukleosider og anvendelser derav
ATE256123T1 (de)	2003-12-15	Pyrimidonderivate
IS6385A (is)	2002-05-15	Ný notkun og nýjar N-asabísýkló-amíð afleiður
DE60026861D1 (de)	2006-05-11	Purin-derivate
ATE238336T1 (de)	2003-05-15	Purin-derivate
IS6196A (is)	2001-12-11	Púrín afleiður
IL185461A0 (en)	2008-01-06	Pyrimidine compounds and their use
DE60007697D1 (de)	2004-02-19	Triazolderivate
DK1106607T3 (da)	2005-11-07	Uracilforbindelser og anvendelse deraf
NO986174D0 (no)	1998-12-29	Triazinderivater og anvendelse derav
AU2792102A (en)	2002-06-03	Pyrimidine derivatives
DE60022934D1 (de)	2006-02-16	Verstärkerschaltungsanordnung
DK1325010T3 (da)	2005-05-17	Substituerede 3,4-dihydro-pyrimido[1,2-a]pyrimidiner og 3,4-dihydro-pyrazino[1,2-a]pyrimidiner
NO993112D0 (no)	1999-06-23	Katamaran og trimaranski

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